TABLE 2

Fractional binding of KP-2067 to CaSR cysteine 482 in HEK293 cells expressing human calcium-sensing receptor (n = 4)

KP-2067 (μM)Mean Percent Bound
0ND
8ND
255.3 ± 3.2a
8012.1 ± 4.4a
  • ND, Not detected.

  • a S.E.M.