Table of Contents

Articles

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  The Selective Activation of the Glutamate Receptor GluR5 by ATPA Is Controlled by Serine 741

  Mai Marie Nielsen, Tommy Liljefors, Povl Krogsgaard-Larsen and Jan Egebjerg

  Molecular Pharmacology January 2003, 63 (1) 19-25; DOI: https://doi.org/10.1124/mol.63.1.19
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  Chemical Synthesis of MT1 and MT7 Muscarinic Toxins: Critical Role of Arg-34 in Their Interaction with M₁ Muscarinic Receptor

  Gilles Mourier, Sébastien Dutertre, Carole Fruchart-Gaillard, André Ménez and Denis Servent

  Molecular Pharmacology January 2003, 63 (1) 26-35; DOI: https://doi.org/10.1124/mol.63.1.26
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  Molecular Basis of Partial Agonism: Orientation of Indoleamine Ligands in the Binding Pocket of the Human Serotonin 5-HT2A Receptor Determines Relative Efficacy

  Barbara J. Ebersole, Irache Visiers, Harel Weinstein and Stuart C. Sealfon

  Molecular Pharmacology January 2003, 63 (1) 36-43; DOI: https://doi.org/10.1124/mol.63.1.36
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  Involvement of a Calcineurin Cascade in Amygdala Depotentiation and Quenching of Fear Memory

  Chia-Ho Lin, Chia-Ching Lee and Po-Wu Gean

  Molecular Pharmacology January 2003, 63 (1) 44-52; DOI: https://doi.org/10.1124/mol.63.1.44
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  Withdrawal from Chronic Intermittent Ethanol Treatment Changes Subunit Composition, Reduces Synaptic Function, and Decreases Behavioral Responses to Positive Allosteric Modulators of GABA_A Receptors

  Elisabetta Cagetti, Jing Liang, Igor Spigelman and Richard W. Olsen

  Molecular Pharmacology January 2003, 63 (1) 53-64; DOI: https://doi.org/10.1124/mol.63.1.53
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  Breast Cancer Resistance Protein (BCRP/ABCG2) Induces Cellular Resistance to HIV-1 Nucleoside Reverse Transcriptase Inhibitors

  Xin Wang, Tatsuhiko Furukawa, Takao Nitanda, Mika Okamoto, Yoshikazu Sugimoto, Shin-Ichi Akiyama and Masanori Baba

  Molecular Pharmacology January 2003, 63 (1) 65-72; DOI: https://doi.org/10.1124/mol.63.1.65
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  Evidence That the Coactivator CBP/p300 Is Important for Phenobarbital-Induced but Not Basal Expression of theCYP2H1 Gene

  Satish C. Dogra, David Tremethick and Brian K. May

  Molecular Pharmacology January 2003, 63 (1) 73-80; DOI: https://doi.org/10.1124/mol.63.1.73
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  The Effect of Insulin on Expression Level of Nucleoside Transporters in Diabetic Rats

  Tadeusz Pawelczyk, Marzena Podgorska and Monika Sakowicz

  Molecular Pharmacology January 2003, 63 (1) 81-88; DOI: https://doi.org/10.1124/mol.63.1.81
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  Coexpression of δ-Opioid Receptors with μ Receptors in GH₃ Cells Changes the Functional Response to μ Agonists from Inhibitory to Excitatory

  Andrew C. Charles, Natalya Mostovskaya, Kathleen Asas, Christopher J. Evans, Megan L. Dankovich and Tim G. Hales

  Molecular Pharmacology January 2003, 63 (1) 89-95; DOI: https://doi.org/10.1124/mol.63.1.89
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  Down-Regulation of Hepatic Nicotine Metabolism and a CYP2A6-Like Enzyme in African Green Monkeys after Long-Term Nicotine Administration

  Kerri A. Schoedel, Edward M. Sellers, Roberta Palmour and Rachel F. Tyndale

  Molecular Pharmacology January 2003, 63 (1) 96-104; DOI: https://doi.org/10.1124/mol.63.1.96
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  Assessment of the Effect of Phosphorylated Metabolites of Anti-Human Immunodeficiency Virus and Anti-Hepatitis B Virus Pyrimidine Analogs on the Behavior of Human Deoxycytidylate Deaminase

  Jieh-Yuan Liou, Preethi Krishnan, Cheng-Chih Hsieh, Ginger E. Dutschman and Yung-chi Cheng

  Molecular Pharmacology January 2003, 63 (1) 105-110; DOI: https://doi.org/10.1124/mol.63.1.105
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  Parathyroid Hormone-Related Peptide Is Induced by Stimulation of α_1A-Adrenoceptors and Improves Resistance against Apoptosis in Coronary Endothelial Cells

  Katja Schorr, Gerhild Taimor, Heike Degenhardt, Kerstin Weber and Klaus-Dieter Schlüter

  Molecular Pharmacology January 2003, 63 (1) 111-118; DOI: https://doi.org/10.1124/mol.63.1.111
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  Mechanism of Rat UDP-Glucuronosyltransferase 1A6 Induction by Oltipraz: Evidence for a Contribution of the Aryl Hydrocarbon Receptor Pathway

  Diana J. Auyeung, Fay K. Kessler and Joseph K. Ritter

  Molecular Pharmacology January 2003, 63 (1) 119-127; DOI: https://doi.org/10.1124/mol.63.1.119
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  Cell-Specific Extracellular Signal-Regulated Kinase Activation by Multiple G Protein-Coupled Receptor Families in Hippocampus

  Jennifer L. Berkeley and Allan I. Levey

  Molecular Pharmacology January 2003, 63 (1) 128-135; DOI: https://doi.org/10.1124/mol.63.1.128
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  Activation of Microsomal Glutathione S-Transferase by Peroxynitrite

  Yanbin Ji and Brian M. Bennett

  Molecular Pharmacology January 2003, 63 (1) 136-146; DOI: https://doi.org/10.1124/mol.63.1.136
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  Cell-Level Pharmacokinetic Model of Granulocyte Colony-Stimulating Factor: Implications for Ligand Lifetime and Potency in Vivo

  Casim A. Sarkar and Douglas A. Lauffenburger

  Molecular Pharmacology January 2003, 63 (1) 147-158; DOI: https://doi.org/10.1124/mol.63.1.147
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  Growth Inhibition by the Farnesyltransferase Inhibitor FTI-277 Involves Bcl-2 Expression and Defective Association with Raf-1 in Liver Cancer Cell Lines

  Antonio Mazzocca, Sabrina Giusti, Andrew D. Hamilton, Said M. Sebti, Pietro Pantaleo and Vinicio Carloni

  Molecular Pharmacology January 2003, 63 (1) 159-166; DOI: https://doi.org/10.1124/mol.63.1.159
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  Detection of Thymidylate Synthase Modulators by a Novel Screening Assay

  Qi Wu and Bruce J. Dolnick

  Molecular Pharmacology January 2003, 63 (1) 167-173; DOI: https://doi.org/10.1124/mol.63.1.167
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  Structural Characteristics That Govern Binding to, and Modulation through, the Cardiac Ryanodine Receptor Nucleotide Binding Site

  Wei Mun Chan, William Welch and Rebecca Sitsapesan

  Molecular Pharmacology January 2003, 63 (1) 174-182; DOI: https://doi.org/10.1124/mol.63.1.174
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  Specificity of Metabotropic Glutamate Receptor 2 Coupling to G Proteins

  Paul J. Kammermeier, Margaret I. Davis and Stephen R. Ikeda

  Molecular Pharmacology January 2003, 63 (1) 183-191; DOI: https://doi.org/10.1124/mol.63.1.183
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  Inhibition of Telomerase Increases Resistance of Melanoma Cells to Temozolomide, but Not to Temozolomide Combined with Poly (ADP-Ribose) Polymerase Inhibitor

  Lucio Tentori, Ilaria Portarena, Marcella Barbarino, Alessandra Balduzzi, Lauretta Levati, Matteo Vergati, Annamaria Biroccio, Barry Gold, Maria Luisa Lombardi and Grazia Graziani

  Molecular Pharmacology January 2003, 63 (1) 192-202; DOI: https://doi.org/10.1124/mol.63.1.192
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  The Anti-HIV Potency of Cyclotriazadisulfonamide Analogs Is Directly Correlated with Their Ability to Down-Modulate the CD4 Receptor

  Kurt Vermeire, Thomas W. Bell, Heung-Jin Choi, Qi Jin, Meinrado F. Samala, Andrej Sodoma, Erik De Clercq and Dominique Schols

  Molecular Pharmacology January 2003, 63 (1) 203-210; DOI: https://doi.org/10.1124/mol.63.1.203
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  Key Structural Features of Nonsteroidal Ligands for Binding and Activation of the Androgen Receptor

  Donghua Yin, Yali He, Minoli A. Perera, Seoung Soo Hong, Craig Marhefka, Nina Stourman, Leonid Kirkovsky, Duane D. Miller and James T. Dalton

  Molecular Pharmacology January 2003, 63 (1) 211-223; DOI: https://doi.org/10.1124/mol.63.1.211
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  All-trans-Retinoic Acid Binds to and Inhibits Adenine Nucleotide Translocase and induces Mitochondrial Permeability Transition

  Belen Notario, Mónica Zamora, Octavi Viñas and Teresa Mampel

  Molecular Pharmacology January 2003, 63 (1) 224-231; DOI: https://doi.org/10.1124/mol.63.1.224
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  Bryostatin 1 and UCN-01 Potentiate 1-β-d-Arabinofuranosylcytosine-Induced Apoptosis in Human Myeloid Leukemia Cells through Disparate Mechanisms

  Shujie Wang, Zhiliang Wang and Steven Grant

  Molecular Pharmacology January 2003, 63 (1) 232-242; DOI: https://doi.org/10.1124/mol.63.1.232
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  Monomeric and Dimeric Byproducts are the Principal Functional Elements of Higher Order P2X₁ Concatamers

  Annette Nicke, Jürgen Rettinger and Günther Schmalzing

  Molecular Pharmacology January 2003, 63 (1) 243-252; DOI: https://doi.org/10.1124/mol.63.1.243
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  Cloning, Sequencing and Tissue Distribution of Rat Flavin-Containing Monooxygenase 4: Two Different Forms Are Produced by Tissue-Specific Alternative Splicing

  Virginie Lattard, Christiane Longin-Sauvageon and Etienne Benoit

  Molecular Pharmacology January 2003, 63 (1) 253-261; DOI: https://doi.org/10.1124/mol.63.1.253