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Molecular Pharmacology

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Table of Contents

May 01, 2002; Volume 61,Issue 5

Accelerated Communication

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    G Protein-Coupled Receptors as Direct Targets of Inhaled Anesthetics
    Yumiko Ishizawa, Ravindernath Pidikiti, Paul A. Liebman and Roderic G. Eckenhoff
    Molecular Pharmacology May 2002, 61 (5) 945-952; DOI: https://doi.org/10.1124/mol.61.5.945

Articles

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    Parthenolide, an Inhibitor of the Nuclear Factor-κB Pathway, Ameliorates Cardiovascular Derangement and Outcome in Endotoxic Shock in Rodents
    Maeve Sheehan, Hector R. Wong, Paul W. Hake, Vivek Malhotra, Michael O'Connor and Basilia Zingarelli
    Molecular Pharmacology May 2002, 61 (5) 953-963; DOI: https://doi.org/10.1124/mol.61.5.953
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    Three-Dimensional Quantitative Structure-Activity Relationships of Inhibitors of P-Glycoprotein
    Sean Ekins, Richard B. Kim, Brenda F. Leake, Anne H. Dantzig, Erin G. Schuetz, Lu-Bin Lan, Kazuto Yasuda, Robert L. Shepard, Mark A. Winter, John D. Schuetz, James H. Wikel and Steven A. Wrighton
    Molecular Pharmacology May 2002, 61 (5) 964-973; DOI: https://doi.org/10.1124/mol.61.5.964
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    Application of Three-Dimensional Quantitative Structure-Activity Relationships of P-Glycoprotein Inhibitors and Substrates
    Sean Ekins, Richard B. Kim, Brenda F. Leake, Anne H. Dantzig, Erin G. Schuetz, Lu-Bin Lan, Kazuto Yasuda, Robert L. Shepard, Mark a Winter, John D. Schuetz, James H. Wikel and Steven A. Wrighton
    Molecular Pharmacology May 2002, 61 (5) 974-981; DOI: https://doi.org/10.1124/mol.61.5.974
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    Expression and Functional Characterization of Rat Organic Anion Transporter 3 (rOat3) in the Choroid Plexus
    Yoshinori Nagata, Hiroyuki Kusuhara, Hitoshi Endou and Yuichi Sugiyama
    Molecular Pharmacology May 2002, 61 (5) 982-988; DOI: https://doi.org/10.1124/mol.61.5.982
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    l-Acetylcarnitine Induces Analgesia by Selectively Up-Regulating mGlu2 Metabotropic Glutamate Receptors
    S. Chiechio, A. Caricasole, E. Barletta, M. Storto, M. V. Catania, A. Copani, M. Vertechy, R. Nicolai, M. Calvani, D. Melchiorri and F. Nicoletti
    Molecular Pharmacology May 2002, 61 (5) 989-996; DOI: https://doi.org/10.1124/mol.61.5.989
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    The Cyclopentenone Prostaglandin 15-Deoxy-Δ12,14-Prostaglandin J2Attenuates the Development of Acute and Chronic Inflammation
    Salvatore Cuzzocrea, Nicole S. Wayman, Emanuela Mazzon, Laura Dugo, Rosanna Di Paola, Ivana Serraino, Domenico Britti, Prabal K. Chatterjee, Achille P. Caputi and Christoph Thiemermann
    Molecular Pharmacology May 2002, 61 (5) 997-1007; DOI: https://doi.org/10.1124/mol.61.5.997
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    Differences in the Cellular Localization and Agonist-Mediated Internalization Properties of the α1-Adrenoceptor Subtypes
    Dan Chalothorn, Dan F. McCune, Stephanie E. Edelmann, Mary L. Garcı́a-Cazarı́n, Gozoh Tsujimoto and Michael T. Piascik
    Molecular Pharmacology May 2002, 61 (5) 1008-1016; DOI: https://doi.org/10.1124/mol.61.5.1008
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    Antidepressant Treatments Induce the Expression of Basic Fibroblast Growth Factor in Cortical and Hippocampal Neurons
    Alessandra Mallei, Bitao Shi and Italo Mocchetti
    Molecular Pharmacology May 2002, 61 (5) 1017-1024; DOI: https://doi.org/10.1124/mol.61.5.1017
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    Mutagenesis and Modelling of the α1b-Adrenergic Receptor Highlight the Role of the Helix 3/Helix 6 Interface in Receptor Activation
    Peter J. Greasley, Francesca Fanelli, Olivier Rossier, Liliane Abuin and Susanna Cotecchia
    Molecular Pharmacology May 2002, 61 (5) 1025-1032; DOI: https://doi.org/10.1124/mol.61.5.1025
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    Reduced Phosphodiesterase 3 Activity and Phosphodiesterase 3A Level in Synthetic Vascular Smooth Muscle Cells: Implications for Use of Phosphodiesterase 3 Inhibitors in Cardiovascular Tissues
    Heather A. Dunkerley, Douglas G. Tilley, Daniel Palmer, Hanguan Liu, Sandra L. Jimmo and Donald H. Maurice
    Molecular Pharmacology May 2002, 61 (5) 1033-1040; DOI: https://doi.org/10.1124/mol.61.5.1033
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    Refinement of the Conformation of a Critical Region of Charge-Charge Interaction between Cholecystokinin and Its Receptor
    Xi-Qin Ding, Delia I. Pinon, Kristina E. Furse, Terry P. Lybrand and Laurence J. Miller
    Molecular Pharmacology May 2002, 61 (5) 1041-1052; DOI: https://doi.org/10.1124/mol.61.5.1041
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    2-Methoxyestradiol and Analogs as Novel Antiproliferative Agents: Analysis of Three-Dimensional Quantitative Structure-Activity Relationships for DNA Synthesis Inhibition and Estrogen Receptor Binding
    Richard A. Hughes, Trudi Harris, Emile Altmann, David McAllister, Ross Vlahos, Alan Robertson, Mark Cushman, Zhiqiang Wang and Alastair G. Stewart
    Molecular Pharmacology May 2002, 61 (5) 1053-1069; DOI: https://doi.org/10.1124/mol.61.5.1053
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    Importance of the γ-Aminobutyric AcidB Receptor C-Termini for G-Protein Coupling
    Sylvia Grünewald, Bettina J. Schupp, Stephen R. Ikeda, Rohini Kuner, Frank Steigerwald, Hans-Christian Kornau and Georg Köhr
    Molecular Pharmacology May 2002, 61 (5) 1070-1080; DOI: https://doi.org/10.1124/mol.61.5.1070
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    Functional and Analytical Evidence for Scavenging of Oxygen Radicals by l-Arginine
    Achim Lass, Astrid Suessenbacher, Gerald Wölkart, Bernd Mayer and Friedrich Brunner
    Molecular Pharmacology May 2002, 61 (5) 1081-1088; DOI: https://doi.org/10.1124/mol.61.5.1081
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    Post-Transcriptional Regulation of Hepatic NADPH-Cytochrome P450 Reductase by Thyroid Hormone: Independent Effects on Poly(A) Tail Length and mRNA Stability
    Dongxu Liu and David J. Waxman
    Molecular Pharmacology May 2002, 61 (5) 1089-1096; DOI: https://doi.org/10.1124/mol.61.5.1089
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    Up-Regulation of Glutamate Receptors in Nucleus Tractus Solitarii Underlies Potentiation of Baroreceptor Reflex by Heat Shock Protein 70
    Samuel H. H. Chan, Kui-Fen Chang, Chen-Chun Ou and Julie Y. H. Chan
    Molecular Pharmacology May 2002, 61 (5) 1097-1104; DOI: https://doi.org/10.1124/mol.61.5.1097
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    Ethylbromide Tamoxifen, a Membrane-Impermeant Antiestrogen, Activates Smooth Muscle Calcium-Activated Large-Conductance Potassium Channels from the Extracellular Side
    Gregory M. Dick, A. Christy Hunter and Kenton M. Sanders
    Molecular Pharmacology May 2002, 61 (5) 1105-1113; DOI: https://doi.org/10.1124/mol.61.5.1105
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    Metabotropic Glutamate Receptor 1 Internalization Induced by Muscarinic Acetylcholine Receptor Activation: Differential Dependency of Internalization of Splice Variants on Nonvisual Arrestins
    Stuart J. Mundell, Anne-Lise Matharu, Giordano Pula, David Holman, Peter J. Roberts and Eamonn Kelly
    Molecular Pharmacology May 2002, 61 (5) 1114-1123; DOI: https://doi.org/10.1124/mol.61.5.1114
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    Methamphetamine Causes Coordinate Regulation of Src, Cas, Crk, and the Jun N-Terminal Kinase–Jun Pathway
    Subramaniam Jayanthi, Michael T. McCoy, Bruce Ladenheim and Jean Lud Cadet
    Molecular Pharmacology May 2002, 61 (5) 1124-1131; DOI: https://doi.org/10.1124/mol.61.5.1124
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    Five Amino Acids of the Xenopus laevis CRF (Corticotropin-Releasing Factor) Type 2 Receptor Mediate Differential Binding of CRF Ligands in Comparison with Its Human Counterpart
    Frank M. Dautzenberg, Jacqueline Higelin, Olaf Brauns, Brigitte Butscha and Richard L. Hauger
    Molecular Pharmacology May 2002, 61 (5) 1132-1139; DOI: https://doi.org/10.1124/mol.61.5.1132
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    Lack of Susceptibility of Bicyclic Nucleoside Analogs, Highly Potent Inhibitors of Varicella-Zoster Virus, to the Catabolic Action of Thymidine Phosphorylase and Dihydropyrimidine Dehydrogenase
    Jan Balzarini, Rebecca Sienaert, Sandra Liekens, André Van Kuilenburg, Antonella Carangio, Robert Esnouf, Erik De Clercq and Chris McGuigan
    Molecular Pharmacology May 2002, 61 (5) 1140-1145; DOI: https://doi.org/10.1124/mol.61.5.1140
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    Native CYP2C11: Heterologous Expression in Saccharomyces cerevisiae Reveals a Role for Vacuolar Proteases Rather Than the Proteasome System in the Degradation of This Endoplasmic Reticulum Protein
    Bernard P. Murray, Victor G. Zgoda and Maria Almira Correia
    Molecular Pharmacology May 2002, 61 (5) 1146-1153; DOI: https://doi.org/10.1124/mol.61.5.1146
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    A G-Quadruplex-Interactive Potent Small-Molecule Inhibitor of Telomerase Exhibiting in Vitro and in Vivo Antitumor Activity
    Sharon M. Gowan, John R. Harrison, Lisa Patterson, Melanie Valenti, Martin A. Read, Stephen Neidle and Lloyd R. Kelland
    Molecular Pharmacology May 2002, 61 (5) 1154-1162; DOI: https://doi.org/10.1124/mol.61.5.1154
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    Regulation of Fibronectin Fibrillogenesis by Protein Kinases in Cultured Rat Osteoblasts
    Rong-Sen Yang, Chih-Hsin Tang, Qing-Dong Ling, Shing-Hwa Liu and Wen-Mei Fu
    Molecular Pharmacology May 2002, 61 (5) 1163-1173; DOI: https://doi.org/10.1124/mol.61.5.1163
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    Identification of Albumin Precursor Protein, Phi AP3, and α-Smooth Muscle Actin as Novel Components of Redox Sensing Machinery in Vascular Smooth Muscle Cells
    M. T. Holderman, K. P. Miller, L. J. Dangott and K. S. Ramos
    Molecular Pharmacology May 2002, 61 (5) 1174-1183; DOI: https://doi.org/10.1124/mol.61.5.1174
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    Substrate-Induced Up-Regulation of Aldose Reductase by Methylglyoxal, a Reactive Oxoaldehyde Elevated in Diabetes
    Ki Churl Chang, Kyung Shin Paek, Hyo Jung Kim, Young Soo Lee, Chihiro Yabe-Nishimura and Han Geuk Seo
    Molecular Pharmacology May 2002, 61 (5) 1184-1191; DOI: https://doi.org/10.1124/mol.61.5.1184
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    Critical Molecular Determinants of Voltage-Gated Sodium Channel Sensitivity to μ-Conotoxins GIIIA/B
    Theodore R. Cummins, Fabio Aglieco and Sulayman D. Dib-Hajj
    Molecular Pharmacology May 2002, 61 (5) 1192-1201; DOI: https://doi.org/10.1124/mol.61.5.1192
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    The Critical Role of Transmembrane Prolines in Human Prostacyclin Receptor Activation
    Jeremiah Stitham, Kathleen A. Martin and John Hwa
    Molecular Pharmacology May 2002, 61 (5) 1202-1210; DOI: https://doi.org/10.1124/mol.61.5.1202
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    Enhanced Detection of Receptor Constitutive Activity in the Presence of Regulators of G Protein Signaling: Applications to the Detection and Analysis of Inverse Agonists and Low-Efficacy Partial Agonists
    Philip J. Welsby, Elaine Kellett, Graeme Wilkinson and Graeme Milligan
    Molecular Pharmacology May 2002, 61 (5) 1211-1221; DOI: https://doi.org/10.1124/mol.61.5.1211
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    The Nicotinic Allosteric Potentiating Ligand Galantamine Facilitates Synaptic Transmission in the Mammalian Central Nervous System
    Máriton D. Santos, Manickavasagom Alkondon, Edna F. R. Pereira, Yasco Aracava, Howard M. Eisenberg, Alfred Maelicke and Edson X. Albuquerque
    Molecular Pharmacology May 2002, 61 (5) 1222-1234; DOI: https://doi.org/10.1124/mol.61.5.1222
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    Maleimide Is a Potent Inhibitor of Topoisomerase II in Vitro and in Vivo: A New Mode of Catalytic Inhibition
    Lars H. Jensen, Axelle Renodon-Corniere, Irene Wessel, Seppo W. Langer, Birgitte Søkilde, Elisabeth V. Carstensen, Maxwell Sehested and Peter B. Jensen
    Molecular Pharmacology May 2002, 61 (5) 1235-1243; DOI: https://doi.org/10.1124/mol.61.5.1235
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    Supersensitivity of Human Metabotropic Glutamate 1a Receptor Signaling in L929sA Cells
    Hilde Lavreysen, Emmanuel Le Poul, Paul Van Gompel, Lieve Dillen, Josée E. Leysen and Anne S. J. Lesage
    Molecular Pharmacology May 2002, 61 (5) 1244-1254; DOI: https://doi.org/10.1124/mol.61.5.1244
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    Further Insight into Mechanism of Action of Clodronate: Inhibition of Mitochondrial ADP/ATP Translocase by a Nonhydrolyzable, Adenine-Containing Metabolite
    Petri P. Lehenkari, Maarit Kellinsalmi, Juha P. Näpänkangas, Kari V. Ylitalo, Jukka Mönkkönen, Michael J. Rogers, Alex Azhayev, H. Kalervo Väänänen and Ilmo E. Hassinen
    Molecular Pharmacology May 2002, 61 (5) 1255-1262; DOI: https://doi.org/10.1124/mol.61.5.1255

Errata

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    Correction to “Antitumor Activity of 2′,3′-Dideoxycytidine Nucleotide Analog Against Tumors Up-Regulating DNA Polymerase β”
    Molecular Pharmacology May 2002, 61 (5) 1263; DOI: https://doi.org/10.1124/mol.61.5.1263
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    Correction to “Caffeic Acid Phenethyl Ester and Curcumin: A Novel Class of Heme Oxygenase-1 Inducers”
    Molecular Pharmacology May 2002, 61 (5) 1264; DOI: https://doi.org/10.1124/mol.61.5.1264
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    Correction to “Novel “Nonkinase” Phorbol Ester Receptors: The C1 Domain Connection”
    Molecular Pharmacology May 2002, 61 (5) 1265; DOI: https://doi.org/10.1124/mol.61.5.1265
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Molecular Pharmacology: 61 (5)
Molecular Pharmacology
Vol. 61, Issue 5
1 May 2002
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  • SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-β Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7
  • The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints
  • Pharmacological Properties of Y-27632, a Specific Inhibitor of Rho-Associated Kinases
  • Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
  • The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation of CYP3A4 by Rifampicin through a Distal Enhancer Module
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