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Molecular Pharmacology

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Table of Contents

March 01, 2009; Volume 75,Issue 3

MINIREVIEW

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    Pharmacological Targeting of the Integrated Protein Kinase B, Phosphatase and Tensin Homolog Deleted on Chromosome 10, and Transforming Growth Factor-β Pathways in Prostate Cancer
    Stephen J. Assinder, Qihan Dong, Helena Mangs and Des R. Richardson
    Molecular Pharmacology March 2009, 75 (3) 429-436; DOI: https://doi.org/10.1124/mol.108.053066

Accelerated Communications

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    5-Fluoro-2-indolyl des-chlorohalopemide (FIPI), a Phospholipase D Pharmacological Inhibitor That Alters Cell Spreading and Inhibits Chemotaxis
    Wenjuan Su, Oladapo Yeku, Srinivas Olepu, Alyssa Genna, Jae-Sook Park, Hongmei Ren, Guangwei Du, Michael H. Gelb, Andrew J. Morris and Michael A. Frohman
    Molecular Pharmacology March 2009, 75 (3) 437-446; DOI: https://doi.org/10.1124/mol.108.053298
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    D5 Dopamine Receptors are Required for Dopaminergic Activation of Phospholipase C
    Asha Sahu, Kimberly R. Tyeryar, Habiba O. Vongtau, David R. Sibley and Ashiwel S. Undieh
    Molecular Pharmacology March 2009, 75 (3) 447-453; DOI: https://doi.org/10.1124/mol.108.053017

Articles

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    Molecular Basis for the Selective Interaction of Synthetic Agonists with the Human Histamine H1-Receptor Compared with the Guinea Pig H1-Receptor
    Andrea Straßer, Hans-Joachim Wittmann, Marc Kunze, Sigurd Elz and Roland Seifert
    Molecular Pharmacology March 2009, 75 (3) 454-465; DOI: https://doi.org/10.1124/mol.108.053009
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    Canonical Transient Receptor Potential Channel (TRPC) 3 and TRPC6 Associate with Large-Conductance Ca2+-Activated K+ (BKCa) Channels: Role in BKCa Trafficking to the Surface of Cultured Podocytes
    Eun Young Kim, Claudia P. Alvarez-Baron and Stuart E. Dryer
    Molecular Pharmacology March 2009, 75 (3) 466-477; DOI: https://doi.org/10.1124/mol.108.051912
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    Cu/Zn Superoxide Dismutase Typical for Familial Amyotrophic Lateral Sclerosis Increases the Vulnerability of Mitochondria and Perturbs Ca2+ Homeostasis in SOD1G93A Mice
    Manoj Kumar Jaiswal and Bernhard U. Keller
    Molecular Pharmacology March 2009, 75 (3) 478-489; DOI: https://doi.org/10.1124/mol.108.050831
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    The Relative Activity of “Function Sparing” HIV-1 Entry Inhibitors on Viral Entry and CCR5 Internalization: Is Allosteric Functional Selectivity a Valuable Therapeutic Property?
    Vanessa M. Muniz-Medina, Stacey Jones, Jodi M. Maglich, Cristin Galardi, Robert E. Hollingsworth, Wieslaw M. Kazmierski, Robert G. Ferris, Mark P. Edelstein, Karen E. Chiswell and Terry P. Kenakin
    Molecular Pharmacology March 2009, 75 (3) 490-501; DOI: https://doi.org/10.1124/mol.108.052555
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    Evidence for a Direct and Functional Interaction between the Regulators of G Protein Signaling-2 and Phosphorylated C Terminus of Cholecystokinin-2 Receptor
    Ingrid Langer, Irina G. Tikhonova, Cyril Boulègue, Jean-Pierre Estève, Sébastien Vatinel, Audrey Ferrand, Luis Moroder, Patrick Robberecht and Daniel Fourmy
    Molecular Pharmacology March 2009, 75 (3) 502-513; DOI: https://doi.org/10.1124/mol.108.051607
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    A Juxtamembrane Mutation in the N Terminus of the Dopamine Transporter Induces Preference for an Inward-Facing Conformation
    Bipasha Guptaroy, Minjia Zhang, Erica Bowton, Francesca Binda, Lei Shi, Harel Weinstein, Aurelio Galli, Jonathan A. Javitch, Richard R. Neubig and Margaret E. Gnegy
    Molecular Pharmacology March 2009, 75 (3) 514-524; DOI: https://doi.org/10.1124/mol.108.048744
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    Butein Suppresses Constitutive and Inducible Signal Transducer and Activator of Transcription (STAT) 3 Activation and STAT3-Regulated Gene Products through the Induction of a Protein Tyrosine Phosphatase SHP-1
    Manoj K. Pandey, Bokyung Sung, Kwang Seok Ahn and Bharat B. Aggarwal
    Molecular Pharmacology March 2009, 75 (3) 525-533; DOI: https://doi.org/10.1124/mol.108.052548
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    Fluorescence Resonance Energy Transfer Analysis of α2a-Adrenergic Receptor Activation Reveals Distinct Agonist-Specific Conformational Changes
    A. Zürn, U. Zabel, J.-P. Vilardaga, H. Schindelin, M. J. Lohse and C. Hoffmann
    Molecular Pharmacology March 2009, 75 (3) 534-541; DOI: https://doi.org/10.1124/mol.108.052399
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    Mechanisms and Functional Significance of Inhibition of Neuronal T-Type Calcium Channels by Isoflurane
    Peihan Orestes, Damir Bojadzic, Robert M. Chow and Slobodan M. Todorovic
    Molecular Pharmacology March 2009, 75 (3) 542-554; DOI: https://doi.org/10.1124/mol.108.051664
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    Knock-In Mouse Lines Expressing either Mitochondrial or Microsomal CYP1A1: Differing Responses to Dietary Benzo[a]pyrene as Proof of Principle
    Hongbin Dong, Timothy P. Dalton, Marian L. Miller, Ying Chen, Shigeyuki Uno, Zhanquan Shi, Howard G. Shertzer, Seema Bansal, Narayan G. Avadhani and Daniel W. Nebert
    Molecular Pharmacology March 2009, 75 (3) 555-567; DOI: https://doi.org/10.1124/mol.108.051888
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    Analysis of DNA Methylation and Histone Modification Profiles of Liver-Specific Transporters
    Satoki Imai, Ryota Kikuchi, Hiroyuki Kusuhara, Shintaro Yagi, Kunio Shiota and Yuichi Sugiyama
    Molecular Pharmacology March 2009, 75 (3) 568-576; DOI: https://doi.org/10.1124/mol.108.052589
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    Discovery and Characterization of Novel Allosteric Potentiators of M1 Muscarinic Receptors Reveals Multiple Modes of Activity
    Joy E. Marlo, Colleen M. Niswender, Emily L. Days, Thomas M. Bridges, Yun Xiang, Alice L. Rodriguez, Jana K. Shirey, Ashley E. Brady, Tasha Nalywajko, Qingwei Luo, Cheryl A. Austin, Michael Baxter Williams, Kwangho Kim, Richard Williams, Darren Orton, H. Alex Brown, Craig W. Lindsley, C. David Weaver and P. Jeffrey Conn
    Molecular Pharmacology March 2009, 75 (3) 577-588; DOI: https://doi.org/10.1124/mol.108.052886
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    Identification of an Activator Protein-1-Like Sequence as the Glucocorticoid Response Element in the Rat Tyrosine Hydroxylase Gene
    C. S. Sheela Rani, Narayanasamy Elango, Shou-shu Wang, Kazuto Kobayashi and Randy Strong
    Molecular Pharmacology March 2009, 75 (3) 589-598; DOI: https://doi.org/10.1124/mol.108.051219
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    Psoralen-Induced DNA Interstrand Cross-Links Block Transcription and Induce p53 in an Ataxia-Telangiectasia and Rad3-Related-Dependent Manner
    Frederick A. Derheimer, J. Kevin Hicks, Michelle T. Paulsen, Christine E. Canman and Mats Ljungman
    Molecular Pharmacology March 2009, 75 (3) 599-607; DOI: https://doi.org/10.1124/mol.108.051698
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    Phospholipase C-Mediated Regulation of Transient Receptor Potential Vanilloid 6 Channels: Implications in Active Intestinal Ca2+ Transport
    Baskaran Thyagarajan, Bryan S. Benn, Sylvia Christakos and Tibor Rohacs
    Molecular Pharmacology March 2009, 75 (3) 608-616; DOI: https://doi.org/10.1124/mol.108.052449
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    Synthetic Small-Molecule Prohormone Convertase 2 Inhibitors
    Dorota Kowalska, Jin Liu, Jon R. Appel, Akihiko Ozawa, Adel Nefzi, Robert B. Mackin, Richard A. Houghten and Iris Lindberg
    Molecular Pharmacology March 2009, 75 (3) 617-625; DOI: https://doi.org/10.1124/mol.108.051334
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    Reciprocal Regulation of the Platelet-Derived Growth Factor Receptor-β and G Protein-Coupled Receptor Kinase 5 by Cross-Phosphorylation: Effects on Catalysis
    Xinjiang Cai, Jiao-Hui Wu, Sabrina T. Exum, Martin Oppermann, Richard T. Premont, Sudha K. Shenoy and Neil J. Freedman
    Molecular Pharmacology March 2009, 75 (3) 626-636; DOI: https://doi.org/10.1124/mol.108.050278
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    Differential Coupling of the Vasopressin V1b Receptor through Compartmentalization within the Plasma Membrane
    Hélène Orcel, Laura Albizu, Sanja Perkovska, Thierry Durroux, Christiane Mendre, Hervé Ansanay, Bernard Mouillac and Alain Rabié
    Molecular Pharmacology March 2009, 75 (3) 637-647; DOI: https://doi.org/10.1124/mol.108.049031
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    Molecular Mechanisms of Corticotropin-Releasing Factor Receptor-Induced Calcium Signaling
    Eric Gutknecht, Ilse Van der Linden, Kristof Van Kolen, Kim F. C. Verhoeven, Georges Vauquelin and Frank M. Dautzenberg
    Molecular Pharmacology March 2009, 75 (3) 648-657; DOI: https://doi.org/10.1124/mol.108.050427
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    Quantification of Focal Adhesion Kinase Activation Loop Phosphorylation as a Biomarker of Src Activity
    Eugene Ciccimaro, Steven K. Hanks and Ian A. Blair
    Molecular Pharmacology March 2009, 75 (3) 658-666; DOI: https://doi.org/10.1124/mol.108.052464
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    Heterocyclic Thioureylenes Protect from Calcium-Dependent Neuronal Cell Death
    Matjaz Humar, Christine Graetz, Martin Roesslein, Ulrich Goebel, Klaus K. Geiger, Bernd Heimrich and Benedikt H. J. Pannen
    Molecular Pharmacology March 2009, 75 (3) 667-676; DOI: https://doi.org/10.1124/mol.108.052183
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    Unveiling a New Essential Cis Element for the Transactivation of the CYP3A4 Gene by Xenobiotics
    Takayoshi Toriyabe, Kiyoshi Nagata, Tomonari Takada, Yusuke Aratsu, Tsutomu Matsubara, Kouichi Yoshinari and Yasushi Yamazoe
    Molecular Pharmacology March 2009, 75 (3) 677-684; DOI: https://doi.org/10.1124/mol.108.050575
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    Angiotensin-Converting Enzyme (ACE) Inhibitors Modulate Cellular Retinol-Binding Protein 1 and Adiponectin Expression in Adipocytes via the ACE-Dependent Signaling Cascade
    Karin Kohlstedt, Cynthia Gershome, Caroline Trouvain, Wolf-Karsten Hofmann, Stephan Fichtlscherer and Ingrid Fleming
    Molecular Pharmacology March 2009, 75 (3) 685-692; DOI: https://doi.org/10.1124/mol.108.051631
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    Molecular Analysis of the Interaction of Anthrax Adenylyl Cyclase Toxin, Edema Factor, with 2′(3′)-O-(N-(methyl)anthraniloyl)-Substituted Purine and Pyrimidine Nucleotides
    Hesham M. Taha, Jennifer Schmidt, Martin Göttle, Srividya Suryanarayana, Yuequan Shen, Wei-Jen Tang, Andreas Gille, Jens Geduhn, Burkhard König, Stefan Dove and Roland Seifert
    Molecular Pharmacology March 2009, 75 (3) 693-703; DOI: https://doi.org/10.1124/mol.108.052340
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    Desipramine Reduces Stress-Activated Dynorphin Expression and CREB Phosphorylation in NAc Tissue
    Elena H. Chartoff, Maria Papadopoulou, Matt L. MacDonald, Aram Parsegian, David Potter, Christine Konradi and William A. Carlezon
    Molecular Pharmacology March 2009, 75 (3) 704-712; DOI: https://doi.org/10.1124/mol.108.051417
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    Facilitatory Interplay in α1a and β2 Adrenoceptor Function Reveals a Non-Gq Signaling Mode: Implications for Diversification of Intracellular Signal Transduction
    Alicja J. Copik, Cynthia Ma, Alan Kosaka, Sunil Sahdeo, Andy Trane, Hoangdung Ho, Paul S. Dietrich, Helen Yu, Anthony P. D. W. Ford, Donald Button and Marcos E. Milla
    Molecular Pharmacology March 2009, 75 (3) 713-728; DOI: https://doi.org/10.1124/mol.108.050765

Errata

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    Correction to “A Dopamine D2 Receptor Mutant Capable of G Protein-Mediated Signaling but Deficient in Arrestin Binding”
    Molecular Pharmacology March 2009, 75 (3) 729; DOI: https://doi.org/10.1124/mol.75.3.729
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    Correction to “Protease-Activated Receptors Differentially Regulate Human Platelet Activation through a Phosphatidic Acid-Dependent Pathway”
    Molecular Pharmacology March 2009, 75 (3) 730-731; DOI: https://doi.org/10.1124/mol.75.3.730
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Molecular Pharmacology: 75 (3)
Molecular Pharmacology
Vol. 75, Issue 3
1 Mar 2009
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