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Research ArticleArticle

Competitive CYP2C9 Inhibitors: Enzyme Inhibition Studies, Protein Homology Modeling, and Three-Dimensional Quantitative Structure-Activity Relationship Analysis

Lovisa Afzelius, Ismael Zamora, Marianne Ridderström, Tommy B. Andersson, Anders Karlén and Collen M. Masimirembwa
Molecular Pharmacology April 2001, 59 (4) 909-919; DOI: https://doi.org/10.1124/mol.59.4.909
Lovisa Afzelius
1 2
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Ismael Zamora
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Marianne Ridderström
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Tommy B. Andersson
1 2
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Anders Karlén
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Collen M. Masimirembwa
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Article Information

vol. 59 no. 4 909-919
DOI 
https://doi.org/10.1124/mol.59.4.909
PubMed 
11259637

Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0026-895X
Online ISSN 
1521-0111
History 
  • Received October 3, 2000
  • Accepted December 20, 2000
  • Published online April 1, 2001.

Copyright & Usage 
The American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. Lovisa Afzelius1,2,
  2. Ismael Zamora1,
  3. Marianne Ridderström1,
  4. Tommy B. Andersson1,
  5. Anders Karlén2, and
  6. Collen M. Masimirembwa1
  1. 1Department of Drug Metabolism and Pharmacokinetics & Bioanalytical Chemistry, AstraZeneca R&D, Mölndal, Sweden (L.A., I.Z., M.R., T.B.A., C.M.M.); and 2Department of Organic Pharmaceutical Chemistry, Biomedical Center, Uppsala University, Uppsala, Sweden (L.A., A.K.)
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Molecular Pharmacology: 59 (4)
Molecular Pharmacology
Vol. 59, Issue 4
1 Apr 2001
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Research ArticleArticle

Competitive CYP2C9 Inhibitors: Enzyme Inhibition Studies, Protein Homology Modeling, and Three-Dimensional Quantitative Structure-Activity Relationship Analysis

Lovisa Afzelius, Ismael Zamora, Marianne Ridderström, Tommy B. Andersson, Anders Karlén and Collen M. Masimirembwa
Molecular Pharmacology April 1, 2001, 59 (4) 909-919; DOI: https://doi.org/10.1124/mol.59.4.909

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Research ArticleArticle

Competitive CYP2C9 Inhibitors: Enzyme Inhibition Studies, Protein Homology Modeling, and Three-Dimensional Quantitative Structure-Activity Relationship Analysis

Lovisa Afzelius, Ismael Zamora, Marianne Ridderström, Tommy B. Andersson, Anders Karlén and Collen M. Masimirembwa
Molecular Pharmacology April 1, 2001, 59 (4) 909-919; DOI: https://doi.org/10.1124/mol.59.4.909
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