Table of Contents

Articles

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  Identification of Novel Alternative Splice Variants of Human Constitutive Androstane Receptor and Characterization of Their Expression in the Liver

  Hideto Jinno, Toshiko Tanaka-Kagawa, Nobumitsu Hanioka, Seiich Ishida, Mayumi Saeki, Akiko Soyama, Masaya Itoda, Tetsuji Nishimura, Yoshiro Saito, Shogo Ozawa, Masanori Ando and Jun-ichi Sawada

  Molecular Pharmacology March 2004, 65 (3) 496-502; DOI: https://doi.org/10.1124/mol.65.3.496
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  Functional Role of Lipid Raft Microdomains in Cyclic Nucleotide-Gated Channel Activation

  James D. Brady, Thomas C. Rich, Xuan Le, Kimberlee Stafford, Cedar J. Fowler, Leatha Lynch, Jeffrey W. Karpen, R. Lane Brown and Jeffrey R. Martens

  Molecular Pharmacology March 2004, 65 (3) 503-511; DOI: https://doi.org/10.1124/mol.65.3.503
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  Functional and Genetic Diversity in the Concentrative Nucleoside Transporter, CNT1, in Human Populations

  Jennifer H. Gray, Lara M. Mangravite, Ryan P. Owen, Thomas J. Urban, Wendy Chan, Elaine J. Carlson, Conrad C. Huang, Michiko Kawamoto, Susan J. Johns, Douglas Stryke, Thomas E. Ferrin and Kathleen M. Giacomini

  Molecular Pharmacology March 2004, 65 (3) 512-519; DOI: https://doi.org/10.1124/mol.65.3.512
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  Valproic Acid Inhibits Angiogenesis in Vitro and in Vivo

  Martin Michaelis, U. Ruth Michaelis, Ingrid Fleming, Tatyana Suhan, Jaroslav Cinatl, Roman A. Blaheta, Katrin Hoffmann, Rouslan Kotchetkov, Rudi Busse, Heinz Nau and Jindrich Cinatl

  Molecular Pharmacology March 2004, 65 (3) 520-527; DOI: https://doi.org/10.1124/mol.65.3.520
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  Distinct Domains of the μ-Opioid Receptor Control Uncoupling and Internalization

  Jeremy Celver, Mei Xu, Wenzhen Jin, Janet Lowe and Charles Chavkin

  Molecular Pharmacology March 2004, 65 (3) 528-537; DOI: https://doi.org/10.1124/mol.65.3.528
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  8R-Lisuride Is a Potent Stereospecific Histamine H₁-Receptor Partial Agonist

  R. A. Bakker, D. M. Weiner, T. ter Laak, T. Beuming, O. P. Zuiderveld, M. Edelbroek, U. Hacksell, H. Timmerman, M. R. Brann and R. Leurs

  Molecular Pharmacology March 2004, 65 (3) 538-549; DOI: https://doi.org/10.1124/mol.65.3.538
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  Retinoid X Receptor α Regulates Glutathione Homeostasis and Xenobiotic Detoxification Processes in Mouse Liver

  Yong Wu, Xiaoxue Zhang, Fawzia Bardag-Gorce, Rose C. V. Robel, Jonathan Aguilo, Lixin Chen, Ying Zeng, Kelly Hwang, Samuel W. French, Shelly C. Lu and Yu-Jui Y. Wan

  Molecular Pharmacology March 2004, 65 (3) 550-557; DOI: https://doi.org/10.1124/mol.65.3.550
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  Molecular Requirements of the Human Nucleoside Transporters hCNT1, hCNT2, and hENT1

  C. Chang, P. W. Swaan, L. Y. Ngo, P. Y. Lum, S. D. Patil and J. D. Unadkat

  Molecular Pharmacology March 2004, 65 (3) 558-570; DOI: https://doi.org/10.1124/mol.65.3.558
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  Evidence of a Functional Role for p21^WAF1/CIP1 Down-Regulation in Synergistic Antileukemic Interactions between the Histone Deacetylase Inhibitor Sodium Butyrate and Flavopiridol

  Roberto R. Rosato, Jorge A. Almenara, Chunrong Yu and Steven Grant

  Molecular Pharmacology March 2004, 65 (3) 571-581; DOI: https://doi.org/10.1124/mol.65.3.571
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  Structural Determinants Required for the Bioactivities of Prokineticins and Identification of Prokineticin Receptor Antagonists

  Clayton M. Bullock, Jia-Da Li and Qun-Yong Zhou

  Molecular Pharmacology March 2004, 65 (3) 582-588; DOI: https://doi.org/10.1124/mol.65.3.582
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  Differential Role of Janus Family Kinases (JAKs) in Interferon-γ–Induced Lung Epithelial ICAM-1 Expression: Involving Protein Interactions between JAKs, Phospholipase Cγ, c-Src, and STAT1

  Ya-Jen Chang, Michael J. Holtzman and Ching-Chow Chen

  Molecular Pharmacology March 2004, 65 (3) 589-598; DOI: https://doi.org/10.1124/mol.65.3.589
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  Caffeic Acid Esters Activate TREK-1 Potassium Channels and Inhibit Depolarization-Dependent Secretion

  Sanjay Danthi, Judith A. Enyeart and John J. Enyeart

  Molecular Pharmacology March 2004, 65 (3) 599-610; DOI: https://doi.org/10.1124/mol.65.3.599
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  Up-Regulation of Brain Nicotinic Acetylcholine Receptors in the Rat during Long-Term Self-Administration of Nicotine: Disproportionate Increase of the α6 Subunit

  Steven L. Parker, Yitong Fu, Kathleen McAllen, Jianhong Luo, J. Michael McIntosh, Jon M. Lindstrom and Burt M. Sharp

  Molecular Pharmacology March 2004, 65 (3) 611-622; DOI: https://doi.org/10.1124/mol.65.3.611
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  Vasopressin Stimulates Insulin Release from Islet Cells through V1b Receptors: a Combined Pharmacological/Knockout Approach

  Sayuri Oshikawa, Akito Tanoue, Taka-aki Koshimizu, Yoko Kitagawa and Gozoh Tsujimoto

  Molecular Pharmacology March 2004, 65 (3) 623-629; DOI: https://doi.org/10.1124/mol.65.3.623
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  Blockage of Intermediate-Conductance Ca²⁺-Activated K⁺ Channels Inhibit Human Pancreatic Cancer Cell Growth in Vitro

  Heike Jäger, Tobias Dreker, Anita Buck, Klaudia Giehl, Thomas Gress and Stephan Grissmer

  Molecular Pharmacology March 2004, 65 (3) 630-638; DOI: https://doi.org/10.1124/mol.65.3.630
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  Dipyridamole Alters Cardiac Substrate Preference by Inducing Translocation of FAT/CD36, but Not That of GLUT4

  Joost J. F. P. Luiken, Susan L. M. Coort, Jodil Willems, Will A. Coumans, Arend Bonen and Jan F. C. Glatz

  Molecular Pharmacology March 2004, 65 (3) 639-645; DOI: https://doi.org/10.1124/mol.65.3.639
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  Selective Knock-Down of P2X₇ ATP Receptor Function by Dominant-Negative Subunits

  Ramin Raouf, Yassar Chakfe, Dominique Blais, Audrey Speelman, Eric Boué-Grabot, Duncan Henderson and Philippe Séguéla

  Molecular Pharmacology March 2004, 65 (3) 646-654; DOI: https://doi.org/10.1124/mol.65.3.646
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  Protein Adduct-Trapping by Hydrazinophthalazine Drugs: Mechanisms of Cytoprotection Against Acrolein-Mediated Toxicity

  Philip C. Burcham, Frank R. Fontaine, Lisa M. Kaminskas, Dennis R. Petersen and Simon M. Pyke

  Molecular Pharmacology March 2004, 65 (3) 655-664; DOI: https://doi.org/10.1124/mol.65.3.655
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  Endocannabinoids Modulate N-Type Calcium Channels and G-Protein-Coupled Inwardly Rectifying Potassium Channels via CB1 Cannabinoid Receptors Heterologously Expressed in Mammalian Neurons

  Juan Guo and Stephen R. Ikeda

  Molecular Pharmacology March 2004, 65 (3) 665-674; DOI: https://doi.org/10.1124/mol.65.3.665
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  The Molecular Basis of the Action of Disulfiram as a Modulator of the Multidrug Resistance-Linked ATP Binding Cassette Transporters MDR1 (ABCB1) and MRP1 (ABCC1)

  Zuben E. Sauna, Xiang-Hong Peng, Krishnamachary Nandigama, Samrawit Tekle and Suresh V. Ambudkar

  Molecular Pharmacology March 2004, 65 (3) 675-684; DOI: https://doi.org/10.1124/mol.65.3.675
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  Combinatorial Interaction of Scorpion Toxins Lqh-2, Lqh-3, and LqhαIT with Sodium Channel Receptor Sites-3

  Enrico Leipold, Songqing Lu, Dalia Gordon, Alfred Hansel and Stefan H. Heinemann

  Molecular Pharmacology March 2004, 65 (3) 685-691; DOI: https://doi.org/10.1124/mol.65.3.685
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  Uptake Inhibitors but not Substrates Induce Protease Resistance in Extracellular Loop Two of the Dopamine Transporter

  Jon D. Gaffaney and Roxanne A. Vaughan

  Molecular Pharmacology March 2004, 65 (3) 692-701; DOI: https://doi.org/10.1124/mol.65.3.692
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  Random Mutagenesis of the Human Adenosine A_2B Receptor Followed by Growth Selection in Yeast. Identification of Constitutively Active and Gain of Function Mutations

  Margot W. Beukers, Joris van Oppenraaij, Patrick P. W. van der Hoorn, Clara C. Blad, Hans den Dulk, Jaap Brouwer and Adriaan P. IJzerman

  Molecular Pharmacology March 2004, 65 (3) 702-710; DOI: https://doi.org/10.1124/mol.65.3.702
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  Expression of A₃ Adenosine Receptors in Human Lymphocytes: Up-Regulation in T Cell Activation

  Stefania Gessi, Katia Varani, Stefania Merighi, Elena Cattabriga, Arianna Avitabile, Riccardo Gavioli, Cinzia Fortini, Edward Leung, Stephen Mac Lennan and Pier Andrea Borea

  Molecular Pharmacology March 2004, 65 (3) 711-719; DOI: https://doi.org/10.1124/mol.65.3.711
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  Dehydroepiandrosterone Sulfotransferase Is a Target for Transcriptional Induction by the Vitamin D Receptor

  Ibtissam Echchgadda, Chung S. Song, Arun K. Roy and Bandana Chatterjee

  Molecular Pharmacology March 2004, 65 (3) 720-729; DOI: https://doi.org/10.1124/mol.65.3.720
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  Regulation of Mouse Renal CYP2J5 Expression by Sex Hormones

  Jixiang Ma, Joan Graves, J. Alyce Bradbury, Yun Zhao, Deborah L. Swope, Lorraine King, Wei Qu, James Clark, Page Myers, Vickie Walker, Jonathan Lindzey, Kenneth S. Korach and Darryl C. Zeldin

  Molecular Pharmacology March 2004, 65 (3) 730-743; DOI: https://doi.org/10.1124/mol.65.3.730
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  SB-505124 Is a Selective Inhibitor of Transforming Growth Factor-β Type I Receptors ALK4, ALK5, and ALK7

  Stacey DaCosta Byfield, Christopher Major, Nicholas J. Laping and Anita B. Roberts

  Molecular Pharmacology March 2004, 65 (3) 744-752; DOI: https://doi.org/10.1124/mol.65.3.744
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  Ligand Function at Constitutively Active Receptor Mutants Is Affected by Two Distinct Yet Interacting Mechanisms

  Martin Beinborn, Yong Ren, Michael Bläker, Ci Chen and Alan S. Kopin

  Molecular Pharmacology March 2004, 65 (3) 753-760; DOI: https://doi.org/10.1124/mol.65.3.753
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  DAXX, FLASH, and FAF-1 Modulate Mineralocorticoid and Glucocorticoid Receptor-Mediated Transcription in Hippocampal Cells—Toward a Basis for the Opposite Actions Elicited by Two Nuclear Receptors?

  D. Obradović, M. Tirard, Zs. Némethy, O. Hirsch, H. Gronemeyer and O. F. X. Almeida

  Molecular Pharmacology March 2004, 65 (3) 761-769; DOI: https://doi.org/10.1124/mol.65.3.761
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  Loss-of-Function Polymorphic Variants of the Human Angiotensin II Type 1 Receptor

  Jakob Lerche Hansen, Stig Haunsø, Mark R. Brann, Søren P. Sheikh and David M. Weiner

  Molecular Pharmacology March 2004, 65 (3) 770-777; DOI: https://doi.org/10.1124/mol.65.3.770
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  Phorbol 12-Myristate 13-Acetate Protects Jurkat Cells from Methylglyoxal-Induced Apoptosis by Preventing c-Jun N-Terminal Kinase-Mediated Leakage of Cytochrome c in an Extracellular Signal-Regulated Kinase-Dependent Manner

  Yoshikazu Takagi, Jun Du, Xiu-Yang Ma, Izumi Nakashima and Fumihiko Nagase

  Molecular Pharmacology March 2004, 65 (3) 778-787; DOI: https://doi.org/10.1124/mol.65.3.778
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  An Apamin- and Scyllatoxin-Insensitive Isoform of the Human SK3 Channel

  Oliver H. Wittekindt, Violeta Visan, Hiroaki Tomita, Faiqa Imtiaz, Jay J. Gargus, Frank Lehmann-Horn, Stephan Grissmer and Deborah J. Morris-Rosendahl

  Molecular Pharmacology March 2004, 65 (3) 788-801; DOI: https://doi.org/10.1124/mol.65.3.788
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  Effects of SEA0400 on Mutant NCX1.1 Na⁺-Ca²⁺ Exchangers with Altered Ionic Regulation

  Ron Bouchard, Alexander Omelchenko, Hoa Dinh Le, Platon Choptiany, Toshio Matsuda, Akemichi Baba, Kenzo Takahashi, Debora A. Nicoll, Kenneth D. Philipson, Mark Hnatowich and Larry V. Hryshko

  Molecular Pharmacology March 2004, 65 (3) 802-810; DOI: https://doi.org/10.1124/mol.65.3.802
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  Correction to “Agonist Binding and Gq-Stimulating Activities of the Purified Human P2Y₁ Receptor”

  Molecular Pharmacology March 2004, 65 (3) 811; DOI: https://doi.org/10.1124/mol.65.3.811