TABLE 4
Log
RA
values from the competitive fit
Compound
Log
RA
GTP coupling
(95% CI)
Log
RA
β
arr2 recruitment
(95% CI)
U69,593
0
0
6′-GNTI
1.2 (0.8 to 1.6)
0.6 (0.4 to 0.9)
Nalbuphine
−1.0 (−1.4 to −0.7)
−0.9 (−1.1 to −0.7)
Nalmefene
0.8 (0.6 to 0.9)
0.3 (0.1 to 0.5)