Sazetidine-A, A Novel Ligand That Desensitizes α4β2 Nicotinic Acetylcholine Receptors without Activating Them

Department of Pharmacology, Georgetown University School of Medicine, Washington DC (Y.X., K.J.K.); Department of Radiology, Johns Hopkins University School of Medicine, Baltimore, Maryland (H.F., J.L.M.); and Department of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, University of Illinois at Chicago, Chicago, Illinois (Z.-L.W., S.K.C., A.P.K.).

Address correspondence to:
Kenneth J. Kellar, Department of Pharmacology, Georgetown University School of Medicine, Washington, DC 20057. E-mail: kellark{at}georgetown.edu

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Feb 2021	23	12	5
Mar 2021	34	8	6
Apr 2021	10	1	1