Table of Contents

Articles

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  Contribution of Binding Enthalpy and Entropy to Affinity of Antagonist and Agonist Binding at Human and Guinea Pig Histamine H₁-Receptor

  Hans-Joachim Wittmann, Roland Seifert and Andrea Strasser

  Molecular Pharmacology July 2009, 76 (1) 25-37; DOI: https://doi.org/10.1124/mol.109.055384
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  Regulation of Renal Outer Medullary Potassium Channel and Renal K⁺ Excretion by Klotho

  Seung-Kuy Cha, Ming-Chang Hu, Hiroshi Kurosu, Makoto Kuro-o, Orson Moe and Chou-Long Huang

  Molecular Pharmacology July 2009, 76 (1) 38-46; DOI: https://doi.org/10.1124/mol.109.055780
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  Thiazolidinediones Mimic Glucose Starvation in Facilitating Sp1 Degradation through the Up-Regulation of β-Transducin Repeat-Containing Protein

  Shuo Wei, Hsiao-Ching Chuang, Wan-Chi Tsai, Hsiao-Ching Yang, Shiuh-Rong Ho, Andrew J. Paterson, Samuel K. Kulp and Ching-Shih Chen

  Molecular Pharmacology July 2009, 76 (1) 47-57; DOI: https://doi.org/10.1124/mol.109.055376
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  In Vivo and in Vitro Structure-Activity Relationships and Structural Conformation of Kisspeptin-10-Related Peptides

  Ester Gutiérrez-Pascual, Jérôme Leprince, Antonio J. Martínez-Fuentes, Isabelle Ségalas-Milazzo, Rafael Pineda, Juan Roa, Mario Duran-Prado, Laure Guilhaudis, Elia Desperrois, Aurélie Lebreton, Leonor Pinilla, Marie-Christine Tonon, María M. Malagón, Hubert Vaudry, Manuel Tena-Sempere and Justo P. Castaño

  Molecular Pharmacology July 2009, 76 (1) 58-67; DOI: https://doi.org/10.1124/mol.108.053751
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  Site Specificity of Agonist and Second Messenger-Activated Kinases for Somatostatin Receptor Subtype 2A (Sst2A) Phosphorylation

  Qisheng Liu, Mark S. Bee and Agnes Schonbrunn

  Molecular Pharmacology July 2009, 76 (1) 68-80; DOI: https://doi.org/10.1124/mol.108.054262
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  Polyethylene Glycosylated Curcumin Conjugate Inhibits Pancreatic Cancer Cell Growth through Inactivation of Jab1

  Jun Li, Yun Wang, Chaozhe Yang, Pengfei Wang, Denise K. Oelschlager, Yong Zheng, De-An Tian, William E. Grizzle, Donald J. Buchsbaum and Mei Wan

  Molecular Pharmacology July 2009, 76 (1) 81-90; DOI: https://doi.org/10.1124/mol.109.054551
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  Apratoxin A Reversibly Inhibits the Secretory Pathway by Preventing Cotranslational Translocation

  Yanxia Liu, Brian K. Law and Hendrik Luesch

  Molecular Pharmacology July 2009, 76 (1) 91-104; DOI: https://doi.org/10.1124/mol.109.056085
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  Inhibition of Aquaporin-1 and Aquaporin-4 Water Permeability by a Derivative of the Loop Diuretic Bumetanide Acting at an Internal Pore-Occluding Binding Site

  Elton Migliati, Nathalie Meurice, Pascale DuBois, Jennifer S. Fang, Suma Somasekharan, Elizabeth Beckett, Gary Flynn and Andrea J. Yool

  Molecular Pharmacology July 2009, 76 (1) 105-112; DOI: https://doi.org/10.1124/mol.108.053744
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  The Spermostatic and Microbicidal Actions of Quinones and Maleimides: Toward a Dual-Purpose Contraceptive Agent

  Louise M. Hughes, Renate Griffith, Alison Carey, Trent Butler, Scott W. Donne, Ken W. Beagley and R. John Aitken

  Molecular Pharmacology July 2009, 76 (1) 113-124; DOI: https://doi.org/10.1124/mol.108.053645
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  S3b Amino Acid Substitutions and Ancillary Subunits Alter the Affinity of Heteropoda venatoria Toxin 2 for Kv4.3

  Christopher V. DeSimone, YiChun Lu, Vladimir E. Bondarenko and Michael J. Morales

  Molecular Pharmacology July 2009, 76 (1) 125-133; DOI: https://doi.org/10.1124/mol.109.055657
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  δ Receptors Are Required for Full Inhibitory Coupling of μ Receptors to Voltage-Dependent Ca²⁺ Channels in Dorsal Root Ganglion Neurons

  Wendy Walwyn, Scott John, Matthew Maga, Christopher J. Evans and Tim G. Hales

  Molecular Pharmacology July 2009, 76 (1) 134-143; DOI: https://doi.org/10.1124/mol.109.055913
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  α₁-Adrenergic Receptor Stimulates Interleukin-6 Expression and Secretion through Both mRNA Stability and Transcriptional Regulation: Involvement of p38 Mitogen-Activated Protein Kinase and Nuclear Factor-κB

  Dianne M. Perez, Robert S. Papay and Ting Shi

  Molecular Pharmacology July 2009, 76 (1) 144-152; DOI: https://doi.org/10.1124/mol.108.054320
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  KLYP956 Is a Non-Imidazole-Based Orally Active Inhibitor of Nitric-Oxide Synthase Dimerization

  Kent T. Symons, Mark E. Massari, Phan M. Nguyen, Tom T. Lee, Jeffrey Roppe, Céline Bonnefous, Joseph E. Payne, Nicholas D. Smith, Stewart A. Noble, Marciano Sablad, Natasha Rozenkrants, Yan Zhang, Tadimeti S. Rao, Andrew K. Shiau and Christian A. Hassig

  Molecular Pharmacology July 2009, 76 (1) 153-162; DOI: https://doi.org/10.1124/mol.109.055434
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  Potent Activity of Indolequinones against Human Pancreatic Cancer: Identification of Thioredoxin Reductase as a Potential Target

  Chao Yan, Biehuoy Shieh, Philip Reigan, Zhiyong Zhang, Marie A. Colucci, Aurélie Chilloux, Jeffery J. Newsome, David Siegel, Dan Chan, Christopher J. Moody and David Ross

  Molecular Pharmacology July 2009, 76 (1) 163-172; DOI: https://doi.org/10.1124/mol.109.055855
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  Heme-Oxygenase-1 Induction and Carbon Monoxide-Releasing Molecule Inhibit Lipopolysaccharide (LPS)-Induced High-Mobility Group Box 1 Release in Vitro and Improve Survival of Mice in LPS- and Cecal Ligation and Puncture-Induced Sepsis Model in Vivo

  Konstantin Tsoyi, Tae Yu Lee, Young Soo Lee, Hye Jung Kim, Han Geuk Seo, Jae Heun Lee and Ki Churl Chang

  Molecular Pharmacology July 2009, 76 (1) 173-182; DOI: https://doi.org/10.1124/mol.109.055137
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  Mesalamine Suppresses the Expression of TC22, a Novel Tropomyosin Isoform Associated with Colonic Neoplasia

  Koushik K. Das, Manisha Bajpai, Yingxin Kong, Jianying Liu, Xin Geng and Kiron M. Das

  Molecular Pharmacology July 2009, 76 (1) 183-191; DOI: https://doi.org/10.1124/mol.109.056028
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  S-Adenosylmethionine and Methylthioadenosine Inhibit Cellular FLICE Inhibitory Protein Expression and Induce Apoptosis in Colon Cancer Cells

  Tony W. H. Li, Qingsong Zhang, Pilsoo Oh, Meng Xia, Hui Chen, Sean Bemanian, Natalie Lastra, Magda Circ, Mary Pat Moyer, José M. Mato, Tak Yee Aw and Shelly C. Lu

  Molecular Pharmacology July 2009, 76 (1) 192-200; DOI: https://doi.org/10.1124/mol.108.054411
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  Activation Switch in the Transmembrane Domain of Metabotropic Glutamate Receptor

  Masataka Yanagawa, Takahiro Yamashita and Yoshinori Shichida

  Molecular Pharmacology July 2009, 76 (1) 201-207; DOI: https://doi.org/10.1124/mol.109.056549
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  Cisplatin-Induced DNA Damage Activates Replication Checkpoint Signaling Components that Differentially Affect Tumor Cell Survival

  Jill M. Wagner and Larry M. Karnitz

  Molecular Pharmacology July 2009, 76 (1) 208-214; DOI: https://doi.org/10.1124/mol.109.055178