TABLE 1
Kinase inhibition profile of CTA056
Kinase
IC
50
μ
M
Itk
0.1
Btk
0.4
Etk
3
Src
1.2
Yes
>10
Lyn
>10
Axl
>10
Mer
>10
EGFR
>10
Abl
>10
Mkk1
>10
PDK1
>10
Akt
>10
Erk1
>10