Table of Contents

Articles

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  Naphtho[1,2-d]thiazol-2-ylamine (SKA-31), a New Activator of KCa2 and KCa3.1 Potassium Channels, Potentiates the Endothelium-Derived Hyperpolarizing Factor Response and Lowers Blood Pressure

  Ananthakrishnan Sankaranarayanan, Girija Raman, Christoph Busch, Tim Schultz, Pavel I. Zimin, Joachim Hoyer, Ralf Köhler and Heike Wulff

  Molecular Pharmacology February 2009, 75 (2) 281-295; DOI: https://doi.org/10.1124/mol.108.051425
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  Molecular Characterization of Novel and Selective Peroxisome Proliferator-Activated Receptor α Agonists with Robust Hypolipidemic Activity in Vivo

  Christopher D. Kane, Kimberly A. Stevens, James E. Fischer, Mehrdad Haghpassand, Lori J. Royer, Charles Aldinger, Katherine T. Landschulz, Panayiotis Zagouras, Scott W. Bagley, William Hada, Robert Dullea, Cheryl M. Hayward and Omar L. Francone

  Molecular Pharmacology February 2009, 75 (2) 296-306; DOI: https://doi.org/10.1124/mol.108.051656
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  Involvement of Transient Receptor Potential Vanilloid Subtype 1 in Analgesic Action of Methylsalicylate

  Toshio Ohta, Toshiaki Imagawa and Shigeo Ito

  Molecular Pharmacology February 2009, 75 (2) 307-317; DOI: https://doi.org/10.1124/mol.108.051292
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  Thermostable Variants of Cocaine Esterase for Long-Time Protection against Cocaine Toxicity

  Daquan Gao, Diwahar L. Narasimhan, Joanne Macdonald, Remy Brim, Mei-Chuan Ko, Donald W. Landry, James H. Woods, Roger K. Sunahara and Chang-Guo Zhan

  Molecular Pharmacology February 2009, 75 (2) 318-323; DOI: https://doi.org/10.1124/mol.108.049486
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  The Role of the Mammalian Copper Transporter 1 in the Cellular Accumulation of Platinum-Based Drugs

  Christopher A. Larson, Brian G. Blair, Roohangiz Safaei and Stephen B. Howell

  Molecular Pharmacology February 2009, 75 (2) 324-330; DOI: https://doi.org/10.1124/mol.108.052381
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  Mutagenic Mapping Suggests a Novel Binding Mode for Selective Agonists of M₁ Muscarinic Acetylcholine Receptors

  Guillaume Lebon, Christopher J. Langmead, Ben G. Tehan and Edward C. Hulme

  Molecular Pharmacology February 2009, 75 (2) 331-341; DOI: https://doi.org/10.1124/mol.108.050963
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  The Reelin and GAD67 Promoters Are Activated by Epigenetic Drugs That Facilitate the Disruption of Local Repressor Complexes

  Marija Kundakovic, Ying Chen, Alessandro Guidotti and Dennis R. Grayson

  Molecular Pharmacology February 2009, 75 (2) 342-354; DOI: https://doi.org/10.1124/mol.108.051763
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  Allosteric LFA-1 Inhibitors Modulate Natural Killer Cell Function

  Gabriele Weitz-Schmidt, Stéphanie Chreng and Simone Riek

  Molecular Pharmacology February 2009, 75 (2) 355-362; DOI: https://doi.org/10.1124/mol.108.051169
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  Preferential Physical and Functional Interaction of Pregnane X Receptor with the SMRTα Isoform

  Chia-Wei Li, Gia Khanh Dinh and J. Don Chen

  Molecular Pharmacology February 2009, 75 (2) 363-373; DOI: https://doi.org/10.1124/mol.108.047845
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  Pharmacological Analysis of the Novel, Rapid, and Potent Inactivation of the Human 5-Hydroxytryptamine₇ Receptor by Risperidone, 9-OH-Risperidone, and Other Inactivating Antagonists

  Jessica A. Knight, Carol Smith, Nicole Toohey, Michael T. Klein and Milt Teitler

  Molecular Pharmacology February 2009, 75 (2) 374-380; DOI: https://doi.org/10.1124/mol.108.052084
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  Estimation of Relative Microscopic Affinity Constants of Agonists for the Active State of the Receptor in Functional Studies on M₂ and M₃ Muscarinic Receptors

  John A. Tran, Alexander Chang, Minoru Matsui and Frederick J. Ehlert

  Molecular Pharmacology February 2009, 75 (2) 381-396; DOI: https://doi.org/10.1124/mol.108.051276
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  Multiple Roles of Charged Amino Acids in Cytoplasmic Loop 7 for Expression and Function of the Multidrug and Organic Anion Transporter MRP1 (ABCC1)

  Gwenaëlle Conseil, Alice J. Rothnie, Roger G. Deeley and Susan P. C. Cole

  Molecular Pharmacology February 2009, 75 (2) 397-406; DOI: https://doi.org/10.1124/mol.108.052860
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  Expression and 1,4-Dihydropyridine-Binding Properties of Brain L-Type Calcium Channel Isoforms

  Martina J. Sinnegger-Brauns, Irene G. Huber, Alexandra Koschak, Claudia Wild, Gerald J Obermair, Ursula Einzinger, Jean-Charles Hoda, Simone B. Sartori and Jörg Striessnig

  Molecular Pharmacology February 2009, 75 (2) 407-414; DOI: https://doi.org/10.1124/mol.108.049981
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  Relaxin Family Peptide Receptor (RXFP1) Coupling to Gα_i3 Involves the C-Terminal Arg⁷⁵² and Localization within Membrane Raft Microdomains

  Michelle L. Halls, Emma T. van der Westhuizen, John D. Wade, Bronwyn A. Evans, Ross A. D. Bathgate and Roger J. Summers

  Molecular Pharmacology February 2009, 75 (2) 415-428; DOI: https://doi.org/10.1124/mol.108.051227