Molecular Pharmacology: 61 (5)

May 01, 2002; Volume 61,Issue 5

Accelerated Communication

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G Protein-Coupled Receptors as Direct Targets of Inhaled Anesthetics
Yumiko Ishizawa, Ravindernath Pidikiti, Paul A. Liebman and Roderic G. Eckenhoff

Molecular Pharmacology May 2002, 61 (5) 945-952; DOI: https://doi.org/10.1124/mol.61.5.945

Articles

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Parthenolide, an Inhibitor of the Nuclear Factor-κB Pathway, Ameliorates Cardiovascular Derangement and Outcome in Endotoxic Shock in Rodents
Maeve Sheehan, Hector R. Wong, Paul W. Hake, Vivek Malhotra, Michael O'Connor and Basilia Zingarelli

Molecular Pharmacology May 2002, 61 (5) 953-963; DOI: https://doi.org/10.1124/mol.61.5.953
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Three-Dimensional Quantitative Structure-Activity Relationships of Inhibitors of P-Glycoprotein
Sean Ekins, Richard B. Kim, Brenda F. Leake, Anne H. Dantzig, Erin G. Schuetz, Lu-Bin Lan, Kazuto Yasuda, Robert L. Shepard, Mark A. Winter, John D. Schuetz, James H. Wikel and Steven A. Wrighton

Molecular Pharmacology May 2002, 61 (5) 964-973; DOI: https://doi.org/10.1124/mol.61.5.964
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Application of Three-Dimensional Quantitative Structure-Activity Relationships of P-Glycoprotein Inhibitors and Substrates
Sean Ekins, Richard B. Kim, Brenda F. Leake, Anne H. Dantzig, Erin G. Schuetz, Lu-Bin Lan, Kazuto Yasuda, Robert L. Shepard, Mark a Winter, John D. Schuetz, James H. Wikel and Steven A. Wrighton

Molecular Pharmacology May 2002, 61 (5) 974-981; DOI: https://doi.org/10.1124/mol.61.5.974
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Expression and Functional Characterization of Rat Organic Anion Transporter 3 (rOat3) in the Choroid Plexus
Yoshinori Nagata, Hiroyuki Kusuhara, Hitoshi Endou and Yuichi Sugiyama

Molecular Pharmacology May 2002, 61 (5) 982-988; DOI: https://doi.org/10.1124/mol.61.5.982
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l-Acetylcarnitine Induces Analgesia by Selectively Up-Regulating mGlu2 Metabotropic Glutamate Receptors
S. Chiechio, A. Caricasole, E. Barletta, M. Storto, M. V. Catania, A. Copani, M. Vertechy, R. Nicolai, M. Calvani, D. Melchiorri and F. Nicoletti

Molecular Pharmacology May 2002, 61 (5) 989-996; DOI: https://doi.org/10.1124/mol.61.5.989
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The Cyclopentenone Prostaglandin 15-Deoxy-Δ^12,14-Prostaglandin J₂Attenuates the Development of Acute and Chronic Inflammation
Salvatore Cuzzocrea, Nicole S. Wayman, Emanuela Mazzon, Laura Dugo, Rosanna Di Paola, Ivana Serraino, Domenico Britti, Prabal K. Chatterjee, Achille P. Caputi and Christoph Thiemermann

Molecular Pharmacology May 2002, 61 (5) 997-1007; DOI: https://doi.org/10.1124/mol.61.5.997
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Differences in the Cellular Localization and Agonist-Mediated Internalization Properties of the α₁-Adrenoceptor Subtypes
Dan Chalothorn, Dan F. McCune, Stephanie E. Edelmann, Mary L. Garcı́a-Cazarı́n, Gozoh Tsujimoto and Michael T. Piascik

Molecular Pharmacology May 2002, 61 (5) 1008-1016; DOI: https://doi.org/10.1124/mol.61.5.1008
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Antidepressant Treatments Induce the Expression of Basic Fibroblast Growth Factor in Cortical and Hippocampal Neurons
Alessandra Mallei, Bitao Shi and Italo Mocchetti

Molecular Pharmacology May 2002, 61 (5) 1017-1024; DOI: https://doi.org/10.1124/mol.61.5.1017
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Mutagenesis and Modelling of the α_1b-Adrenergic Receptor Highlight the Role of the Helix 3/Helix 6 Interface in Receptor Activation
Peter J. Greasley, Francesca Fanelli, Olivier Rossier, Liliane Abuin and Susanna Cotecchia

Molecular Pharmacology May 2002, 61 (5) 1025-1032; DOI: https://doi.org/10.1124/mol.61.5.1025
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Reduced Phosphodiesterase 3 Activity and Phosphodiesterase 3A Level in Synthetic Vascular Smooth Muscle Cells: Implications for Use of Phosphodiesterase 3 Inhibitors in Cardiovascular Tissues
Heather A. Dunkerley, Douglas G. Tilley, Daniel Palmer, Hanguan Liu, Sandra L. Jimmo and Donald H. Maurice

Molecular Pharmacology May 2002, 61 (5) 1033-1040; DOI: https://doi.org/10.1124/mol.61.5.1033
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Refinement of the Conformation of a Critical Region of Charge-Charge Interaction between Cholecystokinin and Its Receptor
Xi-Qin Ding, Delia I. Pinon, Kristina E. Furse, Terry P. Lybrand and Laurence J. Miller

Molecular Pharmacology May 2002, 61 (5) 1041-1052; DOI: https://doi.org/10.1124/mol.61.5.1041
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2-Methoxyestradiol and Analogs as Novel Antiproliferative Agents: Analysis of Three-Dimensional Quantitative Structure-Activity Relationships for DNA Synthesis Inhibition and Estrogen Receptor Binding
Richard A. Hughes, Trudi Harris, Emile Altmann, David McAllister, Ross Vlahos, Alan Robertson, Mark Cushman, Zhiqiang Wang and Alastair G. Stewart

Molecular Pharmacology May 2002, 61 (5) 1053-1069; DOI: https://doi.org/10.1124/mol.61.5.1053
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Importance of the γ-Aminobutyric Acid_B Receptor C-Termini for G-Protein Coupling
Sylvia Grünewald, Bettina J. Schupp, Stephen R. Ikeda, Rohini Kuner, Frank Steigerwald, Hans-Christian Kornau and Georg Köhr

Molecular Pharmacology May 2002, 61 (5) 1070-1080; DOI: https://doi.org/10.1124/mol.61.5.1070
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Functional and Analytical Evidence for Scavenging of Oxygen Radicals by l-Arginine
Achim Lass, Astrid Suessenbacher, Gerald Wölkart, Bernd Mayer and Friedrich Brunner

Molecular Pharmacology May 2002, 61 (5) 1081-1088; DOI: https://doi.org/10.1124/mol.61.5.1081
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Post-Transcriptional Regulation of Hepatic NADPH-Cytochrome P450 Reductase by Thyroid Hormone: Independent Effects on Poly(A) Tail Length and mRNA Stability
Dongxu Liu and David J. Waxman

Molecular Pharmacology May 2002, 61 (5) 1089-1096; DOI: https://doi.org/10.1124/mol.61.5.1089
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Up-Regulation of Glutamate Receptors in Nucleus Tractus Solitarii Underlies Potentiation of Baroreceptor Reflex by Heat Shock Protein 70
Samuel H. H. Chan, Kui-Fen Chang, Chen-Chun Ou and Julie Y. H. Chan

Molecular Pharmacology May 2002, 61 (5) 1097-1104; DOI: https://doi.org/10.1124/mol.61.5.1097
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Ethylbromide Tamoxifen, a Membrane-Impermeant Antiestrogen, Activates Smooth Muscle Calcium-Activated Large-Conductance Potassium Channels from the Extracellular Side
Gregory M. Dick, A. Christy Hunter and Kenton M. Sanders

Molecular Pharmacology May 2002, 61 (5) 1105-1113; DOI: https://doi.org/10.1124/mol.61.5.1105
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Metabotropic Glutamate Receptor 1 Internalization Induced by Muscarinic Acetylcholine Receptor Activation: Differential Dependency of Internalization of Splice Variants on Nonvisual Arrestins
Stuart J. Mundell, Anne-Lise Matharu, Giordano Pula, David Holman, Peter J. Roberts and Eamonn Kelly

Molecular Pharmacology May 2002, 61 (5) 1114-1123; DOI: https://doi.org/10.1124/mol.61.5.1114
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Methamphetamine Causes Coordinate Regulation of Src, Cas, Crk, and the Jun N-Terminal Kinase–Jun Pathway
Subramaniam Jayanthi, Michael T. McCoy, Bruce Ladenheim and Jean Lud Cadet

Molecular Pharmacology May 2002, 61 (5) 1124-1131; DOI: https://doi.org/10.1124/mol.61.5.1124
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Five Amino Acids of the Xenopus laevis CRF (Corticotropin-Releasing Factor) Type 2 Receptor Mediate Differential Binding of CRF Ligands in Comparison with Its Human Counterpart
Frank M. Dautzenberg, Jacqueline Higelin, Olaf Brauns, Brigitte Butscha and Richard L. Hauger

Molecular Pharmacology May 2002, 61 (5) 1132-1139; DOI: https://doi.org/10.1124/mol.61.5.1132
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Lack of Susceptibility of Bicyclic Nucleoside Analogs, Highly Potent Inhibitors of Varicella-Zoster Virus, to the Catabolic Action of Thymidine Phosphorylase and Dihydropyrimidine Dehydrogenase
Jan Balzarini, Rebecca Sienaert, Sandra Liekens, André Van Kuilenburg, Antonella Carangio, Robert Esnouf, Erik De Clercq and Chris McGuigan

Molecular Pharmacology May 2002, 61 (5) 1140-1145; DOI: https://doi.org/10.1124/mol.61.5.1140
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Native CYP2C11: Heterologous Expression in Saccharomyces cerevisiae Reveals a Role for Vacuolar Proteases Rather Than the Proteasome System in the Degradation of This Endoplasmic Reticulum Protein
Bernard P. Murray, Victor G. Zgoda and Maria Almira Correia

Molecular Pharmacology May 2002, 61 (5) 1146-1153; DOI: https://doi.org/10.1124/mol.61.5.1146
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A G-Quadruplex-Interactive Potent Small-Molecule Inhibitor of Telomerase Exhibiting in Vitro and in Vivo Antitumor Activity
Sharon M. Gowan, John R. Harrison, Lisa Patterson, Melanie Valenti, Martin A. Read, Stephen Neidle and Lloyd R. Kelland

Molecular Pharmacology May 2002, 61 (5) 1154-1162; DOI: https://doi.org/10.1124/mol.61.5.1154
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Regulation of Fibronectin Fibrillogenesis by Protein Kinases in Cultured Rat Osteoblasts
Rong-Sen Yang, Chih-Hsin Tang, Qing-Dong Ling, Shing-Hwa Liu and Wen-Mei Fu

Molecular Pharmacology May 2002, 61 (5) 1163-1173; DOI: https://doi.org/10.1124/mol.61.5.1163
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Identification of Albumin Precursor Protein, Phi AP3, and α-Smooth Muscle Actin as Novel Components of Redox Sensing Machinery in Vascular Smooth Muscle Cells
M. T. Holderman, K. P. Miller, L. J. Dangott and K. S. Ramos

Molecular Pharmacology May 2002, 61 (5) 1174-1183; DOI: https://doi.org/10.1124/mol.61.5.1174
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Substrate-Induced Up-Regulation of Aldose Reductase by Methylglyoxal, a Reactive Oxoaldehyde Elevated in Diabetes
Ki Churl Chang, Kyung Shin Paek, Hyo Jung Kim, Young Soo Lee, Chihiro Yabe-Nishimura and Han Geuk Seo

Molecular Pharmacology May 2002, 61 (5) 1184-1191; DOI: https://doi.org/10.1124/mol.61.5.1184
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Critical Molecular Determinants of Voltage-Gated Sodium Channel Sensitivity to μ-Conotoxins GIIIA/B
Theodore R. Cummins, Fabio Aglieco and Sulayman D. Dib-Hajj

Molecular Pharmacology May 2002, 61 (5) 1192-1201; DOI: https://doi.org/10.1124/mol.61.5.1192
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The Critical Role of Transmembrane Prolines in Human Prostacyclin Receptor Activation
Jeremiah Stitham, Kathleen A. Martin and John Hwa

Molecular Pharmacology May 2002, 61 (5) 1202-1210; DOI: https://doi.org/10.1124/mol.61.5.1202
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Enhanced Detection of Receptor Constitutive Activity in the Presence of Regulators of G Protein Signaling: Applications to the Detection and Analysis of Inverse Agonists and Low-Efficacy Partial Agonists
Philip J. Welsby, Elaine Kellett, Graeme Wilkinson and Graeme Milligan

Molecular Pharmacology May 2002, 61 (5) 1211-1221; DOI: https://doi.org/10.1124/mol.61.5.1211
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The Nicotinic Allosteric Potentiating Ligand Galantamine Facilitates Synaptic Transmission in the Mammalian Central Nervous System
Máriton D. Santos, Manickavasagom Alkondon, Edna F. R. Pereira, Yasco Aracava, Howard M. Eisenberg, Alfred Maelicke and Edson X. Albuquerque

Molecular Pharmacology May 2002, 61 (5) 1222-1234; DOI: https://doi.org/10.1124/mol.61.5.1222
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Maleimide Is a Potent Inhibitor of Topoisomerase II in Vitro and in Vivo: A New Mode of Catalytic Inhibition
Lars H. Jensen, Axelle Renodon-Corniere, Irene Wessel, Seppo W. Langer, Birgitte Søkilde, Elisabeth V. Carstensen, Maxwell Sehested and Peter B. Jensen

Molecular Pharmacology May 2002, 61 (5) 1235-1243; DOI: https://doi.org/10.1124/mol.61.5.1235
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Supersensitivity of Human Metabotropic Glutamate 1a Receptor Signaling in L929sA Cells
Hilde Lavreysen, Emmanuel Le Poul, Paul Van Gompel, Lieve Dillen, Josée E. Leysen and Anne S. J. Lesage

Molecular Pharmacology May 2002, 61 (5) 1244-1254; DOI: https://doi.org/10.1124/mol.61.5.1244
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Further Insight into Mechanism of Action of Clodronate: Inhibition of Mitochondrial ADP/ATP Translocase by a Nonhydrolyzable, Adenine-Containing Metabolite
Petri P. Lehenkari, Maarit Kellinsalmi, Juha P. Näpänkangas, Kari V. Ylitalo, Jukka Mönkkönen, Michael J. Rogers, Alex Azhayev, H. Kalervo Väänänen and Ilmo E. Hassinen

Molecular Pharmacology May 2002, 61 (5) 1255-1262; DOI: https://doi.org/10.1124/mol.61.5.1255

Errata

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Correction to “Antitumor Activity of 2′,3′-Dideoxycytidine Nucleotide Analog Against Tumors Up-Regulating DNA Polymerase β”
Molecular Pharmacology May 2002, 61 (5) 1263; DOI: https://doi.org/10.1124/mol.61.5.1263
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Correction to “Caffeic Acid Phenethyl Ester and Curcumin: A Novel Class of Heme Oxygenase-1 Inducers”
Molecular Pharmacology May 2002, 61 (5) 1264; DOI: https://doi.org/10.1124/mol.61.5.1264
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Correction to “Novel “Nonkinase” Phorbol Ester Receptors: The C1 Domain Connection”
Molecular Pharmacology May 2002, 61 (5) 1265; DOI: https://doi.org/10.1124/mol.61.5.1265

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