TABLE 1
Comparison of calculated physical properties for different Y2R antagonists
ID
Molecular Weight
logP
Polar Surface Area
SF-11
447
5.1
44.7
SF-21
471
6.5
75.3
SF-22
491
6.9
75.3
SF-31
415
4.7
86.5
SF-41
341
3.9
60.2
BIIE0246
896
4
219