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Molecular Pharmacology

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Table of Contents

December 01, 2008; Volume 74,Issue 6

Articles

  • You have access
    Comparison of the Potential Multiple Binding Modes of Bicyclam, Monocylam, and Noncyclam Small-Molecule CXC Chemokine Receptor 4 Inhibitors
    Rebecca S. Y. Wong, Veronique Bodart, Markus Metz, Jean Labrecque, Gary Bridger and Simon P. Fricker
    Molecular Pharmacology December 2008, 74 (6) 1485-1495; DOI: https://doi.org/10.1124/mol.108.049775
  • You have access
    Multiple Pharmacophores for the Selective Activation of Nicotinic α7-Type Acetylcholine Receptors
    Nicole A. Horenstein, Fedra M. Leonik and Roger L. Papke
    Molecular Pharmacology December 2008, 74 (6) 1496-1511; DOI: https://doi.org/10.1124/mol.108.048892
  • You have access
    Structural Basis of Human Pregnane X Receptor Activation by the Hops Constituent Colupulone
    Denise G. Teotico, Jason J. Bischof, Li Peng, Steven A. Kliewer and Matthew R. Redinbo
    Molecular Pharmacology December 2008, 74 (6) 1512-1520; DOI: https://doi.org/10.1124/mol.108.050732
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    The Orphan Transporter Rxt1/NTT4 (SLC6A17) Functions as a Synaptic Vesicle Amino Acid Transporter Selective for Proline, Glycine, Leucine, and Alanine
    Leonardo A. Parra, Tracy Baust, Salah El Mestikawy, Marisol Quiroz, Beth Hoffman, Jack M. Haflett, Jeffrey K. Yao and Gonzalo E. Torres
    Molecular Pharmacology December 2008, 74 (6) 1521-1532; DOI: https://doi.org/10.1124/mol.108.050005
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    17-β-Estradiol Inhibits Transforming Growth Factor-β Signaling and Function in Breast Cancer Cells via Activation of Extracellular Signal-Regulated Kinase through the G Protein-Coupled Receptor 30
    Burkhard Kleuser, Daniela Malek, Ronald Gust, Heinz H. Pertz and Henrik Potteck
    Molecular Pharmacology December 2008, 74 (6) 1533-1543; DOI: https://doi.org/10.1124/mol.108.046854
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    Aryl Hydrocarbon Receptor-Mediated Down-Regulation of Sox9b Causes Jaw Malformation in Zebrafish Embryos
    Kong M. Xiong, Richard E. Peterson and Warren Heideman
    Molecular Pharmacology December 2008, 74 (6) 1544-1553; DOI: https://doi.org/10.1124/mol.108.050435
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    Different Interactions between MT7 Toxin and the Human Muscarinic M1 Receptor in Its Free and N-Methylscopolamine-Occupied States
    Carole Fruchart-Gaillard, Gilles Mourier, Catherine Marquer, Enrico Stura, Nigel J. M. Birdsall and Denis Servent
    Molecular Pharmacology December 2008, 74 (6) 1554-1563; DOI: https://doi.org/10.1124/mol.108.050773
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    Overexpression of Heme Oxygenase-1 Protects Dopaminergic Neurons against 1-Methyl-4-Phenylpyridinium-Induced Neurotoxicity
    Shih-Ya Hung, Houng-Chi Liou, Kai-Hsiang Kang, Ruey-Meei Wu, Chun-Chiang Wen and Wen-Mei Fu
    Molecular Pharmacology December 2008, 74 (6) 1564-1575; DOI: https://doi.org/10.1124/mol.108.048611
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    Identification of Quinolines that Inhibit Melanogenesis by Altering Tyrosinase Family Trafficking
    Li Ni-Komatsu, ChunXiang Tong, Guangming Chen, Nelya Brindzei and Seth J. Orlow
    Molecular Pharmacology December 2008, 74 (6) 1576-1586; DOI: https://doi.org/10.1124/mol.108.050633
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    Imidazoquinolinone, Imidazopyridine, and Isoquinolindione Derivatives as Novel and Potent Inhibitors of the Poly(ADP-ribose) Polymerase (PARP): A Comparison with Standard PARP Inhibitors
    Tobias Eltze, Rainer Boer, Thomas Wagner, Steffen Weinbrenner, Michelle C. McDonald, Christoph Thiemermann, Alexander Bürkle and Thomas Klein
    Molecular Pharmacology December 2008, 74 (6) 1587-1598; DOI: https://doi.org/10.1124/mol.108.048751
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    Identification and Functional Characterization of Allosteric Agonists for the G Protein-Coupled Receptor FFA2
    Taeweon Lee, Ralf Schwandner, Gayathri Swaminath, Jennifer Weiszmann, Mario Cardozo, Joanne Greenberg, Peter Jaeckel, Hongfei Ge, Yingcai Wang, Xianyun Jiao, Jiwen Liu, Frank Kayser, Hui Tian and Yang Li
    Molecular Pharmacology December 2008, 74 (6) 1599-1609; DOI: https://doi.org/10.1124/mol.108.049536
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    Endoplasmic Reticulum Stress Induces Leptin Resistance
    Toru Hosoi, Miyako Sasaki, Tsuyoshi Miyahara, Chie Hashimoto, Suguru Matsuo, Michiko Yoshii and Koichiro Ozawa
    Molecular Pharmacology December 2008, 74 (6) 1610-1619; DOI: https://doi.org/10.1124/mol.108.050070
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    Rebeccamycin Derivatives as Dual DNA-Damaging Agents and Potent Checkpoint Kinase 1 Inhibitors
    Christelle Marminon, Fabrice Anizon, Pascale Moreau, Bruno Pfeiffer, Alain Pierré, Roy M. Golsteyn, Paul Peixoto, Marie-Paule Hildebrand, Marie-Hélène David-Cordonnier, Olivier Lozach, Laurent Meijer and Michelle Prudhomme
    Molecular Pharmacology December 2008, 74 (6) 1620-1629; DOI: https://doi.org/10.1124/mol.108.049346
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    Mechanistic Differences between GSH Transport by Multidrug Resistance Protein 1 (MRP1/ABCC1) and GSH Modulation of MRP1-Mediated Transport
    Alice Rothnie, Gwenaëlle Conseil, Andrea Y. T. Lau, Roger G. Deeley and Susan P. C. Cole
    Molecular Pharmacology December 2008, 74 (6) 1630-1640; DOI: https://doi.org/10.1124/mol.108.049080
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    Nicotine Relieves Anxiogenic-Like Behavior in Mice that Overexpress the Read-Through Variant of Acetylcholinesterase but Not in Wild-Type Mice
    R. Salas, A. Main, D. A. Gangitano, G. Zimmerman, S. Ben-Ari, H. Soreq and M. De Biasi
    Molecular Pharmacology December 2008, 74 (6) 1641-1648; DOI: https://doi.org/10.1124/mol.108.048454
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    12(R)-Hydroxy-5(Z),8(Z),10(E),14(Z)-eicosatetraenoic Acid [12(R)-HETE], an Arachidonic Acid Derivative, Is an Activator of the Aryl Hydrocarbon Receptor
    Christopher. R. Chiaro, Rushang D. Patel and Gary. H. Perdew
    Molecular Pharmacology December 2008, 74 (6) 1649-1656; DOI: https://doi.org/10.1124/mol.108.049379
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    Dissecting the Role of Multiple Reductases in Bioactivation and Cytotoxicity of the Antitumor Agent 2,5-Diaziridinyl-3-(hydroxymethyl)-6-methyl-1,4-benzoquinone (RH1)
    Chao Yan, Jadwiga K. Kepa, David Siegel, Ian J. Stratford and David Ross
    Molecular Pharmacology December 2008, 74 (6) 1657-1665; DOI: https://doi.org/10.1124/mol.108.050401
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    P2Y1 Receptor Activation Elicits Its Partition out of Membrane Rafts and Its Rapid Internalization from Human Blood Vessels: Implications for Receptor Signaling
    Andrés Norambuena, M. Inés Poblete, M. Verónica Donoso, C. Sofía Espinoza, Alfonso González and J. Pablo Huidobro-Toro
    Molecular Pharmacology December 2008, 74 (6) 1666-1677; DOI: https://doi.org/10.1124/mol.108.048496
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    The Cannabinoid CB1 Receptor Antagonist Rimonabant Stimulates 2-Deoxyglucose Uptake in Skeletal Muscle Cells by Regulating the Expression of Phosphatidylinositol-3-kinase
    Iolanda Esposito, Maria Chiara Proto, Patrizia Gazzerro, Chiara Laezza, Claudia Miele, Anna Teresa Alberobello, Vittoria D'Esposito, Francesco Beguinot, Pietro Formisano and Maurizio Bifulco
    Molecular Pharmacology December 2008, 74 (6) 1678-1686; DOI: https://doi.org/10.1124/mol.108.049205
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    Tryptophan Mutations at Azi-Etomidate Photo-Incorporation Sites on α1 or β2 Subunits Enhance GABAA Receptor Gating and Reduce Etomidate Modulation
    Deirdre Stewart, Rooma Desai, Qi Cheng, Aiping Liu and Stuart A. Forman
    Molecular Pharmacology December 2008, 74 (6) 1687-1695; DOI: https://doi.org/10.1124/mol.108.050500
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    Potent Activation of Large-Conductance Ca2+-Activated K+ Channels by the Diphenylurea 1,3-Bis-[2-hydroxy-5-(trifluoromethyl)phenyl]urea (NS1643) in Pituitary Tumor (GH3) Cells
    Sheng-Nan Wu, Hsung Peng, Bing-Shuo Chen, Ya-Jean Wang, Pei-Yu Wu and Ming-Wei Lin
    Molecular Pharmacology December 2008, 74 (6) 1696-1704; DOI: https://doi.org/10.1124/mol.108.049106
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    Inhibitors of GlyT1 Affect Glycine Transport via Discrete Binding Sites
    Mario Mezler, Wilfried Hornberger, Reinhold Mueller, Martin Schmidt, Willi Amberg, Wilfried Braje, Michael Ochse, Hans Schoemaker and Berthold Behl
    Molecular Pharmacology December 2008, 74 (6) 1705-1715; DOI: https://doi.org/10.1124/mol.108.049312
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    The Selective Alzheimer's Disease Indicator-1 Gene (Seladin-1/DHCR24) Is a Liver X Receptor Target Gene
    Yongjun Wang, Pamela M. Rogers, Keith R. Stayrook, Chen Su, Gabor Varga, Qi Shen, Sunil Nagpal and Thomas P. Burris
    Molecular Pharmacology December 2008, 74 (6) 1716-1721; DOI: https://doi.org/10.1124/mol.108.048538
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    Mechanisms of Myocyte Cytotoxicity Induced by the Multiple Receptor Tyrosine Kinase Inhibitor Sunitinib
    Brian B. Hasinoff, Daywin Patel and Kimberley A. O'Hara
    Molecular Pharmacology December 2008, 74 (6) 1722-1728; DOI: https://doi.org/10.1124/mol.108.050104
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In this issue

Molecular Pharmacology: 74 (6)
Molecular Pharmacology
Vol. 74, Issue 6
1 Dec 2008
  • Table of Contents
  • Table of Contents (PDF)
  • About the Cover
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  • Back Matter (PDF)
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  • SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-β Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7
  • The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints
  • Pharmacological Properties of Y-27632, a Specific Inhibitor of Rho-Associated Kinases
  • Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
  • The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation of CYP3A4 by Rifampicin through a Distal Enhancer Module
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