TABLE 3

TRPV2 activators and inhibitors

EC50 and IC50 values are given in column with concentration range.


Group

Compound

Compound Number

Conc. R

Species

Reference
M
Activators Probenecid 44 10−5 Rat Bang et al. (2007)
Cannabidiol 45 10−6 Human and rat Qin et al. (2008)
THC 46 10−5 Human and rat Qin et al. (2008)
Cannabidiol 47 10−4 Human and rat Qin et al. (2008)
Inhibitors
SKF96365
48
10−5
Mouse
Juvin et al. (2007)