Design and synthesis of a series of non-peptide high-affinity human corticotropin-releasing factor1 receptor antagonists

J Med Chem. 1996 Oct 25;39(22):4358-60. doi: 10.1021/jm960149e.
No abstract available

MeSH terms

  • Aniline Compounds / chemistry*
  • Corticotropin-Releasing Hormone / metabolism
  • Cyclic AMP / metabolism
  • Drug Compounding / methods*
  • Drug Design*
  • Humans
  • Kinetics
  • Pyrimidines / chemistry*
  • Receptors, Corticotropin-Releasing Hormone / antagonists & inhibitors*
  • Receptors, Corticotropin-Releasing Hormone / metabolism

Substances

  • Aniline Compounds
  • Pyrimidines
  • Receptors, Corticotropin-Releasing Hormone
  • CRF receptor type 1
  • Corticotropin-Releasing Hormone
  • Cyclic AMP