RGS Protein | CCG-63802 | CCG-63808 | ||
---|---|---|---|---|
IC50 | Hill Slope | IC50 | Hill Slope | |
μM | μM | |||
RGS4 | 9 | −0.9 | 10 | −1.4 |
RGS4c | >400 | −0.4 | >400 | −0.8 |
RGS8 | 112 | −0.6 | 74 | −1.1 |
RGS16 | 42 | −1.4 | 21 | −2.1 |
RGS19 | 20 | −0.6 | 46 | −0.8 |
RGS7 | N.I. | N.I. | N.I. | N.I. |
N.I., no inhibition observed at highest concentration tested (100 μM).