Table of Contents

Articles

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  The Interaction of a Constitutively Active Arrestin with the Arrestin-Insensitive 5-HT_2A Receptor Induces Agonist-Independent Internalization

  John A. Gray, Anushree Bhatnagar, Vsevolod V. Gurevich and Bryan L. Roth

  Molecular Pharmacology May 2003, 63 (5) 961-972; DOI: https://doi.org/10.1124/mol.63.5.961
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  Identification of Tyrosine 189 and Asparagine 358 of the Cholecystokinin 2 Receptor in Direct Interaction with the Crucial C-Terminal Amide of Cholecystokinin by Molecular Modeling, Site-Directed Mutagenesis, and Structure/Affinity Studies

  Céline Galés, Marc Poirot, Julien Taillefer, Bernard Maigret, Jean Martinez, Luis Moroder, Chantal Escrieut, Lucien Pradayrol, Daniel Fourmy and Sandrine Silvente-Poirot

  Molecular Pharmacology May 2003, 63 (5) 973-982; DOI: https://doi.org/10.1124/mol.63.5.973
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  Activation and Binding of Peroxisome Proliferator-Activated Receptor γ by Synthetic Cannabinoid Ajulemic Acid

  Jilin Liu, Hui Li, Sumner H. Burstein, Robert B. Zurier and J. Don Chen

  Molecular Pharmacology May 2003, 63 (5) 983-992; DOI: https://doi.org/10.1124/mol.63.5.983
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  Spatial Approximation between a Photolabile Residue in Position 13 of Secretin and the Amino Terminus of the Secretin Receptor

  Mengwei Zang, Maoqing Dong, Delia I. Pinon, Xi-Qin Ding, Elizabeth M. Hadac, Zhijun Li, Terry P. Lybrand and Laurence J. Miller

  Molecular Pharmacology May 2003, 63 (5) 993-1001; DOI: https://doi.org/10.1124/mol.63.5.993
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  Crucial Role of Extracellular Signal-Regulated Kinase Pathway in Reactive Oxygen Species-Mediated Endothelin-1 Gene Expression Induced by Endothelin-1 in Rat Cardiac Fibroblasts

  Cheng-Ming Cheng, Hong-Jye Hong, Ju-Chi Liu, Neng-Lang Shih, Shu-Hui Juan, Shih-Hurng Loh, Paul Chan, Jin-Jer Chen and Tzu-Hurng Cheng

  Molecular Pharmacology May 2003, 63 (5) 1002-1011; DOI: https://doi.org/10.1124/mol.63.5.1002
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  Glucocorticoid Receptor Antagonism by Cyproterone Acetate and RU486

  Christian Honer, Kiyean Nam, Cynthia Fink, Paul Marshall, Gary Ksander, Ricardo E. Chatelain, Wendy Cornell, Ronald Steele, Robert Schweitzer and Christoph Schumacher

  Molecular Pharmacology May 2003, 63 (5) 1012-1020; DOI: https://doi.org/10.1124/mol.63.5.1012
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  Identification of Essential Residues Involved in the Allosteric Modulation of the Human A₃ Adenosine Receptor

  Zhan-Guo Gao, Soo-Kyung Kim, Ariel S. Gross, Aishe Chen, Joshua B. Blaustein and Kenneth A. Jacobson

  Molecular Pharmacology May 2003, 63 (5) 1021-1031; DOI: https://doi.org/10.1124/mol.63.5.1021
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  Fatty Alcohol Phosphates are Subtype-Selective Agonists and Antagonists of Lysophosphatidic Acid Receptors

  Tamas Virag, Don B. Elrod, Karoly Liliom, Vineet M. Sardar, Abby L. Parrill, Kazuaki Yokoyama, Gangadhar Durgam, Wenlin Deng, Duane D. Miller and Gabor Tigyi

  Molecular Pharmacology May 2003, 63 (5) 1032-1042; DOI: https://doi.org/10.1124/mol.63.5.1032
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  Identification of a Compound That Directly Stimulates Phospholipase C Activity

  Yoe-Sik Bae, Taehoon G. Lee, Jun Chul Park, Jung Ho Hur, Youndong Kim, Kyun Heo, Jong-Young Kwak, Pann-Ghill Suh and Sung Ho Ryu

  Molecular Pharmacology May 2003, 63 (5) 1043-1050; DOI: https://doi.org/10.1124/mol.63.5.1043
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  Voltage-Dependent Profile of HumanEther-a-go-go-Related Gene Channel Block Is Influenced by a Single Residue in the S6 Transmembrane Domain

  Jose A. Sănchez-Chapula, Tania Ferrer, Ricardo A. Navarro-Polanco and Michael C. Sanguinetti

  Molecular Pharmacology May 2003, 63 (5) 1051-1058; DOI: https://doi.org/10.1124/mol.63.5.1051
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  The Nicotinic Acetylcholine Receptor Subunit α5 Mediates Short-Term Effects of Nicotine in Vivo

  Ramiro Salas, Avi Orr-Urtreger, Ron S. Broide, Arthur Beaudet, Richard Paylor and Mariella De Biasi

  Molecular Pharmacology May 2003, 63 (5) 1059-1066; DOI: https://doi.org/10.1124/mol.63.5.1059
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  Direct Interaction of Serotonin Type 3 Receptor Ligands with Recombinant and Native α9α10-Containing Nicotinic Cholinergic Receptors

  Carla V. Rothlin, Maria I. Lioudyno, Ana F. Silbering, Paola V. Plazas, Marı́a E. Gomez Casati, Eleonora Katz, Paul S. Guth and A. Belén Elgoyhen

  Molecular Pharmacology May 2003, 63 (5) 1067-1074; DOI: https://doi.org/10.1124/mol.63.5.1067
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  Regulation of Activator Protein-1 by 8-iso-Prostaglandin E₂ in a Thromboxane A₂ Receptor-Dependent and -Independent Manner

  Thomas J. Weber and Lye M. Markillie

  Molecular Pharmacology May 2003, 63 (5) 1075-1081; DOI: https://doi.org/10.1124/mol.63.5.1075
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  [³H]R214127: A Novel High-Affinity Radioligand for the mGlu1 Receptor Reveals a Common Binding Site Shared by Multiple Allosteric Antagonists

  Hilde Lavreysen, Cor Janssen, François Bischoff, Xavier Langlois, Josée E. Leysen and Anne S. J. Lesage

  Molecular Pharmacology May 2003, 63 (5) 1082-1093; DOI: https://doi.org/10.1124/mol.63.5.1082
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  Characterization of the Transport of Nucleoside Analog Drugs by the Human Multidrug Resistance Proteins MRP4 and MRP5

  Glen Reid, Peter Wielinga, Noam Zelcer, Marcel de Haas, Liesbeth van Deemter, Jan Wijnholds, Jan Balzarini and Piet Borst

  Molecular Pharmacology May 2003, 63 (5) 1094-1103; DOI: https://doi.org/10.1124/mol.63.5.1094
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  Genetic Profiling of α₁-Adrenergic Receptor Subtypes by Oligonucleotide Microarrays: Coupling to Interleukin-6 Secretion but Differences in STAT3 Phosphorylation and gp-130

  Pedro J. Gonzalez-Cabrera, Robert J. Gaivin, June Yun, Sean A. Ross, Robert S. Papay, Dan F. McCune, Boyd R. Rorabaugh and Dianne M. Perez

  Molecular Pharmacology May 2003, 63 (5) 1104-1116; DOI: https://doi.org/10.1124/mol.63.5.1104
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  Potent Inhibition of Human Telomerase by Nitrostyrene Derivatives

  Joo Hee Kim, Jun Hyun Kim, Gun Eui Lee, Jong Eun Lee and In Kwon Chung

  Molecular Pharmacology May 2003, 63 (5) 1117-1124; DOI: https://doi.org/10.1124/mol.63.5.1117
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  Destabilization of Na_v1.7 Sodium Channel α-Subunit mRNA by Constitutive Phosphorylation of Extracellular Signal-Regulated Kinase: Negative Regulation of Steady-State Level of Cell Surface Functional Sodium Channels in Adrenal Chromaffin Cells

  Toshihiko Yanagita, Hideyuki Kobayashi, Yasuhito Uezono, Hiroki Yokoo, Takashi Sugano, Tomokazu Saitoh, Shin-Ichi Minami, Seiji Shiraishi and Akihiko Wada

  Molecular Pharmacology May 2003, 63 (5) 1125-1136; DOI: https://doi.org/10.1124/mol.63.5.1125
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  Characterization of Pulmonary CYP4B2, Specific Catalyst of Methyl Oxidation of 3-Methylindole

  Brian A. Carr, Swayampakula Ramakanth, Ghazi A. Dannan and Garold S. Yost

  Molecular Pharmacology May 2003, 63 (5) 1137-1147; DOI: https://doi.org/10.1124/mol.63.5.1137
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  Role of S-Nitrosation of Cysteine Residues in Long-Lasting Inhibitory Effect of Nitric Oxide on Arterial Tone

  Jacicarlos L. Alencar, Irina Lobysheva, Michel Geffard, Mamadou Sarr, Christa Schott, Valérie B. Schini-Kerth, Françoise Nepveu, Jean-Claude Stoclet and Bernard Muller

  Molecular Pharmacology May 2003, 63 (5) 1148-1158; DOI: https://doi.org/10.1124/mol.63.5.1148
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  Probing the Role of Linker Substituents in Bisdioxopiperazine Analogs for Activity against Wild-Type and Mutant Human Topoisomerase IIα

  Axelle Renodon-Cornière, Tina K. Sørensen, Peter B. Jensen, John L. Nitiss, Birgitte Søkilde, Maxwell Sehested and Lars H. Jensen

  Molecular Pharmacology May 2003, 63 (5) 1159-1168; DOI: https://doi.org/10.1124/mol.63.5.1159
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  Differential Declines in Striatal Nicotinic Receptor Subtype Function after Nigrostriatal Damage in Mice

  Maryka Quik, Jocelyn D. Sum, Paul Whiteaker, Sarah E. McCallum, Michael J. Marks, John Musachio, J. Michael Mcintosh, Allan C. Collins and Sharon R. Grady

  Molecular Pharmacology May 2003, 63 (5) 1169-1179; DOI: https://doi.org/10.1124/mol.63.5.1169
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  Transcriptional Regulation of Human CYP3A4 Basal Expression by CCAAT Enhancer-Binding Protein α and Hepatocyte Nuclear Factor-3γ

  C. Rodrı́guez-Antona, R. Bort, R. Jover, N. Tindberg, M. Ingelman-Sundberg, M. J. Gómez-Lechón and J. V. Castell

  Molecular Pharmacology May 2003, 63 (5) 1180-1189; DOI: https://doi.org/10.1124/mol.63.5.1180
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  Release of Cellular UDP-Glucose as a Potential Extracellular Signaling Molecule

  Eduardo R. Lazarowski, Deborah A. Shea, Richard C. Boucher and T. Kendall Harden

  Molecular Pharmacology May 2003, 63 (5) 1190-1197; DOI: https://doi.org/10.1124/mol.63.5.1190