Inhibitors of gamma-aminobutyric acid transport as experimental tools and therapeutic agents

Methods Enzymol. 1998:296:165-75. doi: 10.1016/s0076-6879(98)96013-x.
No abstract available

MeSH terms

  • Animals
  • Brain / metabolism
  • Carrier Proteins / antagonists & inhibitors*
  • Cloning, Molecular
  • Drug Design
  • GABA Antagonists / chemical synthesis*
  • GABA Antagonists / pharmacology
  • GABA Antagonists / therapeutic use
  • GABA Plasma Membrane Transport Proteins
  • Membrane Proteins / antagonists & inhibitors*
  • Membrane Transport Proteins*
  • Molecular Structure
  • Muscimol / analogs & derivatives*
  • Muscimol / chemical synthesis
  • Muscimol / pharmacology
  • Muscimol / therapeutic use
  • Neuroglia / drug effects
  • Neuroglia / metabolism
  • Neurons / drug effects
  • Neurons / metabolism
  • Nipecotic Acids / metabolism
  • Organic Anion Transporters*
  • Proline* / analogs & derivatives*
  • Radioligand Assay
  • Recombinant Proteins / antagonists & inhibitors
  • Tritium
  • gamma-Aminobutyric Acid / analogs & derivatives
  • gamma-Aminobutyric Acid / metabolism

Substances

  • Carrier Proteins
  • GABA Antagonists
  • GABA Plasma Membrane Transport Proteins
  • Membrane Proteins
  • Membrane Transport Proteins
  • Nipecotic Acids
  • Organic Anion Transporters
  • Recombinant Proteins
  • Tritium
  • nipecotic acid
  • Muscimol
  • gamma-Aminobutyric Acid
  • Proline
  • homoproline