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Molecular Pharmacology

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Research ArticleArticle

Mutations within the Cholecystokinin-B/Gastrin Receptor Ligand ‘Pocket’ Interconvert the Functions of Nonpeptide Agonists and Antagonists

Michael Bläker, Yong Ren, Michelle C. Gordon, Jean E. Hsu, Martin Beinborn and Alan S. Kopin
Molecular Pharmacology November 1998, 54 (5) 857-863; DOI: https://doi.org/10.1124/mol.54.5.857
Michael Bläker
Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Yong Ren
Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Michelle C. Gordon
Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Jean E. Hsu
Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Martin Beinborn
Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Alan S. Kopin
Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Article Information

vol. 54 no. 5 857-863
DOI 
https://doi.org/10.1124/mol.54.5.857
PubMed 
9804620

Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0026-895X
Online ISSN 
1521-0111
History 
  • Received January 20, 1998
  • Accepted July 31, 1998
  • Published online November 1, 1998.

Copyright & Usage 
The American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. Michael Bläker,
  2. Yong Ren,
  3. Michelle C. Gordon,
  4. Jean E. Hsu,
  5. Martin Beinborn, and
  6. Alan S. Kopin
  1. Division of Gastroenterology and GRASP Digestive Disease Center, Tupper Research Institute, New England Medical Center, Tufts University School of Medicine, Boston, Massachusetts 02111
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Molecular Pharmacology: 54 (5)
Molecular Pharmacology
Vol. 54, Issue 5
1 Nov 1998
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Research ArticleArticle

Mutations within the Cholecystokinin-B/Gastrin Receptor Ligand ‘Pocket’ Interconvert the Functions of Nonpeptide Agonists and Antagonists

Michael Bläker, Yong Ren, Michelle C. Gordon, Jean E. Hsu, Martin Beinborn and Alan S. Kopin
Molecular Pharmacology November 1, 1998, 54 (5) 857-863; DOI: https://doi.org/10.1124/mol.54.5.857

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Research ArticleArticle

Mutations within the Cholecystokinin-B/Gastrin Receptor Ligand ‘Pocket’ Interconvert the Functions of Nonpeptide Agonists and Antagonists

Michael Bläker, Yong Ren, Michelle C. Gordon, Jean E. Hsu, Martin Beinborn and Alan S. Kopin
Molecular Pharmacology November 1, 1998, 54 (5) 857-863; DOI: https://doi.org/10.1124/mol.54.5.857
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