Amselamine, a new selective histamine H2-receptor agonist

H van der Goot, JC Eriks, R Leurs… - Bioorganic & Medicinal …, 1994 - Elsevier
The synthesis of amselamine (2-amino-5(2-aminoethyl)-4-methyl-1,3-selenazole), a potent
histamine H 2 -agonist, has been described. At the guinea pig right atrium amselamine …
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New activation model for the histamine H2 receptor, explaining the activity of the different classes of histamine H2 receptor agonists.

JC Eriks, H van der Goot, H Timmerman - Molecular pharmacology, 1993 - ASPET
Recently we developed amthamine [2-amino-5-(2-aminoethyl)-4-methylthiazole]. This cyclic
analogue of dimaprit proved to be the most potent and selective histamine H2 receptor …
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Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative structure-activity relationships of substituted 4-and 5-(2-aminoethyl) thiazoles

JC Eriks, H Van der Goot, GJ Sterk… - Journal of medicinal …, 1992 - ACS Publications
It is well known that both histamine and dimaprit show moderate histamine H2-receptor
agonistic activities on the guinea pig right atrium. Quantum chemical calculations on these two …
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4-or 5-(omega-aminoalkyl) thiazoles and derivatives; new selective H2-receptor agonists.

JC Eriks, GJ Sterk, EM Van der Aar… - Agents and actions …, 1991 - europepmc.org
It is well known that both histamine and dimaprit show moderate H2-receptor agonistic
activity (guinea pig right atrium). Quantum chemical calculations indicated that 2-aminothiazole …
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Studies on the active molecular species of the H2-receptor antagonists cimetidine and mifentidine

…, B Rademaker, K Kramer, JC Eriks… - Journal of medicinal …, 1987 - ACS Publications
“See the Experimental Section for Pharmacological Methodology. 6Ratio activity= antilog (pD2
at pH- pD2 at pH).“Ratio species= relative amount of species at pH/relative amount of …
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Determination of formation constants of copper (II) complexes of Adler medium components with a solid-state copper (II) ionselective electrode

JC Eriks, HD Gaisser, H Van Der Goot… - Pharmaceutisch …, 1983 - Springer
A general method for the determination of overall conditional formation constants of copper(II)
complexes of mycoplasma growth medium (Adler) constituents together with the …
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Abstracts of papers

…, GJ Bijloo, EEJ Haaksma, JC Eriks… - Pharmaceutisch …, 1985 - Springer
In the scope of the latter aspect we have compared the effect of a partial muscarinic receptor
block by propylbenzilylcholine mustard (PrBCM) on guinea pig ileal smooth muscle …
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Abstracts of papers

…, WJ Drijfhout, CJ Grol, BHC Westerink, JC Eriks… - Pharmacy World and …, 1993 - Springer
During the last two decades there has been an increased interest among toxicologists to
explain toxic effects of drugs and other xenobiotin chemicals in terms of molecular mechanisms …
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[CITATION][C] The rearrangement of some 2-phenyl-1, 3-indandiones to (Z)-3-benzylidenephthalides

JC Eriks, H Van der Goot - 1979 - pascal-francis.inist.fr
Keyword (fr) HETEROCYCLE OXYGENE COMPOSE BICYCLIQUE LACTONE REACTION
CHIMIQUE HYDROGENE BROMURE! SUB TRANSPOSITION PREPARATION EFFET …
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Novel Alzheimer disease risk loci and pathways in African American individuals using the African genome resources panel: a meta-analysis

…, B Reisberg, SR Joan, MR John, DR Erik… - JAMA …, 2021 - jamanetwork.com
Importance Compared with non-Hispanic White individuals, African American individuals
from the same community are approximately twice as likely to develop Alzheimer disease. …
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