Discovery and development of α7 nicotinic acetylcholine receptor modulators

J Med Chem. 2011 Dec 8;54(23):7943-61. doi: 10.1021/jm2007672. Epub 2011 Sep 29.
No abstract available

Publication types

  • Review

MeSH terms

  • Allosteric Regulation
  • Animals
  • Clinical Trials as Topic
  • Drug Discovery
  • Humans
  • Nicotinic Agonists / chemistry*
  • Nicotinic Agonists / pharmacology
  • Nicotinic Agonists / therapeutic use
  • Nicotinic Antagonists / chemistry*
  • Nicotinic Antagonists / pharmacology
  • Receptors, Nicotinic / physiology*
  • Stereoisomerism
  • alpha7 Nicotinic Acetylcholine Receptor

Substances

  • Chrna7 protein, human
  • Nicotinic Agonists
  • Nicotinic Antagonists
  • Receptors, Nicotinic
  • alpha7 Nicotinic Acetylcholine Receptor