Agonist | Relative Affinity × Efficacy | RAi | ||
---|---|---|---|---|
Null | Operational | |||
Oxotremorine-M | 4.64 (0.67 ± 0.13) | 3.32 (0.52 ± 0.19) | 3.76 (0.58 ± 0.11) | |
Oxotremorine | 3.53 (0.55 ± 0.23) | 1.77 (0.25 ± 0.21) | 2.01 (0.30 ± 0.15) | |
Carbachol | 1.0 (0.0) | 1.0 (0.0) | 1.0 (0.0) | |
(S)-Aceclidine | 1.05 (0.02 ± 0.35) | 0.35 (−0.45 ± 0.19) | 0.44 (−0.35 ± 0.21) | |
McN-A-343 | 0.22a (−0.74 ± 17) | 0.16 (−0.80 ± 0.13) | 0.11 (−0.97 ± 0.33) | |
| 0.10b (−1.02 ± 0.10) |
|
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