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Index by author

December 01, 2009; Volume 76,Issue 6

A

  1. Alvarez, Rosana

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  2. Alvarez, Susana

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  3. Arnold, Andy

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

B

  1. Bailly, Christian

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  2. Barrett, Matthew O.

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  3. Blagg, Brian S. J.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  4. Bonci, Antonello

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  5. Bradley, Sophie J.

    1. Effects of Positive Allosteric Modulators on Single-Cell Oscillatory Ca2+ Signaling Initiated by the Type 5 Metabotropic Glutamate Receptor
      Sophie J. Bradley, Jeannette M. Watson and R. A. John Challiss
      Molecular Pharmacology December 2009, 76 (6) 1302-1313; DOI: https://doi.org/10.1124/mol.109.059170

  6. Brazier, Michel

    1. Agonists and Allosteric Modulators of the Calcium-Sensing Receptor and Their Therapeutic Applications
      Zuzana Saidak, Michel Brazier, Saïd Kamel and Romuald Mentaverri
      Molecular Pharmacology December 2009, 76 (6) 1131-1144; DOI: https://doi.org/10.1124/mol.109.058784

  7. Buchmayer, Florian

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  8. Burianek, Lauren E.

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

C

  1. Cankurtaran-Sayar, Serife

    1. P2X7 Receptor Activates Multiple Selective Dye-Permeation Pathways in RAW 264.7 and Human Embryonic Kidney 293 Cells
      Serife Cankurtaran-Sayar, Kemal Sayar and Mehmet Ugur
      Molecular Pharmacology December 2009, 76 (6) 1323-1332; DOI: https://doi.org/10.1124/mol.109.059923

  2. Carter, Rhonda L.

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  3. Challiss, R. A. John

    1. Effects of Positive Allosteric Modulators on Single-Cell Oscillatory Ca2+ Signaling Initiated by the Type 5 Metabotropic Glutamate Receptor
      Sophie J. Bradley, Jeannette M. Watson and R. A. John Challiss
      Molecular Pharmacology December 2009, 76 (6) 1302-1313; DOI: https://doi.org/10.1124/mol.109.059170

  4. Chen, Cheng-Hsien

    1. Urotensin II Induces Rat Cardiomyocyte Hypertrophy via the Transient Oxidization of Src Homology 2-Containing Tyrosine Phosphatase and Transactivation of Epidermal Growth Factor Receptor
      Ju-Chi Liu, Cheng-Hsien Chen, Jin-Jer Chen and Tzu-Hurng Cheng
      Molecular Pharmacology December 2009, 76 (6) 1186-1195; DOI: https://doi.org/10.1124/mol.109.058297

  5. Chen, Jin-Jer

    1. Urotensin II Induces Rat Cardiomyocyte Hypertrophy via the Transient Oxidization of Src Homology 2-Containing Tyrosine Phosphatase and Transactivation of Epidermal Growth Factor Receptor
      Ju-Chi Liu, Cheng-Hsien Chen, Jin-Jer Chen and Tzu-Hurng Cheng
      Molecular Pharmacology December 2009, 76 (6) 1186-1195; DOI: https://doi.org/10.1124/mol.109.058297

  6. Chen, Ligong

    1. Regulation of Serotonin 1B Receptor by Glycogen Synthase Kinase-3
      Ligong Chen, Gregory D. Salinas and Xiaohua Li
      Molecular Pharmacology December 2009, 76 (6) 1150-1161; DOI: https://doi.org/10.1124/mol.109.056994

  7. Cheng, Tzu-Hurng

    1. Urotensin II Induces Rat Cardiomyocyte Hypertrophy via the Transient Oxidization of Src Homology 2-Containing Tyrosine Phosphatase and Transactivation of Epidermal Growth Factor Receptor
      Ju-Chi Liu, Cheng-Hsien Chen, Jin-Jer Chen and Tzu-Hurng Cheng
      Molecular Pharmacology December 2009, 76 (6) 1186-1195; DOI: https://doi.org/10.1124/mol.109.058297

  8. Chiaroni, Angèle

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  9. Cho, Yoshitake

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

  10. Choi, Mihwa

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

  11. Cravatt, Benjamin F.

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

D

  1. Das, Arijit

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  2. Dascal, Nathan

    1. N Terminus of Type 5 Adenylyl Cyclase Scaffolds Gs Heterotrimer
      Rachna Sadana, Nathan Dascal and Carmen W. Dessauer
      Molecular Pharmacology December 2009, 76 (6) 1256-1264; DOI: https://doi.org/10.1124/mol.109.058370

  3. David-Cordonnier, Marie-Hélène

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  4. de Lera, Angel R.

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  5. Depauw, Sabine

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  6. Dessauer, Carmen W.

    1. N Terminus of Type 5 Adenylyl Cyclase Scaffolds Gs Heterotrimer
      Rachna Sadana, Nathan Dascal and Carmen W. Dessauer
      Molecular Pharmacology December 2009, 76 (6) 1256-1264; DOI: https://doi.org/10.1124/mol.109.058370

  7. Dingledine, Raymond

    1. Control of Glutamate Receptor 2 (GluR2) Translational Initiation by Its Alternative 3′ Untranslated Regions
      Hasan A. Irier, Yi Quan, Justin Yoo and Raymond Dingledine
      Molecular Pharmacology December 2009, 76 (6) 1145-1149; DOI: https://doi.org/10.1124/mol.109.060343

  8. Domínguez, Marta

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  9. Donnelly, Alison C.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

E

  1. Enyeart, John J.

    1. N6-Substituted cAMP Analogs Inhibit bTREK-1 K+ Channels and Stimulate Cortisol Secretion by a Protein Kinase A-Independent Mechanism
      Haiyan Liu, Judith A. Enyeart and John J. Enyeart
      Molecular Pharmacology December 2009, 76 (6) 1290-1301; DOI: https://doi.org/10.1124/mol.109.057075

  2. Enyeart, Judith A.

    1. N6-Substituted cAMP Analogs Inhibit bTREK-1 K+ Channels and Stimulate Cortisol Secretion by a Protein Kinase A-Independent Mechanism
      Haiyan Liu, Judith A. Enyeart and John J. Enyeart
      Molecular Pharmacology December 2009, 76 (6) 1290-1301; DOI: https://doi.org/10.1124/mol.109.057075

F

  1. Freissmuth, Michael

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  2. Fricks, Ingrid P.

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  3. Fujimoto, Katsumi

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

G

  1. Gachet, Christian

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  2. Gaslonde, Thomas

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  3. Gaubitzer, Erwin

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  4. Golczak, Marcin

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  5. Gsandtner, Ingrid

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

H

  1. Hancock, Jane

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

  2. Harden, T. Kendall

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  3. He, Xiaoqing

    1. NRF2 Cysteine Residues Are Critical for Oxidant/Electrophile-Sensing, Kelch-Like ECH-Associated Protein-1-Dependent Ubiquitination-Proteasomal Degradation, and Transcription Activation
      Xiaoqing He and Qiang Ma
      Molecular Pharmacology December 2009, 76 (6) 1265-1278; DOI: https://doi.org/10.1124/mol.109.058453

  4. Hobson, Sally A.

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

  5. Hoffmann, Carsten

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  6. Hu, Sherry Shu-Jung

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

I

  1. Irier, Hasan A.

    1. Control of Glutamate Receptor 2 (GluR2) Translational Initiation by Its Alternative 3′ Untranslated Regions
      Hasan A. Irier, Yi Quan, Justin Yoo and Raymond Dingledine
      Molecular Pharmacology December 2009, 76 (6) 1145-1149; DOI: https://doi.org/10.1124/mol.109.060343

J

  1. Jacobson, Kenneth A.

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

K

  1. Kamel, Saïd

    1. Agonists and Allosteric Modulators of the Calcium-Sensing Receptor and Their Therapeutic Applications
      Zuzana Saidak, Michel Brazier, Saïd Kamel and Romuald Mentaverri
      Molecular Pharmacology December 2009, 76 (6) 1131-1144; DOI: https://doi.org/10.1124/mol.109.058784

  2. Karpushev, Alexey V.

    1. Peroxisome Proliferator-Activated Receptor γ Antagonists Decrease Na+ Transport via the Epithelial Na+ Channel
      Tengis S. Pavlov, Vladislav Levchenko, Alexey V. Karpushev, Alain Vandewalle and Alexander Staruschenko
      Molecular Pharmacology December 2009, 76 (6) 1333-1340; DOI: https://doi.org/10.1124/mol.109.056911

  3. Kato, Yukio

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

  4. Kawamoto, Takeshi

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

  5. Kelly, Eamonn

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

  6. Ko, Hyojin

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  7. Köhler, Gottfried

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  8. Kraus-Berthier, Laurence

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

L

  1. Laine, William

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  2. Lazarowski, Eduardo R.

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  3. Lazo, John S.

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

  4. Lenglet, Gaëlle

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  5. Leon, Catherine

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  6. Léonce, Stéphane

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  7. Levchenko, Vladislav

    1. Peroxisome Proliferator-Activated Receptor γ Antagonists Decrease Na+ Transport via the Epithelial Na+ Channel
      Tengis S. Pavlov, Vladislav Levchenko, Alexey V. Karpushev, Alain Vandewalle and Alexander Staruschenko
      Molecular Pharmacology December 2009, 76 (6) 1333-1340; DOI: https://doi.org/10.1124/mol.109.056911

  8. Levesque, Paul

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  9. Lewen, Michael D.

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

  10. Li, Danshi

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  11. Li, Julia

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  12. Li, Xiaohua

    1. Regulation of Serotonin 1B Receptor by Glycogen Synthase Kinase-3
      Ligong Chen, Gregory D. Salinas and Xiaohua Li
      Molecular Pharmacology December 2009, 76 (6) 1150-1161; DOI: https://doi.org/10.1124/mol.109.056994

  13. Liu, Haiyan

    1. N6-Substituted cAMP Analogs Inhibit bTREK-1 K+ Channels and Stimulate Cortisol Secretion by a Protein Kinase A-Independent Mechanism
      Haiyan Liu, Judith A. Enyeart and John J. Enyeart
      Molecular Pharmacology December 2009, 76 (6) 1290-1301; DOI: https://doi.org/10.1124/mol.109.057075

  14. Liu, Ju-Chi

    1. Urotensin II Induces Rat Cardiomyocyte Hypertrophy via the Transient Oxidization of Src Homology 2-Containing Tyrosine Phosphatase and Transactivation of Epidermal Growth Factor Receptor
      Ju-Chi Liu, Cheng-Hsien Chen, Jin-Jer Chen and Tzu-Hurng Cheng
      Molecular Pharmacology December 2009, 76 (6) 1186-1195; DOI: https://doi.org/10.1124/mol.109.058297

  15. Lobo, Glenn P.

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  16. Lohse, Martin J.

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  17. Long, Jonathan Z.

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

  18. Lorenz, Kristina

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  19. Lu, Yuanming

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

M

  1. Ma, Qiang

    1. NRF2 Cysteine Residues Are Critical for Oxidant/Electrophile-Sensing, Kelch-Like ECH-Associated Protein-1-Dependent Ubiquitination-Proteasomal Degradation, and Transcription Activation
      Xiaoqing He and Qiang Ma
      Molecular Pharmacology December 2009, 76 (6) 1265-1278; DOI: https://doi.org/10.1124/mol.109.058453

  2. Mackie, Ken

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

  3. Makishima, Makoto

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

  4. Mandal, Madhuchhanda

    1. Phosphatidylinositol (4,5)-Bisphosphate Regulation of N-Methyl-d-aspartate Receptor Channels in Cortical Neurons
      Madhuchhanda Mandal and Zhen Yan
      Molecular Pharmacology December 2009, 76 (6) 1349-1359; DOI: https://doi.org/10.1124/mol.109.058701

  5. Marrion, Neil V.

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

  6. Mason, Angharad

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

  7. Matthews, Shawna B.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  8. Matts, Robert L.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  9. McDonald, Peter R.

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

  10. Mentaverri, Romuald

    1. Agonists and Allosteric Modulators of the Calcium-Sensing Receptor and Their Therapeutic Applications
      Zuzana Saidak, Michel Brazier, Saïd Kamel and Romuald Mentaverri
      Molecular Pharmacology December 2009, 76 (6) 1131-1144; DOI: https://doi.org/10.1124/mol.109.058784

  11. Michel, Sylvie

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  12. Milan-Lobo, Laura

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  13. Miller, Keith J.

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  14. Moise, Alexander R.

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  15. Morita, Kentaro

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

N

  1. Noshiro, Mitsuhide

    1. The Basic Helix-Loop-Helix Proteins Differentiated Embryo Chondrocyte (DEC) 1 and DEC2 Function as Corepressors of Retinoid X Receptors
      Yoshitake Cho, Mitsuhide Noshiro, Mihwa Choi, Kentaro Morita, Takeshi Kawamoto, Katsumi Fujimoto, Yukio Kato and Makoto Makishima
      Molecular Pharmacology December 2009, 76 (6) 1360-1369; DOI: https://doi.org/10.1124/mol.109.057000

O

  1. Oldfield, Susan

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

P

  1. Palczewski, Krzysztof

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

  2. Pavlov, Tengis S.

    1. Peroxisome Proliferator-Activated Receptor γ Antagonists Decrease Na+ Transport via the Epithelial Na+ Channel
      Tengis S. Pavlov, Vladislav Levchenko, Alexey V. Karpushev, Alain Vandewalle and Alexander Staruschenko
      Molecular Pharmacology December 2009, 76 (6) 1333-1340; DOI: https://doi.org/10.1124/mol.109.056911

  3. Pfeiffer, Bruno

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  4. Pierré, Alain

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

  5. Pollack, Ian F.

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

Q

  1. Quan, Yi

    1. Control of Glutamate Receptor 2 (GluR2) Translational Initiation by Its Alternative 3′ Untranslated Regions
      Hasan A. Irier, Yi Quan, Justin Yoo and Raymond Dingledine
      Molecular Pharmacology December 2009, 76 (6) 1145-1149; DOI: https://doi.org/10.1124/mol.109.060343

R

  1. Rajewski, Roger A.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  2. Randall, Andrew D.

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

  3. Reiner, Susanne

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  4. Robertson, John D.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  5. Robl, Jeffrey A.

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  6. Rossi, Karen A.

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  7. Rünzler, Dominik

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

S

  1. Sadana, Rachna

    1. N Terminus of Type 5 Adenylyl Cyclase Scaffolds Gs Heterotrimer
      Rachna Sadana, Nathan Dascal and Carmen W. Dessauer
      Molecular Pharmacology December 2009, 76 (6) 1256-1264; DOI: https://doi.org/10.1124/mol.109.058370

  2. Saidak, Zuzana

    1. Agonists and Allosteric Modulators of the Calcium-Sensing Receptor and Their Therapeutic Applications
      Zuzana Saidak, Michel Brazier, Saïd Kamel and Romuald Mentaverri
      Molecular Pharmacology December 2009, 76 (6) 1131-1144; DOI: https://doi.org/10.1124/mol.109.058784

  3. Salinas, Gregory D.

    1. Regulation of Serotonin 1B Receptor by Glycogen Synthase Kinase-3
      Ligong Chen, Gregory D. Salinas and Xiaohua Li
      Molecular Pharmacology December 2009, 76 (6) 1150-1161; DOI: https://doi.org/10.1124/mol.109.056994

  4. Sayar, Kemal

    1. P2X7 Receptor Activates Multiple Selective Dye-Permeation Pathways in RAW 264.7 and Human Embryonic Kidney 293 Cells
      Serife Cankurtaran-Sayar, Kemal Sayar and Mehmet Ugur
      Molecular Pharmacology December 2009, 76 (6) 1323-1332; DOI: https://doi.org/10.1124/mol.109.059923

  5. Shawgo, Mary E.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  6. Shelton, Shary N.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  7. Shen, Yan

    1. An Anticancer Effect of Curcumin Mediated by Down-Regulating Phosphatase of Regenerating Liver-3 Expression on Highly Metastatic Melanoma Cells
      Lu Wang, Yan Shen, Ran Song, Yang Sun, Jianliang Xu and Qiang Xu
      Molecular Pharmacology December 2009, 76 (6) 1238-1245; DOI: https://doi.org/10.1124/mol.109.059105

  8. Shun, Tong Ying

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

  9. Sitte, Harald H.

    1. Subtype-Specific Differences in Corticotropin-Releasing Factor Receptor Complexes Detected by Fluorescence Spectroscopy
      Laura Milan-Lobo, Ingrid Gsandtner, Erwin Gaubitzer, Dominik Rünzler, Florian Buchmayer, Gottfried Köhler, Antonello Bonci, Michael Freissmuth and Harald H. Sitte
      Molecular Pharmacology December 2009, 76 (6) 1196-1210; DOI: https://doi.org/10.1124/mol.109.059139

  10. Song, Ran

    1. An Anticancer Effect of Curcumin Mediated by Down-Regulating Phosphatase of Regenerating Liver-3 Expression on Highly Metastatic Melanoma Cells
      Lu Wang, Yan Shen, Ran Song, Yang Sun, Jianliang Xu and Qiang Xu
      Molecular Pharmacology December 2009, 76 (6) 1238-1245; DOI: https://doi.org/10.1124/mol.109.059105

  11. Staruschenko, Alexander

    1. Peroxisome Proliferator-Activated Receptor γ Antagonists Decrease Na+ Transport via the Epithelial Na+ Channel
      Tengis S. Pavlov, Vladislav Levchenko, Alexey V. Karpushev, Alain Vandewalle and Alexander Staruschenko
      Molecular Pharmacology December 2009, 76 (6) 1333-1340; DOI: https://doi.org/10.1124/mol.109.056911

  12. Straiker, Alex

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

  13. Sun, Yang

    1. An Anticancer Effect of Curcumin Mediated by Down-Regulating Phosphatase of Regenerating Liver-3 Expression on Highly Metastatic Melanoma Cells
      Lu Wang, Yan Shen, Ran Song, Yang Sun, Jianliang Xu and Qiang Xu
      Molecular Pharmacology December 2009, 76 (6) 1238-1245; DOI: https://doi.org/10.1124/mol.109.059105

  14. Szabla, Kristen

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

T

  1. Tanol, Mehmet

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  2. Thaker, Nikhil G.

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

  3. Tillequin, François

    1. Influence of the Stereoisomeric Position of the Reactive Acetate Groups of the Benzo[b]Acronycine derivative S23906-1 on Its DNA Alkylation, Helix-Opening, Cytotoxic, and Antitumor Activities
      Sabine Depauw, Thomas Gaslonde, Stéphane Léonce, Laurence Kraus-Berthier, William Laine, Gaëlle Lenglet, Angèle Chiaroni, Bruno Pfeiffer, Christian Bailly, Sylvie Michel, François Tillequin, Alain Pierré and Marie-Hélène David-Cordonnier
      Molecular Pharmacology December 2009, 76 (6) 1172-1185; DOI: https://doi.org/10.1124/mol.109.057554

U

  1. Ugur, Mehmet

    1. P2X7 Receptor Activates Multiple Selective Dye-Permeation Pathways in RAW 264.7 and Human Embryonic Kidney 293 Cells
      Serife Cankurtaran-Sayar, Kemal Sayar and Mehmet Ugur
      Molecular Pharmacology December 2009, 76 (6) 1323-1332; DOI: https://doi.org/10.1124/mol.109.059923

V

  1. Vandewalle, Alain

    1. Peroxisome Proliferator-Activated Receptor γ Antagonists Decrease Na+ Transport via the Epithelial Na+ Channel
      Tengis S. Pavlov, Vladislav Levchenko, Alexey V. Karpushev, Alain Vandewalle and Alexander Staruschenko
      Molecular Pharmacology December 2009, 76 (6) 1333-1340; DOI: https://doi.org/10.1124/mol.109.056911

  2. Varnes, Jeffrey G.

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  3. Vielhauer, George A.

    1. KU135, a Novel Novobiocin-Derived C-Terminal Inhibitor of the 90-kDa Heat Shock Protein, Exerts Potent Antiproliferative Effects in Human Leukemic Cells
      Shary N. Shelton, Mary E. Shawgo, Shawna B. Matthews, Yuanming Lu, Alison C. Donnelly, Kristen Szabla, Mehmet Tanol, George A. Vielhauer, Roger A. Rajewski, Robert L. Matts, Brian S. J. Blagg and John D. Robertson
      Molecular Pharmacology December 2009, 76 (6) 1314-1322; DOI: https://doi.org/10.1124/mol.109.058545

  4. von Hayn, Kathrin

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467

  5. von Lintig, Johannes

    1. Activation of Retinoic Acid Receptors by Dihydroretinoids
      Alexander R. Moise, Susana Alvarez, Marta Domínguez, Rosana Alvarez, Marcin Golczak, Glenn P. Lobo, Johannes von Lintig, Angel R. de Lera and Krzysztof Palczewski
      Molecular Pharmacology December 2009, 76 (6) 1228-1237; DOI: https://doi.org/10.1124/mol.109.060038

W

  1. Wacker, Dean A.

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  2. Wager-Miller, Jim

    1. Monoacylglycerol Lipase Limits the Duration of Endocannabinoid-Mediated Depolarization-Induced Suppression of Excitation in Autaptic Hippocampal Neurons
      Alex Straiker, Sherry Shu-Jung Hu, Jonathan Z. Long, Andy Arnold, Jim Wager-Miller, Benjamin F. Cravatt and Ken Mackie
      Molecular Pharmacology December 2009, 76 (6) 1220-1227; DOI: https://doi.org/10.1124/mol.109.059030

  3. Wang, Lu

    1. An Anticancer Effect of Curcumin Mediated by Down-Regulating Phosphatase of Regenerating Liver-3 Expression on Highly Metastatic Melanoma Cells
      Lu Wang, Yan Shen, Ran Song, Yang Sun, Jianliang Xu and Qiang Xu
      Molecular Pharmacology December 2009, 76 (6) 1238-1245; DOI: https://doi.org/10.1124/mol.109.059105

  4. Watson, Jeannette M.

    1. Effects of Positive Allosteric Modulators on Single-Cell Oscillatory Ca2+ Signaling Initiated by the Type 5 Metabotropic Glutamate Receptor
      Sophie J. Bradley, Jeannette M. Watson and R. A. John Challiss
      Molecular Pharmacology December 2009, 76 (6) 1302-1313; DOI: https://doi.org/10.1124/mol.109.059170

  5. Wu, Ginger Y.

    1. Position 5.46 of the Serotonin 5-HT2A Receptor Contributes to a Species-Dependent Variation for the 5-HT2C Agonist (R)-9-Ethyl-1,3,4,10b-tetrahydro-7-trifluoromethylpyrazino[2,1-a]isoindol-6(2H)-one: Impact on Selectivity and Toxicological Evaluation
      Keith J. Miller, Ginger Y. Wu, Jeffrey G. Varnes, Paul Levesque, Julia Li, Danshi Li, Jeffrey A. Robl, Karen A. Rossi and Dean A. Wacker
      Molecular Pharmacology December 2009, 76 (6) 1211-1219; DOI: https://doi.org/10.1124/mol.109.059204

  6. Wynick, David

    1. Receptor-Mediated Suppression of Potassium Currents Requires Colocalization within Lipid Rafts
      Susan Oldfield, Jane Hancock, Angharad Mason, Sally A. Hobson, David Wynick, Eamonn Kelly, Andrew D. Randall and Neil V. Marrion
      Molecular Pharmacology December 2009, 76 (6) 1279-1289; DOI: https://doi.org/10.1124/mol.109.058008

X

  1. Xu, Jianliang

    1. An Anticancer Effect of Curcumin Mediated by Down-Regulating Phosphatase of Regenerating Liver-3 Expression on Highly Metastatic Melanoma Cells
      Lu Wang, Yan Shen, Ran Song, Yang Sun, Jianliang Xu and Qiang Xu
      Molecular Pharmacology December 2009, 76 (6) 1238-1245; DOI: https://doi.org/10.1124/mol.109.059105

  2. Xu, Qiang

    1. An Anticancer Effect of Curcumin Mediated by Down-Regulating Phosphatase of Regenerating Liver-3 Expression on Highly Metastatic Melanoma Cells
      Lu Wang, Yan Shen, Ran Song, Yang Sun, Jianliang Xu and Qiang Xu
      Molecular Pharmacology December 2009, 76 (6) 1238-1245; DOI: https://doi.org/10.1124/mol.109.059105

Y

  1. Yan, Zhen

    1. Phosphatidylinositol (4,5)-Bisphosphate Regulation of N-Methyl-d-aspartate Receptor Channels in Cortical Neurons
      Madhuchhanda Mandal and Zhen Yan
      Molecular Pharmacology December 2009, 76 (6) 1349-1359; DOI: https://doi.org/10.1124/mol.109.058701

  2. Yoo, Justin

    1. Control of Glutamate Receptor 2 (GluR2) Translational Initiation by Its Alternative 3′ Untranslated Regions
      Hasan A. Irier, Yi Quan, Justin Yoo and Raymond Dingledine
      Molecular Pharmacology December 2009, 76 (6) 1145-1149; DOI: https://doi.org/10.1124/mol.109.060343

Z

  1. Zhang, Fang

    1. Identification of Survival Genes in Human Glioblastoma Cells by Small Interfering RNA Screening
      Nikhil G. Thaker, Fang Zhang, Peter R. McDonald, Tong Ying Shun, Michael D. Lewen, Ian F. Pollack and John S. Lazo
      Molecular Pharmacology December 2009, 76 (6) 1246-1255; DOI: https://doi.org/10.1124/mol.109.058024

  2. Zhou, Yixing

    1. Quantification of Gi-Mediated Inhibition of Adenylyl Cyclase Activity Reveals That UDP Is a Potent Agonist of the Human P2Y14 Receptor
      Rhonda L. Carter, Ingrid P. Fricks, Matthew O. Barrett, Lauren E. Burianek, Yixing Zhou, Hyojin Ko, Arijit Das, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden
      Molecular Pharmacology December 2009, 76 (6) 1341-1348; DOI: https://doi.org/10.1124/mol.109.058578

  3. Ziegler, Nicole

    1. β-Arrestin-2 Interaction and Internalization of the Human P2Y1 Receptor Are Dependent on C-Terminal Phosphorylation Sites
      Susanne Reiner, Nicole Ziegler, Catherine Leon, Kristina Lorenz, Kathrin von Hayn, Christian Gachet, Martin J. Lohse and Carsten Hoffmann
      Molecular Pharmacology December 2009, 76 (6) 1162-1171; DOI: https://doi.org/10.1124/mol.109.060467
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