Table of Contents

Articles

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  Regulation of the MDR1 Gene by Transcriptional Repressors Selected Using Peptide Combinatorial Libraries

  Victor V. Bartsevich and R. L. Juliano

  Molecular Pharmacology July 2000, 58 (1) 1-10; DOI: https://doi.org/10.1124/mol.58.1.1
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  Subunit-Specific Action of an Anticonvulsant Thiobutyrolactone on Recombinant Glycine Receptors Involves a Residue in the M2 Membrane-Spanning Region

  Joe Henry Steinbach, John Bracamontes, Li Yu, Pengnian Zhang and Douglas F. Covey

  Molecular Pharmacology July 2000, 58 (1) 11-17; DOI: https://doi.org/10.1124/mol.58.1.11
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  Sarco-Endoplasmic ATPase Blocker 2,5-Di(tert-butyl)-1,4-benzohydroquinone Inhibits N-, P-, and Q- but Not T-, L-, or R-Type Calcium Currents in Central and Peripheral Neurons

  Frédérique Scamps, Stéphan Vigues, Sophie Restituito, Brice Campo, Anne Roig, Pierre Charnet and Jean Valmier

  Molecular Pharmacology July 2000, 58 (1) 18-26; DOI: https://doi.org/10.1124/mol.58.1.18
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  Anticancer Derivative of Butyric Acid (Pivalyloxymethyl Butyrate) Specifically Potentiates the Cytotoxicity of Doxorubicin and Daunorubicin through the Suppression of Microsomal Glycosidic Activity

  Nozomi Niitsu, Takashi Kasukabe, Akihiro Yokoyama, Junko Okabe-Kado, Yuri Yamamoto-Yamaguchi, Masanori Umeda and Yoshio Honma

  Molecular Pharmacology July 2000, 58 (1) 27-36; DOI: https://doi.org/10.1124/mol.58.1.27
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  Functional Analysis of a Tryptophan-Less P-glycoprotein: A Tool for Tryptophan Insertion and Fluorescence Spectroscopy

  Tony Kwan, Helen Loughrey, Martine Brault, Samantha Gruenheid, Ina L. Urbatsch, Alan E. Senior and Philippe Gros

  Molecular Pharmacology July 2000, 58 (1) 37-47; DOI: https://doi.org/10.1124/mol.58.1.37
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  Two-Stage Glucocorticoid Induction of CYP3A23through Both the Glucocorticoid and Pregnane X Receptors

  Janice M. Huss and Charles B. Kasper

  Molecular Pharmacology July 2000, 58 (1) 48-57; DOI: https://doi.org/10.1124/mol.58.1.48
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  Mechanism of Action of the Potent Sodium-Retaining Steroid 11,19-Oxidoprogesterone

  Mario D. Galigniana, Guillermo P. Vicent, Graciela Piwien-Pilipuk, Gerardo Burton and Carlos P. Lantos

  Molecular Pharmacology July 2000, 58 (1) 58-70; DOI: https://doi.org/10.1124/mol.58.1.58
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  Acetyl-Boswellic Acids Are Novel Catalytic Inhibitors of Human Topoisomerases I and IIα

  Tatiana Syrovets, Berthold Büchele, Erk Gedig, Joseph R. Slupsky and Thomas Simmet

  Molecular Pharmacology July 2000, 58 (1) 71-81; DOI: https://doi.org/10.1124/mol.58.1.71
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  Brilliant Blue G Selectively Blocks ATP-Gated Rat P2X₇ Receptors

  Lin-Hua Jiang, Amanda B. Mackenzie, R. Alan North and Annmarie Surprenant

  Molecular Pharmacology July 2000, 58 (1) 82-88; DOI: https://doi.org/10.1124/mol.58.1.82
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  Characterization of the UDP-Glucuronosyltransferase 1A Locus in Lagomorphs: Evidence for Duplication of theUGT1A6 Gene

  Qing Li, Greg Lamb and Robert H. Tukey

  Molecular Pharmacology July 2000, 58 (1) 89-97; DOI: https://doi.org/10.1124/mol.58.1.89
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  Anticonvulsants But Not General Anesthetics Have Differential Blocking Effects on Different T-Type Current Variants

  Slobodan M. Todorovic, Edward Perez-Reyes and Christopher J. Lingle

  Molecular Pharmacology July 2000, 58 (1) 98-108; DOI: https://doi.org/10.1124/mol.58.1.98
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  Subtype-Selective Inhibition of Neuronal Nicotinic Acetylcholine Receptors by Cocaine Is Determined by the α4 and β4 Subunits

  Michael M. Francis, Raymond W. Vazquez, Roger L. Papke and Robert E. Oswald

  Molecular Pharmacology July 2000, 58 (1) 109-119; DOI: https://doi.org/10.1124/mol.58.1.109
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  Inhibition of Cell Surface Expression by Mutant Receptors Demonstrates that D2 Dopamine Receptors Exist as Oligomers in the Cell

  Samuel P. Lee, Brian F. O'Dowd, Gordon Y.K. Ng, George Varghese, Huda Akil, Alfred Mansour, Tuan Nguyen and Susan R. George

  Molecular Pharmacology July 2000, 58 (1) 120-128; DOI: https://doi.org/10.1124/mol.58.1.120
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  Molecular Basis for Proton Regulation of Glycine Transport by Glycine Transporter Subtype 1b

  Karin R. Aubrey, Ann D. Mitrovic and Robert J. Vandenberg

  Molecular Pharmacology July 2000, 58 (1) 129-135; DOI: https://doi.org/10.1124/mol.58.1.129
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  Pharmacological Properties of 5-Hydroxytryptamine₄Receptor Antagonists on Constitutively Active Wild-Type and Mutated Receptors

  Sylvie Claeysen, Michèle Sebben, Carine Bécamel, Richard M. Eglen, Robin D. Clark, Joël Bockaert and Aline Dumuis

  Molecular Pharmacology July 2000, 58 (1) 136-144; DOI: https://doi.org/10.1124/mol.58.1.136
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  Elevation of Intracellular cAMP Inhibits Growth Factor-Mediated Matrix Metalloproteinase-9 Induction and Keratinocyte Migration

  Lisa J. McCawley, Shunan Li, Mario Benavidez, Jennifer Halbleib, Elizabeth V. Wattenberg and Laurie G. Hudson

  Molecular Pharmacology July 2000, 58 (1) 145-151; DOI: https://doi.org/10.1124/mol.58.1.145
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  Activation of c-Ha-ras by Benzo(a)pyrene in Vascular Smooth Muscle Cells Involves Redox Stress and Aryl Hydrocarbon Receptor

  J. Kevin Kerzee and Kenneth S. Ramos

  Molecular Pharmacology July 2000, 58 (1) 152-158; DOI: https://doi.org/10.1124/mol.58.1.152
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  Overexpression of Dynamin Is Induced by Chronic Stimulation of μ- but Not δ-Opioid Receptors: Relationships with μ-Related Morphine Dependence

  Florence Noble, Maria Szücs, Brigitte Kieffer and Bernard P. Roques

  Molecular Pharmacology July 2000, 58 (1) 159-166; DOI: https://doi.org/10.1124/mol.58.1.159
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  Cellular Response to a Glutathione S-Transferase P1-1 Activated Prodrug

  Lilliam A. Rosario, Miechelle L. O'Brien, Colin J. Henderson, C. Roland Wolf and Kenneth D. Tew

  Molecular Pharmacology July 2000, 58 (1) 167-174; DOI: https://doi.org/10.1124/mol.58.1.167
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  Scanning Mutagenesis Identifies Amino Acid Side Chains in Transmembrane Domain 5 of the M₁ Muscarinic Receptor that Participate in Binding the Acetyl Methyl Group of Acetylcholine

  Karen Allman, Karen M. Page, Carol A.M. Curtis and Edward C. Hulme

  Molecular Pharmacology July 2000, 58 (1) 175-184; DOI: https://doi.org/10.1124/mol.58.1.175
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  Differences in the Formation of PPARα-RXR/acoPPRE Complexes between Responsive and Nonresponsive Species upon Fibrate Administration

  Cristina Rodríguez, Véronique Noé, Agatha Cabrero, Carlos J. Ciudad and Juan C. Laguna

  Molecular Pharmacology July 2000, 58 (1) 185-193; DOI: https://doi.org/10.1124/mol.58.1.185
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  Allosteric Interactions of Staurosporine and Other Indolocarbazoles withN-[methyl-³H]Scopolamine and Acetylcholine at Muscarinic Receptor Subtypes: Identification of a Second Allosteric Site

  Sebastian Lazareno, Angela Popham and Nigel J. M. Birdsall

  Molecular Pharmacology July 2000, 58 (1) 194-207; DOI: https://doi.org/10.1124/mol.58.1.194
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  Induction of Metabolism-Dependent and -Independent Neutrophil Apoptosis by Clozapine

  Dominic P. Williams, Munir Pirmohamed, Dean J. Naisbitt, Jack P. Uetrecht and Brian K. Park

  Molecular Pharmacology July 2000, 58 (1) 207-216; DOI: https://doi.org/10.1124/mol.58.1.207
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  Molecular Characterization of the Melanin-Concentrating Hormone/Receptor Complex: Identification of Critical Residues Involved in Binding and Activation

  Douglas Macdonald, Nicholas Murgolo, Rumin Zhang, James P. Durkin, Xiaorui Yao, Catherine D. Strader and Michael P. Graziano

  Molecular Pharmacology July 2000, 58 (1) 217-225; DOI: https://doi.org/10.1124/mol.58.1.217
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  A Gα_s Carboxyl-Terminal Peptide Prevents G_s Activation by the A_2A Adenosine Receptor

  Maria R. Mazzoni, Simone Taddei, Laura Giusti, Paolo Rovero, Claudia Galoppini, Annamaria D'Ursi, Stefania Albrizio, Antonio Triolo, Ettore Novellino, Giovanni Greco, Antonio Lucacchini and Heidi E. Hamm

  Molecular Pharmacology July 2000, 58 (1) 226-236; DOI: https://doi.org/10.1124/mol.58.1.226
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  Activation of p55 Tumor Necrosis Factor-α Receptor-1 Coupled to Tumor Necrosis Factor Receptor-Associated Factor 2 Stimulates Intercellular Adhesion Molecule-1 Expression by Modulating a Thapsigargin-Sensitive Pathway in Human Tracheal Smooth Muscle Cells

  Yassine Amrani, Aili L. Lazaar, Rebecca Hoffman, Kunjalata Amin, Samir Ousmer and Reynold A. Panettieri

  Molecular Pharmacology July 2000, 58 (1) 237-245; DOI: https://doi.org/10.1124/mol.58.1.237