TABLE 2

Binding affinity constant of the FFA1 agonists

CompoundLogK ± S.E.M. (n)
AMG 8378.44 ± 0.05 (7)a
8.34 ± 0.14 (8)b
AM 16387.87 ± 0.03 (6)a
7.58 ± 0.07 (6)c
AM 81826.04 ± 0.08 (4)c
DHA5.33 ± 0.03 (6)c
5.19 ± 0.14 (6)b
AM 63318.26 ± 0.03 (4)c
  • a From saturation experiments.

  • b From interaction experiments with [3H]AM 1638.

  • c From interaction experiments with [3H]AMG 837.