New Insights into the Function of M4 Muscarinic Acetylcholine Receptors Gained Using a Novel Allosteric Modulator and a DREADD (Designer Receptor Exclusively Activated by a Designer Drug)

Drug Discovery Biology Laboratory, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Melbourne, Australia (V.N., K.L., N.S., R.E.L., P.M.S., A.C.), Neuroscience, Lilly Corporate Center, Indianapolis, Indiana (C.C.F.); Millipore Inc., St. Louis, Missouri (B.N.A.); and Departments of Pharmacology and Medicinal Chemistry, University of North Carolina Chapel Hill Medical School, North Carolina (B.L.R.)

Address correspondence to:
Prof. Arthur Christopoulos, Drug Discovery Biology Laboratory, Department of Pharmacology, Monash University, Clayton, Victoria 3800, Australia. E-mail: arthur.christopoulos{at}med.monash.edu.au

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