Conformational shifts at the benzodiazepine receptor related to the binding of agonists antagonists and inverse agonists

Life Sci. 1986 Nov 24;39(21):1947-57. doi: 10.1016/0024-3205(86)90318-8.
No abstract available

Publication types

  • Comparative Study

MeSH terms

  • Benzodiazepines / antagonists & inhibitors
  • Benzodiazepines / metabolism*
  • Binding Sites
  • Chemical Phenomena
  • Chemistry
  • Chemistry, Physical
  • Molecular Conformation
  • Protein Conformation
  • Receptors, GABA-A / metabolism*
  • Structure-Activity Relationship

Substances

  • Receptors, GABA-A
  • Benzodiazepines