Skip to main content
Advertisement

Main menu

  • Home
  • Articles
    • Current Issue
    • Fast Forward
    • Latest Articles
    • Archive
  • Information
    • Instructions to Authors
    • Submit a Manuscript
    • FAQs
    • For Subscribers
    • Terms & Conditions of Use
    • Permissions
  • Editorial Board
  • Alerts
    • Alerts
    • RSS Feeds
  • Virtual Issues
  • Feedback
  • Other Publications
    • Drug Metabolism and Disposition
    • Journal of Pharmacology and Experimental Therapeutics
    • Molecular Pharmacology
    • Pharmacological Reviews
    • Pharmacology Research & Perspectives
    • ASPET

User menu

  • My alerts
  • Log in
  • My Cart

Search

  • Advanced search
Molecular Pharmacology
  • Other Publications
    • Drug Metabolism and Disposition
    • Journal of Pharmacology and Experimental Therapeutics
    • Molecular Pharmacology
    • Pharmacological Reviews
    • Pharmacology Research & Perspectives
    • ASPET
  • My alerts
  • Log in
  • My Cart
Molecular Pharmacology

Advanced Search

  • Home
  • Articles
    • Current Issue
    • Fast Forward
    • Latest Articles
    • Archive
  • Information
    • Instructions to Authors
    • Submit a Manuscript
    • FAQs
    • For Subscribers
    • Terms & Conditions of Use
    • Permissions
  • Editorial Board
  • Alerts
    • Alerts
    • RSS Feeds
  • Virtual Issues
  • Feedback
  • Visit molpharm on Facebook
  • Follow molpharm on Twitter
  • Follow molpharm on LinkedIn

Table of Contents

November 01, 2001; Volume 60,Issue 5

Perspective

  • You have access
    Positive Allosteric Modulators for γ-Aminobutyric AcidB Receptors Open New Routes for the Development of Drugs Targeting Family 3 G-Protein-Coupled Receptors
    Jean-Philippe Pin, Marie-Laure Parmentier and Laurent Prézeau
    Molecular Pharmacology November 2001, 60 (5) 881-884; DOI: https://doi.org/10.1124/mol.60.5.881

Articles

  • You have access
    Characterization of a Human Colorectal Carcinoma Cell Line with Acquired Resistance to Flavopiridol
    Victoria Smith, Florence Raynaud, Paul Workman and Lloyd R. Kelland
    Molecular Pharmacology November 2001, 60 (5) 885-893; DOI: https://doi.org/10.1124/mol.60.5.885
  • You have access
    Inflammation Enhances μ-Opioid Receptor Transcription and Expression in Mice Intestine
    Olga Pol, Francesc Alameda and Margarita M. Puig
    Molecular Pharmacology November 2001, 60 (5) 894-899; DOI: https://doi.org/10.1124/mol.60.5.894
  • You have access
    Differential Roles of p21Waf1 and p27Kip1in Modulating Chemosensitivity and Their Possible Application in Drug Discovery Studies
    Mathias Schmidt, Yang Lu, John M. Parant, Guillermina Lozano, Gerald Bacher, Thomas Beckers and Zhen Fan
    Molecular Pharmacology November 2001, 60 (5) 900-906; DOI: https://doi.org/10.1124/mol.60.5.900
  • You have access
    Enhanced Acetaminophen Hepatotoxicity in Transgenic Mice Overexpressing BCL-2
    Michael L. Adams, Robert H. Pierce, Mary E. Vail, Collin C. White, Robert P. Tonge, Terrence J. Kavanagh, Nelson Fausto, Sidney D. Nelson and Sam A. Bruschi
    Molecular Pharmacology November 2001, 60 (5) 907-915; DOI: https://doi.org/10.1124/mol.60.5.907
  • You have access
    The Carboxyl Terminus of the Prolactin-Releasing Peptide Receptor Interacts with PDZ Domain Proteins Involved in α-Amino-3-hydroxy-5-methylisoxazole-4-propionic Acid Receptor Clustering
    Steven H. S. Lin, Amy C. Arai, Zhiwei Wang, Hans-Peter Nothacker and Olivier Civelli
    Molecular Pharmacology November 2001, 60 (5) 916-923; DOI: https://doi.org/10.1124/mol.60.5.916
  • You have access
    Thyrotropin Activates Mitogen-Activated Protein Kinase Pathway in FRTL-5 by a cAMP-Dependent Protein Kinase A-Independent Mechanism
    Luisa Iacovelli, Loredana Capobianco, Lorena Salvatore, Michele Sallese, Gabriel Maximo D'Ancona and Antonio De Blasi
    Molecular Pharmacology November 2001, 60 (5) 924-933; DOI: https://doi.org/10.1124/mol.60.5.924
  • You have access
    Vectorial Transport by Double-Transfected Cells Expressing the Human Uptake Transporter SLC21A8 and the Apical Export Pump ABCC2
    Yunhai Cui, Jörg König and Dietrich Keppler
    Molecular Pharmacology November 2001, 60 (5) 934-943; DOI: https://doi.org/10.1124/mol.60.5.934
  • You have access
    Identification of Essential Residues Involved in the Glutamate Binding Pocket of the Group II Metabotropic Glutamate Receptor
    Pari Malherbe, Frédéric Knoflach, Clemens Broger, Serge Ohresser, Claudia Kratzeisen, Geo Adam, Heinz Stadler, John A. Kemp and Vincent Mutel
    Molecular Pharmacology November 2001, 60 (5) 944-954; DOI: https://doi.org/10.1124/mol.60.5.944
  • You have access
    Differential Distribution of β-Adrenergic Receptor Subtypes in Blood Vessels of Knockout Mice Lacking β1 - or β2-Adrenergic Receptors
    Andrzej Chruscinski, Marc E. Brede, Lorenz Meinel, Martin J. Lohse, Brian K. Kobilka and Lutz Hein
    Molecular Pharmacology November 2001, 60 (5) 955-962; DOI: https://doi.org/10.1124/mol.60.5.955
  • You have access
    Positive Allosteric Modulation of Native and Recombinant γ-Aminobutyric AcidB Receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its Aldehyde Analog CGP13501
    Stephan Urwyler, Johannes Mosbacher, Kurt Lingenhoehl, Jakob Heid, Karin Hofstetter, Wolfgang Froestl, Bernhard Bettler and Klemens Kaupmann
    Molecular Pharmacology November 2001, 60 (5) 963-971; DOI: https://doi.org/10.1124/mol.60.5.963
  • You have access
    Methimazole As an Antioxidant and Immunomodulator in Thyroid Cells: Mechanisms Involving Interferon-γ Signaling and H2O2 Scavenging
    Ho Kim, Tae-Hoon Lee, Young Sun Hwang, Mi Ae Bang, Kang Hwa Kim, Jae Mi Suh, Hyo Kyun Chung, Dae-Yeul Yu, Kyung-Kwang Lee, O-Yu Kwon, Heung Kyu Ro and Minho Shong
    Molecular Pharmacology November 2001, 60 (5) 972-980; DOI: https://doi.org/10.1124/mol.60.5.972
  • You have access
    Potent Inhibition of Telomerase by Small-Molecule Pentacyclic Acridines Capable of Interacting with G-Quadruplexes
    Sharon M. Gowan, Robert Heald, Malcolm F. G. Stevens and Lloyd R. Kelland
    Molecular Pharmacology November 2001, 60 (5) 981-988; DOI: https://doi.org/10.1124/mol.60.5.981
  • You have access
    Activation of Inositol 1,4,5-Trisphosphate Receptor Is Essential for the Opening of Mouse TRP5 Channels
    Hideaki Kanki, Mariko Kinoshita, Akinori Akaike, Masamichi Satoh, Yasuo Mori and Shuji Kaneko
    Molecular Pharmacology November 2001, 60 (5) 989-998; DOI: https://doi.org/10.1124/mol.60.5.989
  • You have access
    Allosteric Effects of G Protein Overexpression on the Binding of β-Adrenergic Ligands with Distinct Inverse Efficacies
    Mounia Azzi, Graciela Piñeyro, Stéphanie Pontier, Stéphane Parent, Hervé Ansanay and Michel Bouvier
    Molecular Pharmacology November 2001, 60 (5) 999-1007; DOI: https://doi.org/10.1124/mol.60.5.999
  • You have access
    Multiple Kinetics of Mitochondrial Cytochrome cRelease in Drug-Induced Apoptosis
    C. Marc Luetjens, Donat Kögel, Claus Reimertz, Heiko Düßmann, Andrea Renz, Klaus Schulze-Osthoff, Anna-Liisa Nieminen, Monika Poppe and Jochen H. M. Prehn
    Molecular Pharmacology November 2001, 60 (5) 1008-1019; DOI: https://doi.org/10.1124/mol.60.5.1008
  • You have access
    Cell-Type Specific Effects of Endocytosis Inhibitors on 5-Hydroxytryptamine2A Receptor Desensitization and Resensitization Reveal an Arrestin-, GRK2-, and GRK5-Independent Mode of Regulation in Human Embryonic Kidney 293 Cells
    John A. Gray, Douglas J. Sheffler, Anushree Bhatnagar, Jason A. Woods, Sandra J. Hufeisen, Jeffrey L. Benovic and Bryan L. Roth
    Molecular Pharmacology November 2001, 60 (5) 1020-1030; DOI: https://doi.org/10.1124/mol.60.5.1020
  • You have access
    Sorting Functions of the Individual Cytoplasmic Domains of the G Protein-Coupled Vasopressin V2 Receptor in Madin Darby Canine Kidney Epithelial Cells
    Ricardo Hermosilla and Ralf Schülein
    Molecular Pharmacology November 2001, 60 (5) 1031-1039; DOI: https://doi.org/10.1124/mol.60.5.1031
  • You have access
    Simultaneous Expression of Guinea Pig UDP-Glucuronosyltransferase 2B21 and 2B22 in COS-7 Cells enhances UDP-Glucuronosyltransferase 2B21-Catalyzed Morphine-6-Glucuronide Formation
    Yuji Ishii, Aya Miyoshi, Ryoichi Watanabe, Kazuoki Tsuruda, Minoru Tsuda, Yuki Yamaguchi-Nagamatsu, Kunihiro Yoshisue, Mitsuko Tanaka, Daisuke Maji, Satoru Ohgiya and Kazuta Oguri
    Molecular Pharmacology November 2001, 60 (5) 1040-1048; DOI: https://doi.org/10.1124/mol.60.5.1040
  • You have access
    Histamine H2 Receptor Desensitization: Involvement of a Select Array of G Protein-Coupled Receptor Kinases
    Carina Shayo, Natalia Fernandez, Bibiana Lemos Legnazzi, Federico Monczor, Alejandro Mladovan, Alberto Baldi and Carlos Davio
    Molecular Pharmacology November 2001, 60 (5) 1049-1056; DOI: https://doi.org/10.1124/mol.60.5.1049
  • You have access
    Allosteric Modulation of A3 Adenosine Receptors by a Series of 3-(2-Pyridinyl)isoquinoline Derivatives
    Zhan-Guo Gao, Jacqueline E. Van Muijlwijk-Koezen, Aishe Chen, Christa E. Müller, Adriaan P. Ijzerman and Kenneth A. Jacobson
    Molecular Pharmacology November 2001, 60 (5) 1057-1063; DOI: https://doi.org/10.1124/mol.60.5.1057
  • You have access
    Inverse Agonist Up-Regulates the Constitutively Active D3.49(164)Q Mutant of the Rat μ-Opioid Receptor by Stabilizing the Structure and Blocking Constitutive Internalization and Down-Regulation
    Jin Li, Chongguang Chen, Peng Huang and Lee-Yuan Liu-Chen
    Molecular Pharmacology November 2001, 60 (5) 1064-1075; DOI: https://doi.org/10.1124/mol.60.5.1064
  • You have access
    Expression of α-Transducin in Chinese Hamster Ovary Cells Stably Transfected with the Human δ-Opioid Receptor Attenuates Chronic Opioid Agonist-Induced Adenylyl Cyclase Superactivation
    Marc Rubenzik, Eva Varga, Dagmar Stropova, William R. Roeske and Henry I. Yamamura
    Molecular Pharmacology November 2001, 60 (5) 1076-1082; DOI: https://doi.org/10.1124/mol.60.5.1076
  • You have access
    Anti-Inflammatory Effects of the Partially Purified Extract of Radix Stephaniae tetrandrae: Comparative Studies of Its Active Principles Tetrandrine and Fangchinoline on Human Polymorphonuclear Leukocyte Functions
    Yuh-Chiang Shen, Cheng-Jen Chou, Wen-Fei Chiou and Chieh-Fu Chen
    Molecular Pharmacology November 2001, 60 (5) 1083-1090; DOI: https://doi.org/10.1124/mol.60.5.1083
  • You have access
    Mercapturic Acids (N-AcetylcysteineS-Conjugates) as Endogenous Substrates for the Renal Organic Anion Transporter-1
    James M. Pombrio, Adam Giangreco, Liqiong Li, Michael F. Wempe, M. W. Anders, Douglas H. Sweet, John B. Pritchard and Nazzareno Ballatori
    Molecular Pharmacology November 2001, 60 (5) 1091-1099; DOI: https://doi.org/10.1124/mol.60.5.1091
  • You have access
    Phorbol 12-myristate 13-acetate Triggers the Protein Kinase A-Mediated Phosphorylation and Activation of the PDE4D5 cAMP Phosphodiesterase in Human Aortic Smooth Muscle Cells through a Route Involving Extracellular Signal Regulated Kinase (ERK)
    George Baillie, Simon J. MacKenzie and Miles D. Houslay
    Molecular Pharmacology November 2001, 60 (5) 1100-1111; DOI: https://doi.org/10.1124/mol.60.5.1100
  • You have access
    Mpl Ligand Increases P2Y1 Receptor Gene Expression in Megakaryocytes with No Concomitant Change in Platelet Response to ADP
    Béatrice Hechler, Paul Toselli, Catherine Ravanat, Christian Gachet and Katya Ravid
    Molecular Pharmacology November 2001, 60 (5) 1112-1120; DOI: https://doi.org/10.1124/mol.60.5.1112
  • You have access
    Block of Cloned Human T-Type Calcium Channels by Succinimide Antiepileptic Drugs
    Juan Carlos Gomora, Asif N. Daud, Marco Weiergräber and Edward Perez-Reyes
    Molecular Pharmacology November 2001, 60 (5) 1121-1132; DOI: https://doi.org/10.1124/mol.60.5.1121
  • You have access
    Histamine H1-Receptor Activation of Nuclear Factor-κB: Roles for Gβγ- and Gαq/11-Subunits in Constitutive and Agonist-Mediated Signaling
    Remko A. Bakker, Stefan B. J. Schoonus, Martine J. Smit, Henk Timmerman and Rob Leurs
    Molecular Pharmacology November 2001, 60 (5) 1133-1142; DOI: https://doi.org/10.1124/mol.60.5.1133
  • You have access
    Acquisition of Human Concentrative Nucleoside Transporter 2 (hCNT2) Activity by Gene Transfer Confers Sensitivity to Fluoropyrimidine Nucleosides in Drug-Resistant Leukemia Cells
    Thack T. Lang, Milada Selner, James D. Young and Carol E. Cass
    Molecular Pharmacology November 2001, 60 (5) 1143-1152; DOI: https://doi.org/10.1124/mol.60.5.1143
Back to top
PreviousNext

In this issue

Molecular Pharmacology: 60 (5)
Molecular Pharmacology
Vol. 60, Issue 5
1 Nov 2001
  • Table of Contents
  • About the Cover
  • Index by author
Sign up for alerts

Jump to

  • Perspective
  • Articles
  • Most Read
Loading
  • How Many G Protein-Coupled Receptors are Drug Targets?
  • Nelfinavir and PXR
  • Wnt Signaling and Drug Resistance in Cancer
  • Coronavirus in the Brain and the Impact of Smoking
  • Arginine-259 of UGT2B7 Confers UDP-Sugar Selectivity
More...
Advertisement
  • Home
  • Alerts
Facebook   Twitter   LinkedIn   RSS

Navigate

  • Current Issue
  • Fast Forward by date
  • Fast Forward by section
  • Latest Articles
  • Archive
  • Search for Articles
  • Feedback
  • ASPET

More Information

  • About Molecular Pharmacology
  • Editorial Board
  • Instructions to Authors
  • Submit a Manuscript
  • Customized Alerts
  • RSS Feeds
  • Subscriptions
  • Permissions
  • Terms & Conditions of Use

ASPET's Other Journals

  • Drug Metabolism and Disposition
  • Journal of Pharmacology and Experimental Therapeutics
  • Pharmacological Reviews
  • Pharmacology Research & Perspectives
ISSN 1521-0111 (Online)

Copyright © 2021 by the American Society for Pharmacology and Experimental Therapeutics