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Molecular Pharmacology

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Table of Contents

November 01, 2000; Volume 58,Issue 5

Articles

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    Differential Modes of Agonist Binding to 5-Hydroxytryptamine2A Serotonin Receptors Revealed by Mutation and Molecular Modeling of Conserved Residues in Transmembrane Region 5
    David A. Shapiro, Kurt Kristiansen, Wesley K. Kroeze and Bryan L. Roth
    Molecular Pharmacology November 2000, 58 (5) 877-886; DOI: https://doi.org/10.1124/mol.58.5.877
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    Spontaneous Activation of β2- but Not β1-Adrenoceptors Expressed in Cardiac Myocytes from β1β2 Double Knockout Mice
    Ying-Ying Zhou, Dongmei Yang, Wei-Zhong Zhu, Sheng-Jun Zhang, Ding-Ji Wang, Dan K. Rohrer, Eric Devic, Brian K. Kobilka, Edward G. Lakatta, Heping Cheng and Rui-Ping Xiao
    Molecular Pharmacology November 2000, 58 (5) 887-894; DOI: https://doi.org/10.1124/mol.58.5.887
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    Functional Comparisons of the Lysophosphatidic Acid Receptors, LPA1/VZG-1/EDG-2, LPA2/EDG-4, and LPA3/EDG-7 in Neuronal Cell Lines Using a Retrovirus Expression System
    Isao Ishii, James J. A. Contos, Nobuyuki Fukushima and Jerold Chun
    Molecular Pharmacology November 2000, 58 (5) 895-902; DOI: https://doi.org/10.1124/mol.58.5.895
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    Cyclic AMP and Protein Kinase A Stimulate Cdc42: Role of A2 Adenosine Receptors in Human Mast Cells
    Igor Feoktistov, Anna E. Goldstein and Italo Biaggioni
    Molecular Pharmacology November 2000, 58 (5) 903-910; DOI: https://doi.org/10.1124/mol.58.5.903
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    Structural Insights into the Amino-Terminus of the Secretin Receptor: I. Status of Cysteine and Cystine Residues
    Yan W. Asmann, Maoqing Dong, Subhas Ganguli, Elizabeth M. Hadac and Laurence J. Miller
    Molecular Pharmacology November 2000, 58 (5) 911-919; DOI: https://doi.org/10.1124/mol.58.5.911
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    Oxaliplatin-Induced Damage of Cellular DNA
    Jan M. Woynarowski, Sandrine Faivre, Maryanne C.S. Herzig, Brenda Arnett, William G. Chapman, Alex V. Trevino, Eric Raymond, Stephen G. Chaney, Alexandra Vaisman, Maria Varchenko and Paul E. Juniewicz
    Molecular Pharmacology November 2000, 58 (5) 920-927; DOI: https://doi.org/10.1124/mol.58.5.920
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    Cyclosaligenyl-2′,3′-didehydro-2′,3′-dideoxythymidine Monophosphate: Efficient Intracellular Delivery of d4TMP
    Jan Balzarini, Stefano Aquaro, Tina Knispel, Chiara Rampazzo, Vera Bianchi, Carlo-Federico Perno, Erik De Clercq and Chris Meier
    Molecular Pharmacology November 2000, 58 (5) 928-935; DOI: https://doi.org/10.1124/mol.58.5.928
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    Characterization of Calcium Signaling by Purinergic Receptor-Channels Expressed in Excitable Cells
    Taka-aki Koshimizu, Fredrick Van Goor, Melanija Tomić, Anderson On-Lam Wong, Akito Tanoue, Gozoh Tsujimoto and Stanko S. Stojilkovic
    Molecular Pharmacology November 2000, 58 (5) 936-945; DOI: https://doi.org/10.1124/mol.58.5.936
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    Evidence That Gαq-Coupled Receptor-Induced Interleukin-6 mRNA in Vascular Smooth Muscle Cells Involves the Nuclear Factor of Activated T Cells
    Karen L. Abbott, James R. Loss, Aaron M. Robida and T. J. Murphy
    Molecular Pharmacology November 2000, 58 (5) 946-953; DOI: https://doi.org/10.1124/mol.58.5.946
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    Molecular Analysis of β2-Adrenoceptor Coupling to Gs-, Gi-, and Gq-Proteins
    Katharina Wenzel-Seifert and Roland Seifert
    Molecular Pharmacology November 2000, 58 (5) 954-966; DOI: https://doi.org/10.1124/mol.58.5.954
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    Structure-Related Inhibition of Calmodulin-Dependent Neuronal Nitric-Oxide Synthase Activity by Melatonin and Synthetic Kynurenines
    Josefa León, Manuel Macías, Germaine Escames, Encarna Camacho, Huda Khaldy, Miguel Martín, Antonio Espinosa, Miguel A. Gallo and Darío Acuña-Castroviejo
    Molecular Pharmacology November 2000, 58 (5) 967-975; DOI: https://doi.org/10.1124/mol.58.5.967
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    Fibronectin-Mediated Hepatocyte Shape Change Reprograms Cytochrome P450 2C11 Gene Expression via an Integrin-Signaled Induction of Ribonuclease Activity
    Conrad P. Hodgkinson, Matthew C. Wright and Alan J. Paine
    Molecular Pharmacology November 2000, 58 (5) 976-981; DOI: https://doi.org/10.1124/mol.58.5.976
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    Analysis of the Interaction between the HIV-Inactivating Protein Cyanovirin-N and Soluble Forms of the Envelope Glycoproteins gp120 and gp41
    Barry R. O'Keefe, Shilpa R. Shenoy, Dong Xie, Wentao Zhang, Jeffrey M. Muschik, Michael J. Currens, Irwin Chaiken and Michael R. Boyd
    Molecular Pharmacology November 2000, 58 (5) 982-992; DOI: https://doi.org/10.1124/mol.58.5.982
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    The Amino Terminus of Gαz is Required for Receptor Recognition, Whereas its α4/β6 Loop Is Essential for Inhibition of Adenylyl Cyclase
    Maurice K.C. Ho and Yung H. Wong
    Molecular Pharmacology November 2000, 58 (5) 993-1000; DOI: https://doi.org/10.1124/mol.58.5.993
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    G1 Phase-Dependent Expression of Bcl-2 mRNA and Protein Correlates with Chemoresistance of Human Cancer Cells
    Gui Gao and Q. Ping Dou
    Molecular Pharmacology November 2000, 58 (5) 1001-1010; DOI: https://doi.org/10.1124/mol.58.5.1001
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    Overexpression of Type 7 Adenylyl Cyclase in the Mouse Brain Enhances Acute and Chronic Actions of Morphine
    Masami Yoshimura, Peter H. Wu, Paula L. Hoffman and Boris Tabakoff
    Molecular Pharmacology November 2000, 58 (5) 1011-1016; DOI: https://doi.org/10.1124/mol.58.5.1011
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    The Essential Role of Phosphatidylinositol 3-Kinase and of p38 Mitogen-Activated Protein Kinase Activation in the Antioxidant Response Element-Mediated rGSTA2 Induction by Decreased Glutathione in H4IIE Hepatoma Cells
    Keon Wook Kang, Ji Hwa Ryu and Sang Geon Kim
    Molecular Pharmacology November 2000, 58 (5) 1017-1025; DOI: https://doi.org/10.1124/mol.58.5.1017
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    The Inhibitory Potency and Selectivity of Arginine Substrate Site Nitric-Oxide Synthase Inhibitors Is Solely Determined by Their Affinity toward the Different Isoenzymes
    Rainer Boer, Wolf-Rüdiger Ulrich, Thomas Klein, Berit Mirau, Sabine Haas and Ilka Baur
    Molecular Pharmacology November 2000, 58 (5) 1026-1034; DOI: https://doi.org/10.1124/mol.58.5.1026
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    Creation of a Selective Antagonist and Agonist of the Rat VPAC1 Receptor Using a Combinatorial Approach with Vasoactive Intestinal Peptide 6–23 as Template
    Jeppe Wegener Tams, Rikke Malene Jørgensen, Arne Holm and Jan Fahrenkrug
    Molecular Pharmacology November 2000, 58 (5) 1035-1041; DOI: https://doi.org/10.1124/mol.58.5.1035
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    Inverse Agonism and Constitutive Activity as Functional Correlates of Serotonin h5-HT1B Receptor/G-Protein Stoichiometry
    Adrian Newman-Tancredi, Valérie Audinot, Celia Moreira, Laurence Verrièle and Mark J. Millan
    Molecular Pharmacology November 2000, 58 (5) 1042-1049; DOI: https://doi.org/10.1124/mol.58.5.1042
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    Identification of G Protein-Coupled Receptor Kinase 2 Phosphorylation Sites Responsible for Agonist-Stimulated δ-Opioid Receptor Phosphorylation
    Jun Guo, Yalan Wu, Wenbo Zhang, Jing Zhao, Lakshmi A. Devi, Gang Pei and Lan Ma
    Molecular Pharmacology November 2000, 58 (5) 1050-1056; DOI: https://doi.org/10.1124/mol.58.5.1050
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    Regulation of Cell Proliferation, Gene Expression, Production of Cytokines, and Cell Cycle Progression in Primary Human T Lymphocytes by Piperlactam S Isolated from Piper kadsura
    Yuh-Chi Kuo, Nai-Shian Yang, Cheng-Jen Chou, Lie-Chwen Lin and Wei-Jern Tsai
    Molecular Pharmacology November 2000, 58 (5) 1057-1066; DOI: https://doi.org/10.1124/mol.58.5.1057
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    Structure Activity Relationship of Carboxylic Ester Antagonists of the Vitamin D3 Receptor
    Yvonne Bury, Andreas Steinmeyer and Carsten Carlberg
    Molecular Pharmacology November 2000, 58 (5) 1067-1074; DOI: https://doi.org/10.1124/mol.58.5.1067
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    Influence of Receptor Number on Functional Responses Elicited by Agonists Acting at the Human Adenosine A1 Receptor: Evidence for Signaling Pathway-Dependent Changes in Agonist Potency and Relative Intrinsic Activity
    Yolande Cordeaux, Stephen J. Briddon, Anne E. Megson, Jacqui McDonnell, John M. Dickenson and Stephen J. Hill
    Molecular Pharmacology November 2000, 58 (5) 1075-1084; DOI: https://doi.org/10.1124/mol.58.5.1075
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    Analysis of the Pharmacological and Molecular Heterogeneity of I2-Imidazoline-Binding Proteins using Monoamine Oxidase-Deficient Mouse Models
    Anne Remaury, Rita Raddatz, Catherine Ordener, Sandra Savic, Jean C. Shih, Kevin Chen, Isabelle Seif, Edward De Maeyer, Stephen M. Lanier and Angelo Parini
    Molecular Pharmacology November 2000, 58 (5) 1085-1090; DOI: https://doi.org/10.1124/mol.58.5.1085
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    Agonist Binding and Function at the Human α2A-Adrenoceptor: Allosteric Modulation by Amilorides
    Ray A. Leppik and Nigel J. M. Birdsall
    Molecular Pharmacology November 2000, 58 (5) 1091-1099; DOI: https://doi.org/10.1124/mol.58.5.1091
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    Polyanionic (i.e., Polysulfonate) Dendrimers Can Inhibit the Replication of Human Immunodeficiency Virus by Interfering with Both Virus Adsorption and Later Steps (Reverse Transcriptase/Integrase) in the Virus Replicative Cycle
    Myriam Witvrouw, Valery Fikkert, Wim Pluymers, Barry Matthews, Karen Mardel, Dominique Schols, John Raff, Zeger Debyser, Erik De Clercq, George Holan and Christophe Pannecouque
    Molecular Pharmacology November 2000, 58 (5) 1100-1108; DOI: https://doi.org/10.1124/mol.58.5.1100
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    Metabolism and Mode of Inhibition of Varicella-Zoster Virus byl-β-5-Bromovinyl-(2-hydroxymethyl)-(1,3-dioxolanyl)uracil Is Dependent on Viral Thymidine Kinase
    Ling Li, Ginger E. Dutschman, Elizabeth A. Gullen, Eisaku Tsujii, Susan P. Grill, Yongseok Choi, Chung K. Chu and Yung-chi Cheng
    Molecular Pharmacology November 2000, 58 (5) 1109-1114; DOI: https://doi.org/10.1124/mol.58.5.1109
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    Pharmacological Blockade of ERG K+ Channels and Ca2+ Influx through Store-Operated Channels Exerts Opposite Effects on Intracellular Ca2+ Oscillations in Pituitary GH3 Cells
    Agnese Secondo, Maurizio Taglialatela, Mauro Cataldi, Giovanna Giorgio, Monica Valore, Gianfranco Di Renzo and Lucio Annunziato
    Molecular Pharmacology November 2000, 58 (5) 1115-1128; DOI: https://doi.org/10.1124/mol.58.5.1115
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    Benzodiazepines Induce a Conformational Change in the Region of the γ-Aminobutyric Acid Type A Receptor α1-Subunit M3 Membrane-Spanning Segment
    Daniel B. Williams and Myles H. Akabas
    Molecular Pharmacology November 2000, 58 (5) 1129-1136; DOI: https://doi.org/10.1124/mol.58.5.1129
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    Sodium Dodecyl Sulfate-Stable Complexes of Echistatin and RGD-Dependent Integrins: A Novel Approach to Study Integrins
    Gaétan Thibault
    Molecular Pharmacology November 2000, 58 (5) 1137-1145; DOI: https://doi.org/10.1124/mol.58.5.1137
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    Establishment of an Isogenic Human Colon Tumor Model forNQO1 Gene Expression: Application to Investigate the Role of DT-Diaphorase in Bioreductive Drug Activation In Vitro and In Vivo
    Swee Y. Sharp, Lloyd R. Kelland, Melanie R. Valenti, Lisa A. Brunton, Steve Hobbs and Paul Workman
    Molecular Pharmacology November 2000, 58 (5) 1146-1155; DOI: https://doi.org/10.1124/mol.58.5.1146

Accelerated Communications

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    Homologous and Heterologous Phosphorylation of the AT2 Angiotensin Receptor by Protein Kinase C
    Jesus A. Olivares-Reyes, Suman Jayadev, László Hunyady, Kevin J. Catt and Roger D. Smith
    Molecular Pharmacology November 2000, 58 (5) 1156-1161; DOI: https://doi.org/10.1124/mol.58.5.1156
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    Localization of the Sites Mediating Desensitization of the β2-Adrenergic Receptor by the GRK Pathway
    Anita Seibold, Bruce Williams, Zai-Feng Huang, Jackie Friedman, Robert H. Moore, Brian J. Knoll and Richard B. Clark
    Molecular Pharmacology November 2000, 58 (5) 1162-1173; DOI: https://doi.org/10.1124/mol.58.5.1162
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Molecular Pharmacology: 58 (5)
Molecular Pharmacology
Vol. 58, Issue 5
1 Nov 2000
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