TABLE 3

Absolute mRNA expression of OATP2B1 TSS variants

Tissue/CellAbsolute mRNA Expression (Copies OATP2B1/Copies of 18S)
1b (FL)1d (Short)1e (Short)
Kidney2.06 × 10−57.42 × 10−88.59 × 10−6
Brain1.59 × 10−41.21 × 10−71.45 × 10−7
Placenta1.45 × 10−5ND2.24 × 10−7
Skeletal Muscle2.84 × 10−53.43 × 10−71.32 × 10−6
Caco-25.00 × 10−51.64 × 10−66.45 × 10−4
HeLa9.86 × 10−73.29 × 10−71.35 × 10−7
HepG29.87 × 10−5ND3.85 × 10−5
Huh-78.22 × 10−4ND3.24 × 10−4
  • ND, not detected.