TABLE 2

Plasma protein binding of VU591

Percentage VU591, warfarin (control), and verapamil (control) bound to human or rat serum protein are shown. Data are mean ± S.D. from 2 replicate experiments.

HumanRat
% bound
VU59199.14 ± 0.005698.39 ± 0.0010
Warfarin99.62 ± 0.000299.57 ± 0.0003
Verapamil93.41 ± 0.008897.14 ± 0.0037