Table of Contents

Articles

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  The Sulfated Steroids Pregnenolone Sulfate and Dehydroepiandrosterone Sulfate Inhibit the α1β3γ2L GABA_A Receptor by Stabilizing a Novel Nonconducting State

  Spencer R. Pierce, Allison L. Germann, Joe Henry Steinbach and Gustav Akk

  Molecular Pharmacology February 2022, 101 (2) 68-77; DOI: https://doi.org/10.1124/molpharm.121.000385
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  Fluorizoline Blocks the Interaction between Prohibitin-2 and γ-Glutamylcyclotransferase and Induces p21^Waf1/Cip1 Expression in MCF7 Breast Cancer Cells

  Hiroko Takagi, Chiami Moyama, Keiko Taniguchi, Kota Ando, Ryohei Matsuda, Shota Ando, Hiromi Ii, Susumu Kageyama, Akihiro Kawauchi, Nora Chouha, Laurent Désaubry and Susumu Nakata

  Molecular Pharmacology February 2022, 101 (2) 78-86; DOI: https://doi.org/10.1124/molpharm.121.000334
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  Phenylalanine 193 in Extracellular Loop 2 of the β₂-Adrenergic Receptor Coordinates β-Arrestin Interaction

  Michael Ippolito, Francesco De Pascali, Asuka Inoue and Jeffrey L. Benovic

  Molecular Pharmacology February 2022, 101 (2) 87-94; DOI: https://doi.org/10.1124/molpharm.121.000332
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  Thermal Unfolding of the Human Serotonin Transporter: Differential Effect by Stabilizing and Destabilizing Mutations and Cholesterol on Thermodynamic and Kinetic Stability

  Markus Ponleitner, Daniel Szöllősi, Ali El-Kasaby, Florian Koban, Michael Freissmuth and Thomas Stockner

  Molecular Pharmacology February 2022, 101 (2) 95-105; DOI: https://doi.org/10.1124/molpharm.121.000413
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  Lysine Demethylase 6B Regulates Prostate Cancer Cell Proliferation by Controlling c-MYC Expression

  Gökçe Yıldırım-Buharalıoğlu

  Molecular Pharmacology February 2022, 101 (2) 106-119; DOI: https://doi.org/10.1124/molpharm.121.000372