cAMP Accumulation in A431 Cells | β-Arrestin Recruitment in CHO-β2 Cells | Internalization of GFP-β2 in U2OS Cells | ||||
---|---|---|---|---|---|---|
KA/EC50 | Emax.KA/EC50 | KA/EC50 | Emax.KA/EC50 | KA/EC50 | Emax.KA/EC50 | |
Adrenaline | 44.7 | 4083 | 44.7 | 4507 | 24.5 | 2339 |
C26 | 1.05 | 123 | 0.38 | 45.1 | 0.49 | 59.3 |
Isoprenaline | 8.13 | 832 | 33.9 | 3405 | 5.75 | 570 |