Molecular Pharmacology: 60 (6)

December 01, 2001; Volume 60,Issue 6

MINIREVIEW

You have access
Identification of Genes That Mediate Sensitivity to Cisplatin
H. Niedner, R. Christen, X. Lin, A. Kondo and S. B. Howell

Molecular Pharmacology December 2001, 60 (6) 1153-1160; DOI: https://doi.org/10.1124/mol.60.6.1153

Perspectives

You have access
Selective Ligands for Lysophosphatidic Acid Receptor Subtypes: Gaining Control over the Endothelial Differentiation Gene Family
Gabor Tigyi

Molecular Pharmacology December 2001, 60 (6) 1161-1164; DOI: https://doi.org/10.1124/mol.60.6.1161
You have access
Old Drugs Learn New Tricks: Insights from Mammalian Trace Amine Receptors
Kyung-Ah Kim and Mark von Zastrow

Molecular Pharmacology December 2001, 60 (6) 1165-1167; DOI: https://doi.org/10.1124/mol.60.6.1165

Accelerated Communications

You have access
Dopamine D₂ Receptor-Induced Heterologous Sensitization of Adenylyl Cyclase Requires Gα_s: Characterization of Gα_s-Insensitive Mutants of Adenylyl Cyclase V
Val J. Watts, Ronald Taussig, Rachael L. Neve and Kim A. Neve

Molecular Pharmacology December 2001, 60 (6) 1168-1172; DOI: https://doi.org/10.1124/mol.60.6.1168
You have access
Activity of 2-Substituted Lysophosphatidic Acid (LPA) Analogs at LPA Receptors: Discovery of a LPA₁/LPA₃Receptor Antagonist
Christopher E. Heise, Webster L. Santos, Ann M. Schreihofer, Brian H. Heasley, Yurii V. Mukhin, Timothy L. Macdonald and Kevin R. Lynch

Molecular Pharmacology December 2001, 60 (6) 1173-1180; DOI: https://doi.org/10.1124/mol.60.6.1173
You have access
Amphetamine, 3,4-Methylenedioxymethamphetamine, Lysergic Acid Diethylamide, and Metabolites of the Catecholamine Neurotransmitters Are Agonists of a Rat Trace Amine Receptor
James R. Bunzow, Mark S. Sonders, Seksiri Arttamangkul, Laura M. Harrison, Ge Zhang, Denise I. Quigley, Tristan Darland, Katherine L. Suchland, Shailaja Pasumamula, James L. Kennedy, Susan B. Olson, R. Ellen Magenis, Susan G. Amara and David K. Grandy

Molecular Pharmacology December 2001, 60 (6) 1181-1188; DOI: https://doi.org/10.1124/mol.60.6.1181
You have access
Identification of toxicologically predictive gene sets using cDNA microarrays
Russell S. Thomas, David R. Rank, Sharron G. Penn, Gina M. Zastrow, Kevin R. Hayes, Kalyan Pande, Edward Glover, Tomi Silander, Mark W. Craven, Janardan K. Reddy, Stevan B. Jovanovich and Christopher A. Bradfield

Molecular Pharmacology December 2001, 60 (6) 1189-1194; DOI: https://doi.org/10.1124/mol.60.6.1189
You have access
Cooling Evokes Redistribution of α_2C-Adrenoceptors from Golgi to Plasma Membrane in Transfected Human Embryonic Kidney 293 Cells
Selvi C. Jeyaraj, Maqsood A. Chotani, Srabani Mitra, Herbert E. Gregg, Nicholas A. Flavahan and Keith J. Morrison

Molecular Pharmacology December 2001, 60 (6) 1195-1200; DOI: https://doi.org/10.1124/mol.60.6.1195

Articles

You have access
Human Bronchial Epithelial and Endothelial Cells Express α7 Nicotinic Acetylcholine Receptors
Y. Wang, E. F. R. Pereira, A. D. J. Maus, N. S. Ostlie, D. Navaneetham, S. Lei, E. X. Albuquerque and B. M. Conti-Fine

Molecular Pharmacology December 2001, 60 (6) 1201-1209; DOI: https://doi.org/10.1124/mol.60.6.1201
You have access
Distinct Interaction of Human and Guinea Pig Histamine H₂-Receptor with Guanidine-Type Agonists
Melissa T. Kelley, Tilmann Bürckstümmer, Katharina Wenzel-Seifert, Stefan Dove, Armin Buschauer and Roland Seifert

Molecular Pharmacology December 2001, 60 (6) 1210-1225; DOI: https://doi.org/10.1124/mol.60.6.1210
You have access
Interactions between Collagen IV and Collagen-Binding Integrins in Renal Cell Repair after Sublethal Injury
Paul A. Nony and Rick G. Schnellmann

Molecular Pharmacology December 2001, 60 (6) 1226-1234; DOI: https://doi.org/10.1124/mol.60.6.1226
You have access
A New Bis-Indole, KARs, Induces Selective M Arrest with Specific Spindle Aberration in Neuroblastoma Cell Line SH-SY5Y
Begoña Comı́n-Anduix, Neus Agell, Oriol Bachs, Judit Ovádi and Marta Cascante

Molecular Pharmacology December 2001, 60 (6) 1235-1242; DOI: https://doi.org/10.1124/mol.60.6.1235
You have access
Agonist-Stimulated and Tonic Internalization of Metabotropic Glutamate Receptor 1a in Human Embryonic Kidney 293 Cells: Agonist-Stimulated Endocytosis Is β-Arrestin1 Isoform-Specific
Lianne B. Dale, Moshmi Bhattacharya, Jennifer L. Seachrist, Pieter H. Anborgh and Stephen S. G. Ferguson

Molecular Pharmacology December 2001, 60 (6) 1243-1253; DOI: https://doi.org/10.1124/mol.60.6.1243
You have access
Anticancer Agent E7070 Inhibits Amino Acid and Uracil Transport in Fission Yeast
Kappei Tsukahara, Tatsuo Watanabe, Naoko Hata-Sugi, Kentaro Yoshimatsu, Hiroto Okayama and Takeshi Nagasu

Molecular Pharmacology December 2001, 60 (6) 1254-1259; DOI: https://doi.org/10.1124/mol.60.6.1254
You have access
The CYP2D6 Humanized Mouse: Effect of the HumanCYP2D6 Transgene and HNF4α on the Disposition of Debrisoquine in the Mouse
Javier Corchero, Camille P. Granvil, Taro E. Akiyama, Graham P. Hayhurst, Satish Pimprale, Lionel Feigenbaum, Jeffrey R. Idle and Frank J. Gonzalez

Molecular Pharmacology December 2001, 60 (6) 1260-1267; DOI: https://doi.org/10.1124/mol.60.6.1260
You have access
Cyclophosphamide Induces Caspase 9-Dependent Apoptosis in 9L Tumor Cells
Pamela S. Schwartz and David J. Waxman

Molecular Pharmacology December 2001, 60 (6) 1268-1279; DOI: https://doi.org/10.1124/mol.60.6.1268
You have access
Role of Aspartate7.32(302) of the Human Gonadotropin-Releasing Hormone Receptor in Stabilizing a High-Affinity Ligand Conformation
Bernhard J. Fromme, Arieh A. Katz, Roger W. Roeske, Robert P. Millar and Colleen A. Flanagan

Molecular Pharmacology December 2001, 60 (6) 1280-1287; DOI: https://doi.org/10.1124/mol.60.6.1280
You have access
Impact of Extracellular Folate Levels on Global Gene Expression
Mona S. Jhaveri, Conrad Wagner and Jane B. Trepel

Molecular Pharmacology December 2001, 60 (6) 1288-1295; DOI: https://doi.org/10.1124/mol.60.6.1288
You have access
Inhibition of Potentially Anti-Apoptotic Proteins by Antisense Protein Kinase C-α (Isis 3521) and Antisense bcl-2 (G3139) Phosphorothioate Oligodeoxynucleotides: Relationship to the Decreased Viability of T24 Bladder and PC3 Prostate Cancer Cells
Luba Benimetskaya, Paul Miller, Simon Benimetsky, Anna Maciaszek, Piotr Guga, Serge L. Beaucage, Andrzej Wilk, Andrzej Grajkowski, Anthony L. Halperin and C. A. Stein

Molecular Pharmacology December 2001, 60 (6) 1296-1307; DOI: https://doi.org/10.1124/mol.60.6.1296
You have access
Agonist-Mediated Down-Regulation of Rat β₁-Adrenergic Receptor Transcripts: Role of Potential Post-Transcriptional Degradation Factors
Philbert Kirigiti, Ying Bai, Yong-Feng Yang, Xiaorong Li, Biao Li, Gary Brewer and Curtis A. Machida

Molecular Pharmacology December 2001, 60 (6) 1308-1324; DOI: https://doi.org/10.1124/mol.60.6.1308
You have access
14-3-3 Inhibits Bad-Induced Cell Death through Interaction with Serine-136
Shane C. Masters, Hongzhu Yang, Sandeep Robert Datta, Michael E. Greenberg and Haian Fu

Molecular Pharmacology December 2001, 60 (6) 1325-1331; DOI: https://doi.org/10.1124/mol.60.6.1325
You have access
Transcriptional Mechanism of Protein Kinase C-Induced Isoform-Specific Expression of the Gene for Endothelin-Converting Enzyme-1in Human Endothelial Cells
Hans-Dieter Orzechowski, Astrid Günther, Stefan Menzel, Andreas Zimmermann, Heiko Funke-Kaiser, Robert Real, Thomas Subkowski, Frank S. Zollmann and Martin Paul

Molecular Pharmacology December 2001, 60 (6) 1332-1342; DOI: https://doi.org/10.1124/mol.60.6.1332
You have access
Molecular Determinants of Inactivation and Dofetilide Block inether a-go-go (EAG) Channels and EAG-Related K⁺ Channels
Eckhard Ficker, Wolfgang Jarolimek and Arthur M. Brown

Molecular Pharmacology December 2001, 60 (6) 1343-1348; DOI: https://doi.org/10.1124/mol.60.6.1343
You have access
Allosteric Modulation of the Human 5-HT_7A Receptor by Lipidic Amphipathic Compounds
Glen L. Alberts, Christopher L. Chio and Wha Bin Im

Molecular Pharmacology December 2001, 60 (6) 1349-1355; DOI: https://doi.org/10.1124/mol.60.6.1349
You have access
Ryanodine Receptor Dysfunction in Hearts of Streptozotocin-Induced Diabetic Rats
Keshore R. Bidasee, Ü. Deniz Dinçer and Henry R. Besch

Molecular Pharmacology December 2001, 60 (6) 1356-1364; DOI: https://doi.org/10.1124/mol.60.6.1356
You have access
Inhibition of Wild-Type and Mutant Neuronal Nicotinic Acetylcholine Receptors by Local Anesthetics
Roger L. Papke, Benjamin A. Horenstein and Andon N. Placzek

Molecular Pharmacology December 2001, 60 (6) 1365-1374; DOI: https://doi.org/10.1124/mol.60.6.1365
You have access
An Arginine/Glutamine Difference at the Juxtaposition of Transmembrane Domain 6 and the Third Extracellular Loop Contributes to the Markedly Different Nucleotide Selectivities of Human and Canine P2Y₁₁ Receptors
Ai-Dong Qi, Alexander C. Zambon, Paul A. Insel and Robert A. Nicholas

Molecular Pharmacology December 2001, 60 (6) 1375-1382; DOI: https://doi.org/10.1124/mol.60.6.1375
You have access
Induction of Cyclin E and Inhibition of DNA Synthesis by the Novel Acronycine Derivative S23906-1 Precede the Irreversible Arrest of Tumor Cells in S Phase Leading to Apoptosis
Stéphane Léonce, Valérie Pérez, Stéphanie Lambel, Delphine Peyroulan, François Tillequin, Sylvie Michel, Michel Koch, Bruno Pfeiffer, Ghanem Atassi, John A Hickman and Alain Pierré

Molecular Pharmacology December 2001, 60 (6) 1383-1391; DOI: https://doi.org/10.1124/mol.60.6.1383
You have access
Agonism, Inverse Agonism, and Neutral Antagonism at the Constitutively Active Human Neurotensin Receptor 2
Françoise Richard, Séverine Barroso, Jean Martinez, Catherine Labbé-Jullié and Patrick Kitabgi

Molecular Pharmacology December 2001, 60 (6) 1392-1398; DOI: https://doi.org/10.1124/mol.60.6.1392
You have access
Transcriptional Control of Intestinal Cytochrome P-4503A by 1α,25-Dihydroxy Vitamin D₃
Kenneth E. Thummel, Cynthia Brimer, Kazuto Yasuda, Jaideep Thottassery, Tauri Senn, Yvonne Lin, Hitoshi Ishizuka, Evan Kharasch, John Schuetz and Erin Schuetz

Molecular Pharmacology December 2001, 60 (6) 1399-1406; DOI: https://doi.org/10.1124/mol.60.6.1399
You have access
O-Acetylsalicylhydroxamic Acid, a Novel Acetylating Inhibitor of Prostaglandin H₂ Synthase: Structural and Functional Characterization of Enzyme-Inhibitor Interactions
P. J. Loll, C. T. Sharkey, S. J. O'Connor, C. M. Dooley, E. O'Brien, M. Devocelle, K. B. Nolan, B. S. Selinsky and D. J. Fitzgerald

Molecular Pharmacology December 2001, 60 (6) 1407-1413; DOI: https://doi.org/10.1124/mol.60.6.1407
You have access
ALX 5407: A Potent, Selective Inhibitor of the hGlyT1 Glycine Transporter
B. N. Atkinson, S. C. Bell, M. De Vivo, L. R. Kowalski, S. M. Lechner, V. I. Ognyanov, C.-S. Tham, C. Tsai, J. Jia, D. Ashton and M. A. Klitenick

Molecular Pharmacology December 2001, 60 (6) 1414-1420; DOI: https://doi.org/10.1124/mol.60.6.1414
You have access
Regulation of Flavin-Containing Monooxygenase 1 Expression by Ying Yang 1 and Hepatic Nuclear Factors 1 and 4
Zhaohui Luo and Ronald N. Hines

Molecular Pharmacology December 2001, 60 (6) 1421-1430; DOI: https://doi.org/10.1124/mol.60.6.1421
You have access
Negative Regulation of the SHPTP1 Protein Tyrosine Phosphatase by Protein Kinase C δ in Response to DNA Damage
Kiyotsugu Yoshida and Donald Kufe

Molecular Pharmacology December 2001, 60 (6) 1431-1438; DOI: https://doi.org/10.1124/mol.60.6.1431
You have access
Conjugated Polyhydroxybenzene Derivatives Block Tumor Necrosis Factor-α–Mediated Nuclear Factor-κB Activation and Cyclooxygenase-2 Gene Transcription by Targeting IκB Kinase Activity
Ching-Chow Chen, Kuo-Tung Chiu, Shu-Ting Chan and Ji-Wang Chern

Molecular Pharmacology December 2001, 60 (6) 1439-1448; DOI: https://doi.org/10.1124/mol.60.6.1439

Main menu

User menu

Search

Table of Contents

MINIREVIEW

Perspectives

Accelerated Communications

Articles

In this issue

Jump to

Navigate

More Information

ASPET's Other Journals