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Molecular Pharmacology

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Table of Contents

January 01, 2003; Volume 63,Issue 1

ANNOUNCEMENT

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    Announcement
    Molecular Pharmacology January 2003, 63 (1) 1; DOI: https://doi.org/10.1124/mol.63.1.1

Accelerated Communication

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    Tonically Activated GABAA Receptors in Hippocampal Neurons Are High-Affinity, Low-Conductance Sensors for Extracellular GABA
    Jacky Y. T. Yeung, Kevin J. Canning, Guoyun Zhu, Peter Pennefather, John F. MacDonald and Beverley A. Orser
    Molecular Pharmacology January 2003, 63 (1) 2-8; DOI: https://doi.org/10.1124/mol.63.1.2

MINIREVIEW

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    Regulation of G Protein-Coupled Receptor Kinases and Arrestins During Receptor Desensitization
    Trudy A. Kohout and Robert J. Lefkowitz
    Molecular Pharmacology January 2003, 63 (1) 9-18; DOI: https://doi.org/10.1124/mol.63.1.9

Articles

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    The Selective Activation of the Glutamate Receptor GluR5 by ATPA Is Controlled by Serine 741
    Mai Marie Nielsen, Tommy Liljefors, Povl Krogsgaard-Larsen and Jan Egebjerg
    Molecular Pharmacology January 2003, 63 (1) 19-25; DOI: https://doi.org/10.1124/mol.63.1.19
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    Chemical Synthesis of MT1 and MT7 Muscarinic Toxins: Critical Role of Arg-34 in Their Interaction with M1 Muscarinic Receptor
    Gilles Mourier, Sébastien Dutertre, Carole Fruchart-Gaillard, André Ménez and Denis Servent
    Molecular Pharmacology January 2003, 63 (1) 26-35; DOI: https://doi.org/10.1124/mol.63.1.26
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    Molecular Basis of Partial Agonism: Orientation of Indoleamine Ligands in the Binding Pocket of the Human Serotonin 5-HT2A Receptor Determines Relative Efficacy
    Barbara J. Ebersole, Irache Visiers, Harel Weinstein and Stuart C. Sealfon
    Molecular Pharmacology January 2003, 63 (1) 36-43; DOI: https://doi.org/10.1124/mol.63.1.36
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    Involvement of a Calcineurin Cascade in Amygdala Depotentiation and Quenching of Fear Memory
    Chia-Ho Lin, Chia-Ching Lee and Po-Wu Gean
    Molecular Pharmacology January 2003, 63 (1) 44-52; DOI: https://doi.org/10.1124/mol.63.1.44
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    Withdrawal from Chronic Intermittent Ethanol Treatment Changes Subunit Composition, Reduces Synaptic Function, and Decreases Behavioral Responses to Positive Allosteric Modulators of GABAA Receptors
    Elisabetta Cagetti, Jing Liang, Igor Spigelman and Richard W. Olsen
    Molecular Pharmacology January 2003, 63 (1) 53-64; DOI: https://doi.org/10.1124/mol.63.1.53
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    Breast Cancer Resistance Protein (BCRP/ABCG2) Induces Cellular Resistance to HIV-1 Nucleoside Reverse Transcriptase Inhibitors
    Xin Wang, Tatsuhiko Furukawa, Takao Nitanda, Mika Okamoto, Yoshikazu Sugimoto, Shin-Ichi Akiyama and Masanori Baba
    Molecular Pharmacology January 2003, 63 (1) 65-72; DOI: https://doi.org/10.1124/mol.63.1.65
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    Evidence That the Coactivator CBP/p300 Is Important for Phenobarbital-Induced but Not Basal Expression of theCYP2H1 Gene
    Satish C. Dogra, David Tremethick and Brian K. May
    Molecular Pharmacology January 2003, 63 (1) 73-80; DOI: https://doi.org/10.1124/mol.63.1.73
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    The Effect of Insulin on Expression Level of Nucleoside Transporters in Diabetic Rats
    Tadeusz Pawelczyk, Marzena Podgorska and Monika Sakowicz
    Molecular Pharmacology January 2003, 63 (1) 81-88; DOI: https://doi.org/10.1124/mol.63.1.81
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    Coexpression of δ-Opioid Receptors with μ Receptors in GH3 Cells Changes the Functional Response to μ Agonists from Inhibitory to Excitatory
    Andrew C. Charles, Natalya Mostovskaya, Kathleen Asas, Christopher J. Evans, Megan L. Dankovich and Tim G. Hales
    Molecular Pharmacology January 2003, 63 (1) 89-95; DOI: https://doi.org/10.1124/mol.63.1.89
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    Down-Regulation of Hepatic Nicotine Metabolism and a CYP2A6-Like Enzyme in African Green Monkeys after Long-Term Nicotine Administration
    Kerri A. Schoedel, Edward M. Sellers, Roberta Palmour and Rachel F. Tyndale
    Molecular Pharmacology January 2003, 63 (1) 96-104; DOI: https://doi.org/10.1124/mol.63.1.96
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    Assessment of the Effect of Phosphorylated Metabolites of Anti-Human Immunodeficiency Virus and Anti-Hepatitis B Virus Pyrimidine Analogs on the Behavior of Human Deoxycytidylate Deaminase
    Jieh-Yuan Liou, Preethi Krishnan, Cheng-Chih Hsieh, Ginger E. Dutschman and Yung-chi Cheng
    Molecular Pharmacology January 2003, 63 (1) 105-110; DOI: https://doi.org/10.1124/mol.63.1.105
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    Parathyroid Hormone-Related Peptide Is Induced by Stimulation of α1A-Adrenoceptors and Improves Resistance against Apoptosis in Coronary Endothelial Cells
    Katja Schorr, Gerhild Taimor, Heike Degenhardt, Kerstin Weber and Klaus-Dieter Schlüter
    Molecular Pharmacology January 2003, 63 (1) 111-118; DOI: https://doi.org/10.1124/mol.63.1.111
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    Mechanism of Rat UDP-Glucuronosyltransferase 1A6 Induction by Oltipraz: Evidence for a Contribution of the Aryl Hydrocarbon Receptor Pathway
    Diana J. Auyeung, Fay K. Kessler and Joseph K. Ritter
    Molecular Pharmacology January 2003, 63 (1) 119-127; DOI: https://doi.org/10.1124/mol.63.1.119
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    Cell-Specific Extracellular Signal-Regulated Kinase Activation by Multiple G Protein-Coupled Receptor Families in Hippocampus
    Jennifer L. Berkeley and Allan I. Levey
    Molecular Pharmacology January 2003, 63 (1) 128-135; DOI: https://doi.org/10.1124/mol.63.1.128
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    Activation of Microsomal Glutathione S-Transferase by Peroxynitrite
    Yanbin Ji and Brian M. Bennett
    Molecular Pharmacology January 2003, 63 (1) 136-146; DOI: https://doi.org/10.1124/mol.63.1.136
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    Cell-Level Pharmacokinetic Model of Granulocyte Colony-Stimulating Factor: Implications for Ligand Lifetime and Potency in Vivo
    Casim A. Sarkar and Douglas A. Lauffenburger
    Molecular Pharmacology January 2003, 63 (1) 147-158; DOI: https://doi.org/10.1124/mol.63.1.147
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    Growth Inhibition by the Farnesyltransferase Inhibitor FTI-277 Involves Bcl-2 Expression and Defective Association with Raf-1 in Liver Cancer Cell Lines
    Antonio Mazzocca, Sabrina Giusti, Andrew D. Hamilton, Said M. Sebti, Pietro Pantaleo and Vinicio Carloni
    Molecular Pharmacology January 2003, 63 (1) 159-166; DOI: https://doi.org/10.1124/mol.63.1.159
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    Detection of Thymidylate Synthase Modulators by a Novel Screening Assay
    Qi Wu and Bruce J. Dolnick
    Molecular Pharmacology January 2003, 63 (1) 167-173; DOI: https://doi.org/10.1124/mol.63.1.167
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    Structural Characteristics That Govern Binding to, and Modulation through, the Cardiac Ryanodine Receptor Nucleotide Binding Site
    Wei Mun Chan, William Welch and Rebecca Sitsapesan
    Molecular Pharmacology January 2003, 63 (1) 174-182; DOI: https://doi.org/10.1124/mol.63.1.174
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    Specificity of Metabotropic Glutamate Receptor 2 Coupling to G Proteins
    Paul J. Kammermeier, Margaret I. Davis and Stephen R. Ikeda
    Molecular Pharmacology January 2003, 63 (1) 183-191; DOI: https://doi.org/10.1124/mol.63.1.183
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    Inhibition of Telomerase Increases Resistance of Melanoma Cells to Temozolomide, but Not to Temozolomide Combined with Poly (ADP-Ribose) Polymerase Inhibitor
    Lucio Tentori, Ilaria Portarena, Marcella Barbarino, Alessandra Balduzzi, Lauretta Levati, Matteo Vergati, Annamaria Biroccio, Barry Gold, Maria Luisa Lombardi and Grazia Graziani
    Molecular Pharmacology January 2003, 63 (1) 192-202; DOI: https://doi.org/10.1124/mol.63.1.192
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    The Anti-HIV Potency of Cyclotriazadisulfonamide Analogs Is Directly Correlated with Their Ability to Down-Modulate the CD4 Receptor
    Kurt Vermeire, Thomas W. Bell, Heung-Jin Choi, Qi Jin, Meinrado F. Samala, Andrej Sodoma, Erik De Clercq and Dominique Schols
    Molecular Pharmacology January 2003, 63 (1) 203-210; DOI: https://doi.org/10.1124/mol.63.1.203
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    Key Structural Features of Nonsteroidal Ligands for Binding and Activation of the Androgen Receptor
    Donghua Yin, Yali He, Minoli A. Perera, Seoung Soo Hong, Craig Marhefka, Nina Stourman, Leonid Kirkovsky, Duane D. Miller and James T. Dalton
    Molecular Pharmacology January 2003, 63 (1) 211-223; DOI: https://doi.org/10.1124/mol.63.1.211
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    All-trans-Retinoic Acid Binds to and Inhibits Adenine Nucleotide Translocase and induces Mitochondrial Permeability Transition
    Belen Notario, Mónica Zamora, Octavi Viñas and Teresa Mampel
    Molecular Pharmacology January 2003, 63 (1) 224-231; DOI: https://doi.org/10.1124/mol.63.1.224
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    Bryostatin 1 and UCN-01 Potentiate 1-β-d-Arabinofuranosylcytosine-Induced Apoptosis in Human Myeloid Leukemia Cells through Disparate Mechanisms
    Shujie Wang, Zhiliang Wang and Steven Grant
    Molecular Pharmacology January 2003, 63 (1) 232-242; DOI: https://doi.org/10.1124/mol.63.1.232
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    Monomeric and Dimeric Byproducts are the Principal Functional Elements of Higher Order P2X1 Concatamers
    Annette Nicke, Jürgen Rettinger and Günther Schmalzing
    Molecular Pharmacology January 2003, 63 (1) 243-252; DOI: https://doi.org/10.1124/mol.63.1.243
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    Cloning, Sequencing and Tissue Distribution of Rat Flavin-Containing Monooxygenase 4: Two Different Forms Are Produced by Tissue-Specific Alternative Splicing
    Virginie Lattard, Christiane Longin-Sauvageon and Etienne Benoit
    Molecular Pharmacology January 2003, 63 (1) 253-261; DOI: https://doi.org/10.1124/mol.63.1.253
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Molecular Pharmacology: 63 (1)
Molecular Pharmacology
Vol. 63, Issue 1
1 Jan 2003
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  • The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints
  • Pharmacological Properties of Y-27632, a Specific Inhibitor of Rho-Associated Kinases
  • Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
  • The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation of CYP3A4 by Rifampicin through a Distal Enhancer Module
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