Table of Contents

Articles

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  Characterization of a Human Colorectal Carcinoma Cell Line with Acquired Resistance to Flavopiridol

  Victoria Smith, Florence Raynaud, Paul Workman and Lloyd R. Kelland

  Molecular Pharmacology November 2001, 60 (5) 885-893; DOI: https://doi.org/10.1124/mol.60.5.885
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  Inflammation Enhances μ-Opioid Receptor Transcription and Expression in Mice Intestine

  Olga Pol, Francesc Alameda and Margarita M. Puig

  Molecular Pharmacology November 2001, 60 (5) 894-899; DOI: https://doi.org/10.1124/mol.60.5.894
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  Differential Roles of p21^Waf1 and p27^Kip1in Modulating Chemosensitivity and Their Possible Application in Drug Discovery Studies

  Mathias Schmidt, Yang Lu, John M. Parant, Guillermina Lozano, Gerald Bacher, Thomas Beckers and Zhen Fan

  Molecular Pharmacology November 2001, 60 (5) 900-906; DOI: https://doi.org/10.1124/mol.60.5.900
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  Enhanced Acetaminophen Hepatotoxicity in Transgenic Mice Overexpressing BCL-2

  Michael L. Adams, Robert H. Pierce, Mary E. Vail, Collin C. White, Robert P. Tonge, Terrence J. Kavanagh, Nelson Fausto, Sidney D. Nelson and Sam A. Bruschi

  Molecular Pharmacology November 2001, 60 (5) 907-915; DOI: https://doi.org/10.1124/mol.60.5.907
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  The Carboxyl Terminus of the Prolactin-Releasing Peptide Receptor Interacts with PDZ Domain Proteins Involved in α-Amino-3-hydroxy-5-methylisoxazole-4-propionic Acid Receptor Clustering

  Steven H. S. Lin, Amy C. Arai, Zhiwei Wang, Hans-Peter Nothacker and Olivier Civelli

  Molecular Pharmacology November 2001, 60 (5) 916-923; DOI: https://doi.org/10.1124/mol.60.5.916
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  Thyrotropin Activates Mitogen-Activated Protein Kinase Pathway in FRTL-5 by a cAMP-Dependent Protein Kinase A-Independent Mechanism

  Luisa Iacovelli, Loredana Capobianco, Lorena Salvatore, Michele Sallese, Gabriel Maximo D'Ancona and Antonio De Blasi

  Molecular Pharmacology November 2001, 60 (5) 924-933; DOI: https://doi.org/10.1124/mol.60.5.924
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  Vectorial Transport by Double-Transfected Cells Expressing the Human Uptake Transporter SLC21A8 and the Apical Export Pump ABCC2

  Yunhai Cui, Jörg König and Dietrich Keppler

  Molecular Pharmacology November 2001, 60 (5) 934-943; DOI: https://doi.org/10.1124/mol.60.5.934
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  Identification of Essential Residues Involved in the Glutamate Binding Pocket of the Group II Metabotropic Glutamate Receptor

  Pari Malherbe, Frédéric Knoflach, Clemens Broger, Serge Ohresser, Claudia Kratzeisen, Geo Adam, Heinz Stadler, John A. Kemp and Vincent Mutel

  Molecular Pharmacology November 2001, 60 (5) 944-954; DOI: https://doi.org/10.1124/mol.60.5.944
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  Differential Distribution of β-Adrenergic Receptor Subtypes in Blood Vessels of Knockout Mice Lacking β₁ - or β₂-Adrenergic Receptors

  Andrzej Chruscinski, Marc E. Brede, Lorenz Meinel, Martin J. Lohse, Brian K. Kobilka and Lutz Hein

  Molecular Pharmacology November 2001, 60 (5) 955-962; DOI: https://doi.org/10.1124/mol.60.5.955
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  Positive Allosteric Modulation of Native and Recombinant γ-Aminobutyric Acid_B Receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its Aldehyde Analog CGP13501

  Stephan Urwyler, Johannes Mosbacher, Kurt Lingenhoehl, Jakob Heid, Karin Hofstetter, Wolfgang Froestl, Bernhard Bettler and Klemens Kaupmann

  Molecular Pharmacology November 2001, 60 (5) 963-971; DOI: https://doi.org/10.1124/mol.60.5.963
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  Methimazole As an Antioxidant and Immunomodulator in Thyroid Cells: Mechanisms Involving Interferon-γ Signaling and H₂O₂ Scavenging

  Ho Kim, Tae-Hoon Lee, Young Sun Hwang, Mi Ae Bang, Kang Hwa Kim, Jae Mi Suh, Hyo Kyun Chung, Dae-Yeul Yu, Kyung-Kwang Lee, O-Yu Kwon, Heung Kyu Ro and Minho Shong

  Molecular Pharmacology November 2001, 60 (5) 972-980; DOI: https://doi.org/10.1124/mol.60.5.972
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  Potent Inhibition of Telomerase by Small-Molecule Pentacyclic Acridines Capable of Interacting with G-Quadruplexes

  Sharon M. Gowan, Robert Heald, Malcolm F. G. Stevens and Lloyd R. Kelland

  Molecular Pharmacology November 2001, 60 (5) 981-988; DOI: https://doi.org/10.1124/mol.60.5.981
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  Activation of Inositol 1,4,5-Trisphosphate Receptor Is Essential for the Opening of Mouse TRP5 Channels

  Hideaki Kanki, Mariko Kinoshita, Akinori Akaike, Masamichi Satoh, Yasuo Mori and Shuji Kaneko

  Molecular Pharmacology November 2001, 60 (5) 989-998; DOI: https://doi.org/10.1124/mol.60.5.989
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  Allosteric Effects of G Protein Overexpression on the Binding of β-Adrenergic Ligands with Distinct Inverse Efficacies

  Mounia Azzi, Graciela Piñeyro, Stéphanie Pontier, Stéphane Parent, Hervé Ansanay and Michel Bouvier

  Molecular Pharmacology November 2001, 60 (5) 999-1007; DOI: https://doi.org/10.1124/mol.60.5.999
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  Multiple Kinetics of Mitochondrial Cytochrome cRelease in Drug-Induced Apoptosis

  C. Marc Luetjens, Donat Kögel, Claus Reimertz, Heiko Düßmann, Andrea Renz, Klaus Schulze-Osthoff, Anna-Liisa Nieminen, Monika Poppe and Jochen H. M. Prehn

  Molecular Pharmacology November 2001, 60 (5) 1008-1019; DOI: https://doi.org/10.1124/mol.60.5.1008
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  Cell-Type Specific Effects of Endocytosis Inhibitors on 5-Hydroxytryptamine_2A Receptor Desensitization and Resensitization Reveal an Arrestin-, GRK2-, and GRK5-Independent Mode of Regulation in Human Embryonic Kidney 293 Cells

  John A. Gray, Douglas J. Sheffler, Anushree Bhatnagar, Jason A. Woods, Sandra J. Hufeisen, Jeffrey L. Benovic and Bryan L. Roth

  Molecular Pharmacology November 2001, 60 (5) 1020-1030; DOI: https://doi.org/10.1124/mol.60.5.1020
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  Sorting Functions of the Individual Cytoplasmic Domains of the G Protein-Coupled Vasopressin V₂ Receptor in Madin Darby Canine Kidney Epithelial Cells

  Ricardo Hermosilla and Ralf Schülein

  Molecular Pharmacology November 2001, 60 (5) 1031-1039; DOI: https://doi.org/10.1124/mol.60.5.1031
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  Simultaneous Expression of Guinea Pig UDP-Glucuronosyltransferase 2B21 and 2B22 in COS-7 Cells enhances UDP-Glucuronosyltransferase 2B21-Catalyzed Morphine-6-Glucuronide Formation

  Yuji Ishii, Aya Miyoshi, Ryoichi Watanabe, Kazuoki Tsuruda, Minoru Tsuda, Yuki Yamaguchi-Nagamatsu, Kunihiro Yoshisue, Mitsuko Tanaka, Daisuke Maji, Satoru Ohgiya and Kazuta Oguri

  Molecular Pharmacology November 2001, 60 (5) 1040-1048; DOI: https://doi.org/10.1124/mol.60.5.1040
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  Histamine H2 Receptor Desensitization: Involvement of a Select Array of G Protein-Coupled Receptor Kinases

  Carina Shayo, Natalia Fernandez, Bibiana Lemos Legnazzi, Federico Monczor, Alejandro Mladovan, Alberto Baldi and Carlos Davio

  Molecular Pharmacology November 2001, 60 (5) 1049-1056; DOI: https://doi.org/10.1124/mol.60.5.1049
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  Allosteric Modulation of A₃ Adenosine Receptors by a Series of 3-(2-Pyridinyl)isoquinoline Derivatives

  Zhan-Guo Gao, Jacqueline E. Van Muijlwijk-Koezen, Aishe Chen, Christa E. Müller, Adriaan P. Ijzerman and Kenneth A. Jacobson

  Molecular Pharmacology November 2001, 60 (5) 1057-1063; DOI: https://doi.org/10.1124/mol.60.5.1057
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  Inverse Agonist Up-Regulates the Constitutively Active D3.49(164)Q Mutant of the Rat μ-Opioid Receptor by Stabilizing the Structure and Blocking Constitutive Internalization and Down-Regulation

  Jin Li, Chongguang Chen, Peng Huang and Lee-Yuan Liu-Chen

  Molecular Pharmacology November 2001, 60 (5) 1064-1075; DOI: https://doi.org/10.1124/mol.60.5.1064
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  Expression of α-Transducin in Chinese Hamster Ovary Cells Stably Transfected with the Human δ-Opioid Receptor Attenuates Chronic Opioid Agonist-Induced Adenylyl Cyclase Superactivation

  Marc Rubenzik, Eva Varga, Dagmar Stropova, William R. Roeske and Henry I. Yamamura

  Molecular Pharmacology November 2001, 60 (5) 1076-1082; DOI: https://doi.org/10.1124/mol.60.5.1076
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  Anti-Inflammatory Effects of the Partially Purified Extract of Radix Stephaniae tetrandrae: Comparative Studies of Its Active Principles Tetrandrine and Fangchinoline on Human Polymorphonuclear Leukocyte Functions

  Yuh-Chiang Shen, Cheng-Jen Chou, Wen-Fei Chiou and Chieh-Fu Chen

  Molecular Pharmacology November 2001, 60 (5) 1083-1090; DOI: https://doi.org/10.1124/mol.60.5.1083
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  Mercapturic Acids (N-AcetylcysteineS-Conjugates) as Endogenous Substrates for the Renal Organic Anion Transporter-1

  James M. Pombrio, Adam Giangreco, Liqiong Li, Michael F. Wempe, M. W. Anders, Douglas H. Sweet, John B. Pritchard and Nazzareno Ballatori

  Molecular Pharmacology November 2001, 60 (5) 1091-1099; DOI: https://doi.org/10.1124/mol.60.5.1091
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  Phorbol 12-myristate 13-acetate Triggers the Protein Kinase A-Mediated Phosphorylation and Activation of the PDE4D5 cAMP Phosphodiesterase in Human Aortic Smooth Muscle Cells through a Route Involving Extracellular Signal Regulated Kinase (ERK)

  George Baillie, Simon J. MacKenzie and Miles D. Houslay

  Molecular Pharmacology November 2001, 60 (5) 1100-1111; DOI: https://doi.org/10.1124/mol.60.5.1100
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  Mpl Ligand Increases P2Y1 Receptor Gene Expression in Megakaryocytes with No Concomitant Change in Platelet Response to ADP

  Béatrice Hechler, Paul Toselli, Catherine Ravanat, Christian Gachet and Katya Ravid

  Molecular Pharmacology November 2001, 60 (5) 1112-1120; DOI: https://doi.org/10.1124/mol.60.5.1112
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  Block of Cloned Human T-Type Calcium Channels by Succinimide Antiepileptic Drugs

  Juan Carlos Gomora, Asif N. Daud, Marco Weiergräber and Edward Perez-Reyes

  Molecular Pharmacology November 2001, 60 (5) 1121-1132; DOI: https://doi.org/10.1124/mol.60.5.1121
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  Histamine H₁-Receptor Activation of Nuclear Factor-κB: Roles for Gβγ- and Gα_q/11-Subunits in Constitutive and Agonist-Mediated Signaling

  Remko A. Bakker, Stefan B. J. Schoonus, Martine J. Smit, Henk Timmerman and Rob Leurs

  Molecular Pharmacology November 2001, 60 (5) 1133-1142; DOI: https://doi.org/10.1124/mol.60.5.1133
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  Acquisition of Human Concentrative Nucleoside Transporter 2 (hCNT2) Activity by Gene Transfer Confers Sensitivity to Fluoropyrimidine Nucleosides in Drug-Resistant Leukemia Cells

  Thack T. Lang, Milada Selner, James D. Young and Carol E. Cass

  Molecular Pharmacology November 2001, 60 (5) 1143-1152; DOI: https://doi.org/10.1124/mol.60.5.1143