Table of Contents

Articles

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  The Steroid 17α-Acetoxy-6-dimethylaminomethyl-21-fluoro-3-ethoxy-pregna-3,5-dien-20-one (SC17599) Is a Selective μ-Opioid Agonist: Implications for the μ-Opioid Pharmacophore

  Iain J. McFadyen, Hani Houshyar, Lee-Yuan Liu-Chen, James H. Woods and John R. Traynor

  Molecular Pharmacology October 2000, 58 (4) 669-676; DOI: https://doi.org/10.1124/mol.58.4.669
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  The Dopamine D3 Receptor Interacts with Itself and the Truncated D3 Splice Variant D3nf: D3-D3nf Interaction Causes Mislocalization of D3 Receptors

  Kelly D. Karpa, Ridwan Lin, Nadine Kabbani and Robert Levenson

  Molecular Pharmacology October 2000, 58 (4) 677-683; DOI: https://doi.org/10.1124/mol.58.4.677
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  A Single Amino Acid Mutation of Ala-773 in the Mineralocorticoid Receptor Confers Agonist Properties to 11β-Substituted Spirolactones

  Gilles Auzou, Jérôme Fagart, Anny Souque, Chantal Hellal-Lévy, Jean-Marie Wurtz, Dino Moras and Marie-Edith Rafestin-Oblin

  Molecular Pharmacology October 2000, 58 (4) 684-691; DOI: https://doi.org/10.1124/mol.58.4.684
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  An Analysis of the Variations in Potency of Grayanotoxin Analogs in Modifying Frog Sodium Channels of Differing Subtypes

  Masuhide Yakehiro, Tsunetsugu Yuki, Kaoru Yamaoka, Toshiaki Furue, Yasuo Mori, Keiji Imoto and Issei Seyama

  Molecular Pharmacology October 2000, 58 (4) 692-700; DOI: https://doi.org/10.1124/mol.58.4.692
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  Cyclosporin A Selectively Inhibits Mitogen-Induced Cyclooxygenase-2 Gene Transcription in Vascular Smooth Muscle Cells

  Aaron M. Robida, Kaiming Xu, Michelle L. Ellington and T. J. Murphy

  Molecular Pharmacology October 2000, 58 (4) 701-708; DOI: https://doi.org/10.1124/mol.58.4.701
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  Cellular Resistance to the Antitumor DNA Topoisomerase II Inhibitor S16020-2: Importance of the N-[2(Dimethylamino)ethyl]carbamoyl Side Chain

  Sandrine Le Mée, Françoise Chaminade, Charlotte Delaporte, Judith Markovits, Jean-Marie Saucier and Alain Jacquemin-Sablon

  Molecular Pharmacology October 2000, 58 (4) 709-718; DOI: https://doi.org/10.1124/mol.58.4.709
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  RGS3 Is a GTPase-Activating Protein for G_iα and G_qα and a Potent Inhibitor of Signaling by GTPase-Deficient Forms of G_qα and G_11α

  Astrid Scheschonka, Carmen W. Dessauer, Srikumar Sinnarajah, Peter Chidiac, Chong-Shan Shi and John H. Kehrl

  Molecular Pharmacology October 2000, 58 (4) 719-728; DOI: https://doi.org/10.1124/mol.58.4.719
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  Photo-Induced Inactivation of Protein Kinase Cα by Dequalinium Inhibits Motility of Murine Melanoma Cells

  Regina M. Sullivan, Michael Stone, John F. Marshall, Florian Uberall and Susan A. Rotenberg

  Molecular Pharmacology October 2000, 58 (4) 729-737; DOI: https://doi.org/10.1124/mol.58.4.729
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  Organic Vanadium Chelators Potentiate Vanadium-Evoked Glucose Metabolism In Vitro and In Vivo: Establishing Criteria for Optimal Chelators

  Itzhak Goldwaser, Sun Qian, Eytan Gershonov, Mati Fridkin and Yoram Shechter

  Molecular Pharmacology October 2000, 58 (4) 738-746; DOI: https://doi.org/10.1124/mol.58.4.738
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  Duplications and Defects in the CYP2A6 Gene: Identification, Genotyping, and In Vivo Effects on Smoking

  Yushu Rao, Ewa Hoffmann, Mohammad Zia, Laurent Bodin, Marilyn Zeman, Edward M. Sellers and Rachel F. Tyndale

  Molecular Pharmacology October 2000, 58 (4) 747-755; DOI: https://doi.org/10.1124/mol.58.4.747
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  Characterization of the Interaction of Zopiclone with γ-Aminobutyric Acid Type A Receptors

  Martin Davies, J. Glen Newell, Jason M. C. Derry, Ian L. Martin and Susan M. J. Dunn

  Molecular Pharmacology October 2000, 58 (4) 756-762; DOI: https://doi.org/10.1124/mol.58.4.756
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  Glycine Receptor β Subunits Play a Critical Role in Potentiation of Glycine Responses by ICS-205,930

  Stephane Supplisson and Dominique Chesnoy-Marchais

  Molecular Pharmacology October 2000, 58 (4) 763-770; DOI: https://doi.org/10.1124/mol.58.4.763
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  Adenosine A_2A Receptors are Colocalized with and Activate G_olf in Rat Striatum

  Björn Kull, Per Svenningsson and Bertil B. Fredholm

  Molecular Pharmacology October 2000, 58 (4) 771-777; DOI: https://doi.org/10.1124/mol.58.4.771
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  Rapid Relief of Block by Mecamylamine of Neuronal Nicotinic Acetylcholine Receptors of Rat Chromaffin Cells In Vitro: An Electrophysiological and Modeling Study

  Rashid A. Giniatullin, Elena M. Sokolova, Silvia Di Angelantonio, Andrei Skorinkin, Maria V. Talantova and Andrea Nistri

  Molecular Pharmacology October 2000, 58 (4) 778-787; DOI: https://doi.org/10.1124/mol.58.4.778
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  Structure-Activity Relationships for Growth Inhibition and Induction of Apoptosis by 4-Hydroxy-2-nonenal in Raw 264.7 Cells

  Robin L. Haynes, Luke Szweda, Kerry Pickin, Mark E. Welker and Alan J. Townsend

  Molecular Pharmacology October 2000, 58 (4) 788-794; DOI: https://doi.org/10.1124/mol.58.4.788
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  Mechanisms of Agonist-Induced Down-Regulation of the Human κ-Opioid Receptor: Internalization Is Required for Down-Regulation

  Jian-Guo Li, Jeffrey L. Benovic and Lee-Yuan Liu-Chen

  Molecular Pharmacology October 2000, 58 (4) 795-801; DOI: https://doi.org/10.1124/mol.58.4.795
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  Effects of the Potent Ampakine CX614 on Hippocampal and Recombinant AMPA Receptors: Interactions with Cyclothiazide and GYKI 52466

  Amy C. Arai, Markus Kessler, Gary Rogers and Gary Lynch

  Molecular Pharmacology October 2000, 58 (4) 802-813; DOI: https://doi.org/10.1124/mol.58.4.802
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  The CB₁ Cannabinoid Receptor Is Coupled to the Activation of c-Jun N-Terminal Kinase

  Daniel Rueda, Ismael Galve-Roperh, Amador Haro and Manuel Guzmán

  Molecular Pharmacology October 2000, 58 (4) 814-820; DOI: https://doi.org/10.1124/mol.58.4.814
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  Transcriptional Down-Regulation of the Human α2C-Adrenergic Receptor by cAMP

  Stéphane Schaak, Cécile Cayla, Anastasios Lymperopoulos, Christodoulos Flordellis, Daniel Cussac, Colette Denis and Hervé Paris

  Molecular Pharmacology October 2000, 58 (4) 821-827; DOI: https://doi.org/10.1124/mol.58.4.821
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  Human Bradykinin B₂ Receptor Is Activated by Kallikrein and Other Serine Proteases

  Claudie Hecquet, Fulong Tan, Branislav M. Marcic and Ervin G. Erdös

  Molecular Pharmacology October 2000, 58 (4) 828-836; DOI: https://doi.org/10.1124/mol.58.4.828
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  15-Deoxy-Δ^12,14-prostaglandin J₂Induces G₁ Arrest and Differentiation Marker Expression in Vascular Smooth Muscle Cells

  Yoshikazu Miwa, Toshiyuki Sasaguri, Hiroyasu Inoue, Yoji Taba, Akio Ishida and Takeo Abumiya

  Molecular Pharmacology October 2000, 58 (4) 837-844; DOI: https://doi.org/10.1124/mol.58.4.837
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  Aryl Hydrocarbon Receptor Is Required for p300-Mediated Induction of DNA Synthesis by Adenovirus E1A

  Masahiro Tohkin, Morio Fukuhara, Guillermo Elizondo, Shuhei Tomita and Frank J. Gonzalez

  Molecular Pharmacology October 2000, 58 (4) 845-851; DOI: https://doi.org/10.1124/mol.58.4.845
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  Interaction of Methoxychlor and Related Compounds with Estrogen Receptor α and β, and Androgen Receptor: Structure-Activity Studies

  Kevin W. Gaido, Susan C. Maness, Donald P. McDonnell, Shangara S. Dehal, David Kupfer and Stephen Safe

  Molecular Pharmacology October 2000, 58 (4) 852-858; DOI: https://doi.org/10.1124/mol.58.4.852