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Molecular Pharmacology

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Table of Contents

May 01, 2001; Volume 59,Issue 5

Accelerated Communications

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    Cyanovirin-N Defines a New Class of Antiviral Agent Targeting N-Linked, High-Mannose Glycans in an Oligosaccharide-Specific Manner
    Anders J. Bolmstedt, Barry R. O'Keefe, Shilpa R. Shenoy, James B. McMahon and Michael R. Boyd
    Molecular Pharmacology May 2001, 59 (5) 949-954; DOI: https://doi.org/10.1124/mol.59.5.949
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    The CB1 Cannabinoid Receptor of Astrocytes Is Coupled to Sphingomyelin Hydrolysis through the Adaptor Protein Fan
    Cristina Sánchez, Daniel Rueda, Bruno Ségui, Ismael Galve-Roperh, Thierry Levade and Manuel Guzmán
    Molecular Pharmacology May 2001, 59 (5) 955-959; DOI: https://doi.org/10.1124/mol.59.5.955
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    Evidence for Direct Protein Kinase-C Mediated Modulation ofN-Methyl-d-aspartate Receptor Current
    Guey-Ying Liao, David A. Wagner, Michael H. Hsu and John P. Leonard
    Molecular Pharmacology May 2001, 59 (5) 960-964; DOI: https://doi.org/10.1124/mol.59.5.960
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    BAY36-7620: A Potent Non-Competitive mGlu1 Receptor Antagonist with Inverse Agonist Activity.
    Fiona Y. Carroll, Andreas Stolle, Philip M. Beart, Arnd Voerste, Isabelle Brabet, Frank Mauler, Cécile Joly, Horst Antonicek, Joël Bockaert, Thomas Müller, Jean Philippe Pin and Laurent Prézeau
    Molecular Pharmacology May 2001, 59 (5) 965-973; DOI: https://doi.org/10.1124/mol.59.5.965

Articles

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    Increased Bioavailability of the Food-Derived Carcinogen 2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine in MRP2-Deficient Rats
    Christoph G. Dietrich, D. Rudi de Waart, Roel Ottenhoff, Ivo G. Schoots and Ronald P. J. Oude Elferink
    Molecular Pharmacology May 2001, 59 (5) 974-980; DOI: https://doi.org/10.1124/mol.59.5.974
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    Zn2+ Induces Stimulation of the c-Jun N-Terminal Kinase Signaling Pathway through Phosphoinositide 3-Kinase
    Soo-Jung Eom, Eun Young Kim, Ji Eun Lee, Hyo Jung Kang, Jaekyung Shim, Seong Up Kim, Byoung Joo Gwag and Eui-Ju Choi
    Molecular Pharmacology May 2001, 59 (5) 981-986; DOI: https://doi.org/10.1124/mol.59.5.981
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    Transcriptional Induction of Hepatic NADPH: Cytochrome P450 Oxidoreductase by Thyroid Hormone
    Huan-Chen Li, Dongxu Liu and David J. Waxman
    Molecular Pharmacology May 2001, 59 (5) 987-995; DOI: https://doi.org/10.1124/mol.59.5.987
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    Molecular Cloning, Genomic Positioning, Promoter Identification, and Characterization of the Novel Cyclic AMP-Specific Phosphodiesterase PDE4A10
    Graham Rena, Fiona Begg, Annette Ross, Carolynn MacKenzie, Ian McPhee, Lachlan Campbell, Elaine Huston, Michael Sullivan and Miles D. Houslay
    Molecular Pharmacology May 2001, 59 (5) 996-1011; DOI: https://doi.org/10.1124/mol.59.5.996
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    Role of Protein Kinase Cα in Signaling from the Histamine H1 Receptor to the Nucleus
    A. C. Megson, E. M. Walker and S. J. Hill
    Molecular Pharmacology May 2001, 59 (5) 1012-1021; DOI: https://doi.org/10.1124/mol.59.5.1012
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    Mutational Analysis of the Functional Role of Conserved Arginine and Lysine Residues in Transmembrane Domains of the Murine Reduced Folate Carrier
    Iraida G. Sharina, Rongbao Zhao, Yanhua Wang, Solomon Babani and I. David Goldman
    Molecular Pharmacology May 2001, 59 (5) 1022-1028; DOI: https://doi.org/10.1124/mol.59.5.1022
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    Expression of Multiple Subtypes of Muscarinic Receptors and Cellular Distribution in the Human Heart
    Huizhen Wang, Hong Han, Liming Zhang, Hong Shi, Gernot Schram, Stanley Nattel and Zhiguo Wang
    Molecular Pharmacology May 2001, 59 (5) 1029-1036; DOI: https://doi.org/10.1124/mol.59.5.1029
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    Characterization of Glutamate-Gated Chloride Channels in the Pharynx of Wild-Type and Mutant Caenorhabditis elegansDelineates the Role of the Subunit GluCl-α2 in the Function of the Native Receptor
    Darrel J. Pemberton, Christopher J. Franks, Robert J. Walker and Lindy Holden-Dye
    Molecular Pharmacology May 2001, 59 (5) 1037-1043; DOI: https://doi.org/10.1124/mol.59.5.1037
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    Antimitogenic Actions of Organic Nitrates Are Potentiated by Sildenafil and Mediated Via Activation of Protein Kinase A
    Michael T. Osinski, Bernhard H. Rauch and Karsten Schrör
    Molecular Pharmacology May 2001, 59 (5) 1044-1050; DOI: https://doi.org/10.1124/mol.59.5.1044
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    Characterization of the Dizocilpine Binding Site on the Nicotinic Acetylcholine Receptor
    Hugo R. Arias, Elizabeth A. McCardy and Michael P. Blanton
    Molecular Pharmacology May 2001, 59 (5) 1051-1060; DOI: https://doi.org/10.1124/mol.59.5.1051
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    Direct Activation of an Inwardly Rectifying Potassium Channel by Arachidonic Acid
    Yi Liu, Dong Liu, Louise Heath, Diane M. Meyers, Douglas S. Krafte, P. Kay Wagoner, Christopher P. Silvia, Weifeng Yu and Mark E. Curran
    Molecular Pharmacology May 2001, 59 (5) 1061-1068; DOI: https://doi.org/10.1124/mol.59.5.1061
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    Cocaine Blocks HERG, but Not KvLQT1+minK, Potassium Channels
    Shetuan Zhang, Sridharan Rajamani, Yuenmu Chen, Qiuming Gong, Yajing Rong, Zhengfeng Zhou, Arnold Ruoho and Craig T. January
    Molecular Pharmacology May 2001, 59 (5) 1069-1076; DOI: https://doi.org/10.1124/mol.59.5.1069
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    Charged Amino Acids in the Transmembrane Domains Are Involved in the Determination of the Substrate Specificity of Rat Mrp2
    Kousei Ito, Hiroshi Suzuki and Yuichi Sugiyama
    Molecular Pharmacology May 2001, 59 (5) 1077-1085; DOI: https://doi.org/10.1124/mol.59.5.1077
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    Phospholipids as Modulators of KATP Channels: Distinct Mechanisms for Control of Sensitivity to Sulphonylureas, K+ Channel Openers, and ATP
    Tobias Krauter, J. Peter Ruppersberg and Thomas Baukrowitz
    Molecular Pharmacology May 2001, 59 (5) 1086-1093; DOI: https://doi.org/10.1124/mol.59.5.1086
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    The Novel Triterpenoid CDDO Induces Apoptosis and Differentiation of Human Osteosarcoma Cells by a Caspase-8 Dependent Mechanism
    Yasumasa Ito, Pramod Pandey, Michael B. Sporn, Rakesh Datta, Surender Kharbanda and Donald Kufe
    Molecular Pharmacology May 2001, 59 (5) 1094-1099; DOI: https://doi.org/10.1124/mol.59.5.1094
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    Disparate Role of Na+ Channel D2-S6 Residues in Batrachotoxin and Local Anesthetic Action
    Sho-Ya Wang, Maria Barile and Ging Kuo Wang
    Molecular Pharmacology May 2001, 59 (5) 1100-1107; DOI: https://doi.org/10.1124/mol.59.5.1100
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    Effect of α Subunit on Allosteric Modulation of Ion Channel Function in Stably Expressed Human Recombinant γ-Aminobutyric AcidA Receptors Determined Using36Cl Ion Flux
    Alison J. Smith, Luanda Alder, Jonathan Silk, Charles Adkins, Alan E. Fletcher, Tim Scales, Julie Kerby, George Marshall, Keith A. Wafford, Ruth M. McKernan and John R. Atack
    Molecular Pharmacology May 2001, 59 (5) 1108-1118; DOI: https://doi.org/10.1124/mol.59.5.1108
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    High-Intensity p38 Kinase Activity Is Critical for p21 cip1 Induction and the Antiproliferative Function of Gi Protein-Coupled Receptors
    Forbes Alderton, Patrick P. A. Humphrey and Lynda A. Sellers
    Molecular Pharmacology May 2001, 59 (5) 1119-1128; DOI: https://doi.org/10.1124/mol.59.5.1119
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    Quantitative Analysis of Inward and Outward Transport Rates in Cells Stably Expressing the Cloned Human Serotonin Transporter: Inconsistencies with the Hypothesis of Facilitated Exchange Diffusion
    Harald H. Sitte, Birgit Hiptmair, Julia Zwach, Christian Pifl, Ernst A. Singer and Petra Scholze
    Molecular Pharmacology May 2001, 59 (5) 1129-1137; DOI: https://doi.org/10.1124/mol.59.5.1129
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    PI3K Inhibitors Reverse the Suppressive Actions of Insulin on CYP2E1 Expression by Activating Stress-Response Pathways in Primary Rat Hepatocytes
    Jaspreet S. Sidhu, Fei Liu, Sean M. Boyle and Curtis J. Omiecinski
    Molecular Pharmacology May 2001, 59 (5) 1138-1146; DOI: https://doi.org/10.1124/mol.59.5.1138
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    Activation of Phosphatidylinositol 3-Kinase and Akt bytert-Butylhydroquinone Is Responsible for Antioxidant Response Element-Mediated rGSTA2 Induction in H4IIE Cells
    Keon Wook Kang, Min Kyung Cho, Chang Ho Lee and Sang Geon Kim
    Molecular Pharmacology May 2001, 59 (5) 1147-1156; DOI: https://doi.org/10.1124/mol.59.5.1147
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    Dual Incorporation of Photoaffinity Ligands on Dopamine Transporters Implicates Proximity of Labeled Domains
    Roxanne A. Vaughan, Jon D. Gaffaney, John R. Lever, Maarten E. A. Reith and Aloke K. Dutta
    Molecular Pharmacology May 2001, 59 (5) 1157-1164; DOI: https://doi.org/10.1124/mol.59.5.1157
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    Involvement of Nuclear Factor κB in c-Myc Induction by Tubulin Polymerization Inhibitors
    V. Bourgarel-Rey, S. Vallee, O. Rimet, S. Champion, D. Braguer, A. Desobry, C. Briand and Y. Barra
    Molecular Pharmacology May 2001, 59 (5) 1165-1170; DOI: https://doi.org/10.1124/mol.59.5.1165
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    Modulation of Multidrug Resistance Protein 1 (MRP1/ABCC1) Transport and ATPase Activities by Interaction with Dietary Flavonoids
    Elaine M. Leslie, Qingcheng Mao, Curtis J. Oleschuk, Roger G. Deeley and Susan P. C. Cole
    Molecular Pharmacology May 2001, 59 (5) 1171-1180; DOI: https://doi.org/10.1124/mol.59.5.1171
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    Phosphorylation of Uridine and Cytidine Nucleoside Analogs by Two Human Uridine-Cytidine Kinases
    An R. Van Rompay, Ameli Norda, Karin Lindén, Magnus Johansson and Anna Karlsson
    Molecular Pharmacology May 2001, 59 (5) 1181-1186; DOI: https://doi.org/10.1124/mol.59.5.1181
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    Determination of Amino Acid Residues that are Accessible from the Ligand Binding Crevice in the Seventh Transmembrane-Spanning Region of the Human A1 Adenosine Receptor
    Eric S. Dawson and Jack N. Wells
    Molecular Pharmacology May 2001, 59 (5) 1187-1195; DOI: https://doi.org/10.1124/mol.59.5.1187
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    Tripterygium wilfordii Hook F Extract Suppresses Proinflammatory Cytokine-Induced Expression of Matrix Metalloproteinase Genes in Articular Chondrocytes by Inhibiting Activating Protein-1 and Nuclear Factor-κB Activities
    Judith Sylvester, Abdelhamid Liacini, Wen Qing Li, Faramaze Dehnade and Muhammad Zafarullah
    Molecular Pharmacology May 2001, 59 (5) 1196-1205; DOI: https://doi.org/10.1124/mol.59.5.1196
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    Structural Determinants of Adenophostin A Activity at Inositol Trisphosphate Receptors
    Vanessa Correa, Andrew M. Riley, Satoshi Shuto, Graeme Horne, Edmund P. Nerou, Rachel D. Marwood, Barry V. L. Potter and Colin W. Taylor
    Molecular Pharmacology May 2001, 59 (5) 1206-1215; DOI: https://doi.org/10.1124/mol.59.5.1206
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    Mitogen-Activated Protein Kinase Kinase Inhibitor PD98059 Blocks the trans-Activation but Not the Stabilization or DNA Binding Ability of Hypoxia-Inducible Factor-1α
    Eunseon Hur, Keun Young Chang, Eunjung Lee, Seung-Ki Lee and Hyunsung Park
    Molecular Pharmacology May 2001, 59 (5) 1216-1224; DOI: https://doi.org/10.1124/mol.59.5.1216
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    Cloning and Characterization of the Mouse α1C/A-Adrenergic Receptor Gene and Analysis of an α1C Promoter in Cardiac Myocytes: Role of an MCAT Element That Binds Transcriptional Enhancer Factor-1 (TEF-1)
    Timothy D. O'Connell, D. Gregg Rokosh and Paul C. Simpson
    Molecular Pharmacology May 2001, 59 (5) 1225-1234; DOI: https://doi.org/10.1124/mol.59.5.1225
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    Use of Antisense Oligonucleotides to Verify the Role of the α1A-Adrenergic Receptor in the Contractility of the Rat Uterus Post Partum
    E. Ducza, R. Gáspár, A. Márki, P. Gyula, S. Bottka and G. Falkay
    Molecular Pharmacology May 2001, 59 (5) 1235-1242; DOI: https://doi.org/10.1124/mol.59.5.1235
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    Calcium Channel α2δ Subunits—Structure and Gabapentin Binding
    Elsé Marais, Norbert Klugbauer and Franz Hofmann
    Molecular Pharmacology May 2001, 59 (5) 1243-1248; DOI: https://doi.org/10.1124/mol.59.5.1243
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    Synthetic Phytoceramides Induce Apoptosis with Higher Potency than Ceramides
    Onyou Hwang, Guncheol Kim, Yeon Joo Jang, Seong Who Kim, Guiyong Choi, Hyun Jin Choi, Seon Young Jeon, Don Gyu Lee and Jae Dam Lee
    Molecular Pharmacology May 2001, 59 (5) 1249-1255; DOI: https://doi.org/10.1124/mol.59.5.1249
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    Agonist-Dependent Delivery of M2 Muscarinic Acetylcholine Receptors to the Cell Surface after Pertussis Toxin Treatment
    Aaron G. Roseberry, Moritz Bünemann, Jyoti Elavunkal and M. Marlene Hosey
    Molecular Pharmacology May 2001, 59 (5) 1256-1268; DOI: https://doi.org/10.1124/mol.59.5.1256
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    Induction of Differentiation in F9 Cells and Activation of Peroxisome Proliferator-Activated Receptor δ by Valproic Acid and Its Teratogenic Derivatives
    Uwe Werling, Sandra Siehler, Margarethe Litfin, Heinz Nau and Martin Göttlicher
    Molecular Pharmacology May 2001, 59 (5) 1269-1276; DOI: https://doi.org/10.1124/mol.59.5.1269
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    Identification and Characterization of Human Organic Anion Transporter 3 Expressing Predominantly in the Kidney
    Seok Ho Cha, Takashi Sekine, Jun-ichi Fukushima, Yoshikatsu Kanai, Yukari Kobayashi, Tomoyuki Goya and Hitoshi Endou
    Molecular Pharmacology May 2001, 59 (5) 1277-1286; DOI: https://doi.org/10.1124/mol.59.5.1277
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    Scabronine G-Methylester Enhances Secretion of Neurotrophic Factors Mediated by an Activation of Protein Kinase C-ζ
    Yutaro Obara, Hironori Kobayashi, Tomihisa Ohta, Yasushi Ohizumi and Norimichi Nakahata
    Molecular Pharmacology May 2001, 59 (5) 1287-1297; DOI: https://doi.org/10.1124/mol.59.5.1287
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    Diamidine Compounds: Selective Uptake and Targeting inPlasmodium falciparum
    Andrew M. W. Stead, Patrick G. Bray, I. Geoffrey Edwards, Harry P. DeKoning, Barry C. Elford, Paul A. Stocks and Stephen A. Ward
    Molecular Pharmacology May 2001, 59 (5) 1298-1306; DOI: https://doi.org/10.1124/mol.59.5.1298
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    Antimineralocorticoid 11β-Substituted Spirolactones Exhibit Androgen Receptor Agonistic Activity: A Structure Function Study
    Philippe Nirdé, Béatrice Térouanne, Nadine Gallais, Charles Sultan and Gilles Auzou
    Molecular Pharmacology May 2001, 59 (5) 1307-1313; DOI: https://doi.org/10.1124/mol.59.5.1307
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    Involvement of Caveolin in Ligand-Induced Recruitment and Internalization of A1 Adenosine Receptor and Adenosine Deaminase in an Epithelial Cell Line
    Silvia Ginés, Franciso Ciruela, Javier Burgueño, Vicent Casadó, Enric. I. Canela, Josefa Mallol, Carme Lluı́s and Rafael Franco
    Molecular Pharmacology May 2001, 59 (5) 1314-1323; DOI: https://doi.org/10.1124/mol.59.5.1314
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    Carboxypeptidase D Is Up-Regulated in RAW 264.7 Macrophages and Stimulates Nitric Oxide Synthesis by Cells in Arginine-Free Medium
    Vaishali Hadkar and Randal A. Skidgel
    Molecular Pharmacology May 2001, 59 (5) 1324-1332; DOI: https://doi.org/10.1124/mol.59.5.1324
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    Rhodostomin, A Snake Venom Disintegrin, Inhibits Angiogenesis Elicited by Basic Fibroblast Growth Factor and Suppresses Tumor Growth by A Selective αvβ3 Blockade of Endothelial Cells
    Chia-Hsin Yeh, Hui-Chin Peng, Rong-Seng Yang and Tur-Fu Huang
    Molecular Pharmacology May 2001, 59 (5) 1333-1342; DOI: https://doi.org/10.1124/mol.59.5.1333
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    Molecular Mechanism for Agonist-Promoted α2A-Adrenoceptor Activation by Norepinephrine and Epinephrine
    Tommi Nyrönen, Marjo Pihlavisto, Juha M. Peltonen, Anna-Marja Hoffrén, Minna Varis, Tiina Salminen, Siegfried Wurster, Anne Marjamäki, Liisa Kanerva, Erja Katainen, Leif Laaksonen, Juha-Matti Savola, Mika Scheinin and Mark S. Johnson
    Molecular Pharmacology May 2001, 59 (5) 1343-1354; DOI: https://doi.org/10.1124/mol.59.5.1343

Erratum

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    Correction to “Mechanisms of agonist-induced down-regulation of the human κ-opioid receptor: internalization is required for down-regulation”
    Molecular Pharmacology May 2001, 59 (5) 1355; DOI: https://doi.org/10.1124/mol.59.5.1355
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Molecular Pharmacology: 59 (5)
Molecular Pharmacology
Vol. 59, Issue 5
1 May 2001
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