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Table representation of search results timeline featuring number of search results per year.

Year Number of Results
1989 3
1993 3
1995 2
1996 1
1999 1
2000 3
2001 2
2003 3
2004 1
2005 3
2006 3
2007 2
2008 3
2009 4
2010 3
2012 1
2013 2
2014 1
2015 3
2016 3
2017 2
2018 1
2019 5
2020 2
2021 1
2024 0

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51 results

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Page 1
Two-step activity-based protein profiling of diacylglycerol lipase.
van Rooden EJ, Kreekel R, Hansen T, Janssen APA, van Esbroeck ACM, den Dulk H, van den Berg RJBHN, Codée JDC, van der Stelt M. van Rooden EJ, et al. Among authors: den dulk h. Org Biomol Chem. 2018 Jul 25;16(29):5250-5253. doi: 10.1039/c8ob01499j. Org Biomol Chem. 2018. PMID: 30004552
ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction.
Baggelaar MP, den Dulk H, Florea BI, Fazio D, Bernabò N, Raspa M, Janssen APA, Scavizzi F, Barboni B, Overkleeft HS, Maccarrone M, van der Stelt M. Baggelaar MP, et al. Among authors: den dulk h. ACS Chem Biol. 2019 Oct 18;14(10):2295-2304. doi: 10.1021/acschembio.9b00640. Epub 2019 Oct 1. ACS Chem Biol. 2019. PMID: 31525885 Free PMC article.
Activity-Based Protein Profiling Identifies α-Ketoamides as Inhibitors for Phospholipase A2 Group XVI.
Zhou J, Mock ED, Martella A, Kantae V, Di X, Burggraaff L, Baggelaar MP, Al-Ayed K, Bakker A, Florea BI, Grimm SH, den Dulk H, Li CT, Mulder L, Overkleeft HS, Hankemeier T, van Westen GJP, van der Stelt M. Zhou J, et al. Among authors: den dulk h. ACS Chem Biol. 2019 Feb 15;14(2):164-169. doi: 10.1021/acschembio.8b00969. Epub 2019 Jan 18. ACS Chem Biol. 2019. PMID: 30620559 Free PMC article.
ABHD2 Inhibitor Identified by Activity-Based Protein Profiling Reduces Acrosome Reaction.
Baggelaar MP, den Dulk H, Florea BI, Fazio D, Perruzza D, Bernabò N, Raspa M, Janssen APA, Scavizzi F, Barboni B, Overkleeft HS, Maccarrone M, van der Stelt M. Baggelaar MP, et al. Among authors: den dulk h. ACS Chem Biol. 2019 Dec 20;14(12):2943. doi: 10.1021/acschembio.9b00824. Epub 2019 Nov 7. ACS Chem Biol. 2019. PMID: 31697462 Free PMC article. No abstract available.
Development of a Retinal-Based Probe for the Profiling of Retinaldehyde Dehydrogenases in Cancer Cells.
Koenders STA, Wijaya LS, Erkelens MN, Bakker AT, van der Noord VE, van Rooden EJ, Burggraaff L, Putter PC, Botter E, Wals K, van den Elst H, den Dulk H, Florea BI, van de Water B, van Westen GJP, Mebius RE, Overkleeft HS, Le Dévédec SE, van der Stelt M. Koenders STA, et al. Among authors: den dulk h. ACS Cent Sci. 2019 Dec 26;5(12):1965-1974. doi: 10.1021/acscentsci.9b01022. Epub 2019 Dec 12. ACS Cent Sci. 2019. PMID: 31893226 Free PMC article.
Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.
van Esbroeck ACM, Janssen APA, Cognetta AB 3rd, Ogasawara D, Shpak G, van der Kroeg M, Kantae V, Baggelaar MP, de Vrij FMS, Deng H, Allarà M, Fezza F, Lin Z, van der Wel T, Soethoudt M, Mock ED, den Dulk H, Baak IL, Florea BI, Hendriks G, De Petrocellis L, Overkleeft HS, Hankemeier T, De Zeeuw CI, Di Marzo V, Maccarrone M, Cravatt BF, Kushner SA, van der Stelt M. van Esbroeck ACM, et al. Among authors: den dulk h. Science. 2017 Jun 9;356(6342):1084-1087. doi: 10.1126/science.aaf7497. Science. 2017. PMID: 28596366 Free PMC article.
Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding.
Deng H, Kooijman S, van den Nieuwendijk AM, Ogasawara D, van der Wel T, van Dalen F, Baggelaar MP, Janssen FJ, van den Berg RJ, den Dulk H, Cravatt BF, Overkleeft HS, Rensen PC, van der Stelt M. Deng H, et al. Among authors: den dulk h. J Med Chem. 2017 Jan 12;60(1):428-440. doi: 10.1021/acs.jmedchem.6b01482. Epub 2016 Dec 19. J Med Chem. 2017. PMID: 27992221
Chemical genetics strategy to profile kinase target engagement reveals role of FES in neutrophil phagocytosis.
van der Wel T, Hilhorst R, den Dulk H, van den Hooven T, Prins NM, Wijnakker JAPM, Florea BI, Lenselink EB, van Westen GJP, Ruijtenbeek R, Overkleeft HS, Kaptein A, Barf T, van der Stelt M. van der Wel T, et al. Among authors: den dulk h. Nat Commun. 2020 Jun 25;11(1):3216. doi: 10.1038/s41467-020-17027-5. Nat Commun. 2020. PMID: 32587248 Free PMC article.
Identification of α,β-Hydrolase Domain Containing Protein 6 as a Diacylglycerol Lipase in Neuro-2a Cells.
van Esbroeck ACM, Kantae V, Di X, van der Wel T, den Dulk H, Stevens AF, Singh S, Bakker AT, Florea BI, Stella N, Overkleeft HS, Hankemeier T, van der Stelt M. van Esbroeck ACM, et al. Among authors: den dulk h. Front Mol Neurosci. 2019 Nov 26;12:286. doi: 10.3389/fnmol.2019.00286. eCollection 2019. Front Mol Neurosci. 2019. PMID: 31849602 Free PMC article.
51 results