Drug | Concentration | Ca2+ Leak | Caffeine-Induced Ca2+ Release |
---|---|---|---|
μM | |||
Anandamide | 4 | 0.020 ± 0.010 | 0.000 ± 0.034 |
Capsaicin | 40 | 0.512 ± 0.039 | 0.798 ± 0.096 |
Capsazepine | 8 | 0.138 ± 0.024 | 0.618 ± 0.142 |
HC 030031 | 80 | 0.709 ± 0.012 | 0.879 ± 0.032 |
Icilin | 40 | 0.791 ± 0.147 | 0.964 ± 0.108 |
(−)Menthol | 1000 | 2.344 ± 0.199 | 1.257 ± 0.015 |
(+)Menthol | 1000 | 0.804 ± 0.113 | 0.941 ± 0.018 |
Piperine | 160 | 0.350 ± 0.009 | 0.779 ± 0.020 |
Pseudocapsaicin | 32 | 0.246 ± 0.063 | 0.703 ± 0.009 |
RTX | 0.8 | 0.120 ± 0.017 | 1.050 ± 0.232 |
HC 030031, 2-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-(4-isopropylphenyl)acetamide.