Table of Contents

Articles

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  Thermal Proteome Profiling Reveals Glutathione Peroxidase 4 as the Target of the Autophagy Inducer Conophylline

  Junya Kakegawa, Satoshi Ohtsuka, Masahiro Yokoyama, Toru Hosoi, Koichiro Ozawa and Takashi Hatanaka

  Molecular Pharmacology September 2021, 100 (3) 181-192; DOI: https://doi.org/10.1124/molpharm.121.000243
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  Selection and Characterization of FD164, a High-Affinity Signal Regulatory Protein α Variant with Balanced Safety and Effectiveness, from a Targeted Epitope Mammalian Cell-Displayed Antibody Library

  Zhihong Wang, Naijing Hu, Xinying Li, Haitao Wang, Caiping Ren, Chunxia Qiao, Guojiang Chen, Jing Wang, Liuzhong Zhou, Jiaguo Wu, Dingmu Zhang, Jiannan Feng, Beifen Shen, Hui Peng and Longlong Luo

  Molecular Pharmacology September 2021, 100 (3) 193-202; DOI: https://doi.org/10.1124/molpharm.120.000202
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  Physiological Temperature Changes Fine-Tune β₂- Adrenergic Receptor-Induced Cytosolic cAMP Accumulation

  Dennis Faro, Ingrid Boekhoff, Thomas Gudermann and Andreas Breit

  Molecular Pharmacology September 2021, 100 (3) 203-216; DOI: https://doi.org/10.1124/molpharm.121.000309
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  Mice Expressing Regulators of G protein Signaling–insensitive Gαo Define Roles of μ Opioid Receptor Gαo and Gαi Subunit Coupling in Inhibition of Presynaptic GABA Release

  Courtney A. Bouchet, Kylie B. McPherson, Ming-hua Li, John R. Traynor and Susan L. Ingram

  Molecular Pharmacology September 2021, 100 (3) 217-223; DOI: https://doi.org/10.1124/molpharm.121.000249
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  Differential Reversible and Irreversible Interactions between Benzbromarone and Human Cytochrome P450s 3A4 and 3A5

  Lloyd Wei Tat Tang, Ravi Kumar Verma, Ren Ping Yong, Xin Li, Lili Wang, Qingsong Lin, Hao Fan and Eric Chun Yong Chan

  Molecular Pharmacology September 2021, 100 (3) 224-236; DOI: https://doi.org/10.1124/molpharm.121.000256
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  High-Throughput Screening of TRPV1 Ligands in the Light of the Bioluminescence Resonance Energy Transfer Technique

  Yann Chappe, Pauline Michel, Alexandre Joushomme, Solène Barbeau, Sandra Pierredon, Luc Baron, André Garenne, Florence Poulletier De Gannes, Annabelle Hurtier, Stanislas Mayer, Isabelle Lagroye, Jean-François Quignard, Thomas Ducret, Vincent Compan, Christelle Franchet and Yann Percherancier

  Molecular Pharmacology September 2021, 100 (3) 237-257; DOI: https://doi.org/10.1124/molpharm.121.000271
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  Open Access

  Functional Interaction between Transient Receptor Potential V4 Channel and Neuronal Calcium Sensor 1 and the Effects of Paclitaxel

  Julio C. Sánchez and Barbara E. Ehrlich

  Molecular Pharmacology September 2021, 100 (3) 258-270; DOI: https://doi.org/10.1124/molpharm.121.000244
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  Ligand-Independent G Protein–Coupled Estrogen Receptor/G Protein–Coupled Receptor 30 Activity: Lack of Receptor-Dependent Effects of G-1 and 17β-Estradiol

  Julia Tutzauer, Ernesto Gonzalez de Valdivia, Karl Swärd, Ioannis Alexandrakis Eilard, Stefan Broselid, Robin Kahn, Björn Olde and L. M. Fredrik Leeb-Lundberg

  Molecular Pharmacology September 2021, 100 (3) 271-282; DOI: https://doi.org/10.1124/molpharm.121.000259
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  The Benzene Hematotoxic and Reactive Metabolite 1,4-Benzoquinone Impairs the Activity of the Histone Methyltransferase SET Domain Containing 2 (SETD2) and Causes Aberrant Histone H3 Lysine 36 Trimethylation (H3K36me3)

  Jérémy Berthelet, Christina Michail, Linh-Chi Bui, Louise Le Coadou, Valentina Sirri, Li Wang, Nicolas Dulphy, Jean-Marie Dupret, Christine Chomienne, Fabien Guidez and Fernando Rodrigues-Lima

  Molecular Pharmacology September 2021, 100 (3) 283-294; DOI: https://doi.org/10.1124/molpharm.121.000303
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  Dynamic Expression of Transient Receptor Potential Vanilloid-3 and Integrated Signaling with Growth Factor Pathways during Lung Epithelial Wound Repair following Wood Smoke Particle and Other Forms of Lung Cell Injury

  Katherine L. Burrell, Nam D. Nguyen, Cassandra E. Deering-Rice, Tosifa A. Memon, Marysol Almestica-Roberts, Emmanuel Rapp, Samantha N. Serna, John G. Lamb and Christopher A. Reilly

  Molecular Pharmacology September 2021, 100 (3) 295-307; DOI: https://doi.org/10.1124/molpharm.121.000280