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Molecular Pharmacology

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OtherMINIREVIEW

Functional Selectivity through Protean and Biased Agonism: Who Steers the Ship?

Terry Kenakin
Molecular Pharmacology December 2007, 72 (6) 1393-1401; DOI: https://doi.org/10.1124/mol.107.040352
Terry Kenakin
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In this issue

Molecular Pharmacology: 72 (6)
Molecular Pharmacology
Vol. 72, Issue 6
1 Dec 2007
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OtherMINIREVIEW

Functional Selectivity through Protean and Biased Agonism: Who Steers the Ship?

Terry Kenakin
Molecular Pharmacology December 1, 2007, 72 (6) 1393-1401; DOI: https://doi.org/10.1124/mol.107.040352

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OtherMINIREVIEW

Functional Selectivity through Protean and Biased Agonism: Who Steers the Ship?

Terry Kenakin
Molecular Pharmacology December 1, 2007, 72 (6) 1393-1401; DOI: https://doi.org/10.1124/mol.107.040352
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  • Article
    • Abstract
    • Single Receptor State Receptor Selectivity
    • Receptor-Based Biased Functional Selectivity
    • Protean Agonism
    • Indirect Ligand-Induced Bias
    • Receptor-Based Selectivity
    • Should Functional Selectivity Be an Expected Event?
    • Conclusions
    • Appendix
    • Footnotes
    • References
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