Table of Contents

Articles

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  Live Cell Analysis of G Protein β₅ Complex Formation, Function, and Targeting

  Evan A. Yost, Stacy M. Mervine, Jonathan L. Sabo, Thomas R. Hynes and Catherine H. Berlot

  Molecular Pharmacology October 2007, 72 (4) 812-825; DOI: https://doi.org/10.1124/mol.107.038075
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  Discovery of Osmosensitive Transcriptional Regulation of Human Cytochrome P450 3As by the Tonicity-Responsive Enhancer Binding Protein (Nuclear Factor of Activated T Cells 5)

  Kazuhiro Kosuge, Andrew I. Chuang, Satoko Uematsu, Kah Poh Tan, Kyoichi Ohashi, Ben C.B. Ko and Shinya Ito

  Molecular Pharmacology October 2007, 72 (4) 826-837; DOI: https://doi.org/10.1124/mol.107.034504
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  Structural Determinates for Apolipoprotein E-Derived Peptide Interaction with the α7 Nicotinic Acetylcholine Receptor

  Elaine A. Gay, Rachelle J. Bienstock, Patricia W. Lamb and Jerrel L. Yakel

  Molecular Pharmacology October 2007, 72 (4) 838-849; DOI: https://doi.org/10.1124/mol.107.035527
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  Insulin Facilitates the Hepatic Clearance of Plasma Amyloid β-Peptide (1–40) by Intracellular Translocation of Low-Density Lipoprotein Receptor-Related Protein 1 (LRP-1) to the Plasma Membrane in Hepatocytes

  Chihiro Tamaki, Sumio Ohtsuki and Tetsuya Terasaki

  Molecular Pharmacology October 2007, 72 (4) 850-855; DOI: https://doi.org/10.1124/mol.107.036913
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  Activation of the Adenosine A₁ Receptor Inhibits HIV-1 Tat-Induced Apoptosis by Reducing Nuclear Factor-κB Activation and Inducible Nitric-Oxide Synthase

  Sandeep C. Pingle, Sarvesh Jajoo, Debashree Mukherjea, Lynn F. Sniderhan, Krishna A. Jhaveri, Adriana Marcuzzi, Leonard P. Rybak, Sanjay B. Maggirwar and Vickram Ramkumar

  Molecular Pharmacology October 2007, 72 (4) 856-867; DOI: https://doi.org/10.1124/mol.106.031427
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  Application of β-Lactamase Enzyme Complementation to the High-Throughput Screening of Toll-Like Receptor Signaling Inhibitors

  Hyun-Ku Lee, Steven J. Brown, Hugh Rosen and Peter S. Tobias

  Molecular Pharmacology October 2007, 72 (4) 868-875; DOI: https://doi.org/10.1124/mol.107.038349
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  Identification of a Bis-guanylhydrazone [4,4′-Diacetyldiphenylurea-bis(guanylhydrazone); NSC 109555] as a Novel Chemotype for Inhibition of Chk2 Kinase

  Andrew G. Jobson, John H. Cardellina, Dominic Scudiero, Sudhir Kondapaka, Hongliang Zhang, Hijoo Kim, Robert Shoemaker and Yves Pommier

  Molecular Pharmacology October 2007, 72 (4) 876-884; DOI: https://doi.org/10.1124/mol.107.035832
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  Serotonin 5-Hydroxytryptamine_2C Receptor Signaling in Hypothalamic Proopiomelanocortin Neurons: Role in Energy Homeostasis in Females

  Jian Qiu, Changhui Xue, Martha A. Bosch, Jonathan G. Murphy, Wei Fan, Oline K. Rønnekleiv and Martin J. Kelly

  Molecular Pharmacology October 2007, 72 (4) 885-896; DOI: https://doi.org/10.1124/mol.107.038083
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  Neutralization of Plasminogen Activator Inhibitor I (PAI-1) by the Synthetic Antagonist PAI-749 via a Dual Mechanism of Action

  Stephen J. Gardell, Julie A. Krueger, Thomas A. Antrilli, Hassan Elokdah, Scott Mayer, Steven J. Orcutt, David L. Crandall and George P. Vlasuk

  Molecular Pharmacology October 2007, 72 (4) 897-906; DOI: https://doi.org/10.1124/mol.107.037010
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  Subunit-Specific Agonist Activity at NR2A-, NR2B-, NR2C-, and NR2D-Containing N-Methyl-d-aspartate Glutamate Receptors

  Kevin Erreger, Matthew T. Geballe, Anders Kristensen, Philip E. Chen, Kasper B. Hansen, C. Justin Lee, Hongjie Yuan, Phuong Le, Polina N. Lyuboslavsky, Nicola Micale, Lars Jørgensen, Rasmus P. Clausen, David J. A. Wyllie, James P. Snyder and Stephen F. Traynelis

  Molecular Pharmacology October 2007, 72 (4) 907-920; DOI: https://doi.org/10.1124/mol.107.037333
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  Identification of Regions of the σ-1 Receptor Ligand Binding Site Using a Novel Photoprobe

  Arindam Pal, Abdol R. Hajipour, Dominique Fontanilla, Subramaniam Ramachandran, Uyen B. Chu, Timur Mavlyutov and Arnold E. Ruoho

  Molecular Pharmacology October 2007, 72 (4) 921-933; DOI: https://doi.org/10.1124/mol.107.038307
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  Gemfibrozil Ameliorates Relapsing-Remitting Experimental Autoimmune Encephalomyelitis Independent of Peroxisome Proliferator-Activated Receptor-α

  Subhajit Dasgupta, Avik Roy, Malabendu Jana, Dean M. Hartley and Kalipada Pahan

  Molecular Pharmacology October 2007, 72 (4) 934-946; DOI: https://doi.org/10.1124/mol.106.033787
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  Physiological Differences between Human and Rat Primary Hepatocytes in Response to Liver X Receptor Activation by 3-[3-[N-(2-Chloro-3-trifluoromethylbenzyl)-(2,2-diphenylethyl)amino]propyloxy]phenylacetic Acid Hydrochloride (GW3965)

  Pia Kotokorpi, Ewa Ellis, Paolo Parini, Lisa-Mari Nilsson, Stephen Strom, Knut R. Steffensen, Jan-Åke Gustafsson and Agneta Mode

  Molecular Pharmacology October 2007, 72 (4) 947-955; DOI: https://doi.org/10.1124/mol.107.037358
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  Aryl Hydrocarbon Receptor Splice Variants in the Dioxin-Resistant Rat: Tissue Expression and Transactivational Activity

  Ivy D. Moffat, Steven Roblin, Patricia A. Harper, Allan B. Okey and Raimo Pohjanvirta

  Molecular Pharmacology October 2007, 72 (4) 956-966; DOI: https://doi.org/10.1124/mol.107.037218
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  Effect of Breast Cancer Resistance Protein (Bcrp/Abcg2) on the Disposition of Phytoestrogens

  Junichi Enokizono, Hiroyuki Kusuhara and Yuichi Sugiyama

  Molecular Pharmacology October 2007, 72 (4) 967-975; DOI: https://doi.org/10.1124/mol.107.034751
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  Pharmacological Characterization of a Novel Nonpeptide Antagonist for Formyl Peptide Receptor-Like 1

  Caihong Zhou, Song Zhang, Masakatsu Nanamori, Yueyun Zhang, Qing Liu, Na Li, Meiling Sun, Jun Tian, Patrick P. Ye, Ni Cheng, Richard D. Ye and Ming-Wei Wang

  Molecular Pharmacology October 2007, 72 (4) 976-983; DOI: https://doi.org/10.1124/mol.107.037564
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  Antithrombotic Effect of a Protein-Type I Class Snake Venom Metalloproteinase, Kistomin, Is Mediated by Affecting Glycoprotein Ib-von Willebrand Factor Interaction

  Chun-Chieh Hsu, Wen-Bin Wu, Ya-Hui Chang, Heng-Lan Kuo and Tur-Fu Huang

  Molecular Pharmacology October 2007, 72 (4) 984-992; DOI: https://doi.org/10.1124/mol.107.038018
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  Disruption of Oligomerization Induces Nucleocytoplasmic Shuttling of Leukemia-Associated Rho Guanine-Nucleotide Exchange Factor

  Elda Grabocka and Philip B. Wedegaertner

  Molecular Pharmacology October 2007, 72 (4) 993-1002; DOI: https://doi.org/10.1124/mol.107.035162
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  A Mouse Model for Studying the Interaction of Bisdioxopiperazines with Topoisomerase IIα in Vivo

  Morten Grauslund, Annemette Vinding Thougaard, Annette Füchtbauer, Kenneth Francis Hofland, Peter Hansen Hjorth, Peter B. Jensen, Maxwell Sehested, Ernst-Martin Füchtbauer and Lars H. Jensen

  Molecular Pharmacology October 2007, 72 (4) 1003-1014; DOI: https://doi.org/10.1124/mol.107.036970
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  γ-Glutamylcysteine Synthetase Mediates the c-Myc-Dependent Response to Antineoplastic Agents in Melanoma Cells

  Barbara Benassi, Gabriella Zupi and Annamaria Biroccio

  Molecular Pharmacology October 2007, 72 (4) 1015-1023; DOI: https://doi.org/10.1124/mol.107.038687
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  The Endocannabinoid Anandamide Inhibits the Function of α4β2 Nicotinic Acetylcholine Receptors

  Charles E. Spivak, Carl R. Lupica and Murat Oz

  Molecular Pharmacology October 2007, 72 (4) 1024-1032; DOI: https://doi.org/10.1124/mol.107.036939
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  The Small Molecule NS11021 Is a Potent and Specific Activator of Ca²⁺-Activated Big-Conductance K⁺ Channels

  Bo Hjorth Bentzen, Antonio Nardi, Kirstine Calloe, Lars Siim Madsen, Søren-Peter Olesen and Morten Grunnet

  Molecular Pharmacology October 2007, 72 (4) 1033-1044; DOI: https://doi.org/10.1124/mol.107.038331
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  Down-Regulation of Pregnane X Receptor Contributes to Cell Growth Inhibition and Apoptosis by Anticancer Agents in Endometrial Cancer Cells

  Hisashi Masuyama, Hideki Nakatsukasa, Norio Takamoto and Yuji Hiramatsu

  Molecular Pharmacology October 2007, 72 (4) 1045-1053; DOI: https://doi.org/10.1124/mol.107.037937
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  Critical Roles of Residues 36 and 40 in the Phenol and Tertiary Amine Aglycone Substrate Selectivities of UDP-Glucuronosyltransferases 1A3 and 1A4

  Takahiro Kubota, Benjamin C. Lewis, David J. Elliot, Peter I. Mackenzie and John O. Miners

  Molecular Pharmacology October 2007, 72 (4) 1054-1062; DOI: https://doi.org/10.1124/mol.107.037952
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  Electrophysiological Properties of Cardiomyocytes Isolated from CYP2J2 Transgenic Mice

  Qingen Ke, Yong-Fu Xiao, J. Alyce Bradbury, Joan P. Graves, Laura M. DeGraff, John M. Seubert and Darryl C. Zeldin

  Molecular Pharmacology October 2007, 72 (4) 1063-1073; DOI: https://doi.org/10.1124/mol.107.035881
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  Translational Control of Nrf2 Protein in Activation of Antioxidant Response by Oxidants

  Sally E. Purdom-Dickinson, Elena V. Sheveleva, Haipeng Sun and Qin M. Chen

  Molecular Pharmacology October 2007, 72 (4) 1074-1081; DOI: https://doi.org/10.1124/mol.107.035360
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  Induction of Glutathione Transferase in Insulin-Like Growth Factor Type I Receptor-Overexpressed Hepatoma Cells

  Jeong Yong Lee, Chang Yeob Han, Jin Won Yang, Christopher Smith, Sang Kyum Kim, Eva Y.-H. P. Lee, Sang Geon Kim and Keon Wook Kang

  Molecular Pharmacology October 2007, 72 (4) 1082-1093; DOI: https://doi.org/10.1124/mol.107.038174