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Index by author

October 01, 2010; Volume 78,Issue 4

A

  1. Abankwa, Daniel

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

  2. Abood, Mary E.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  3. Adler, Martin W.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  4. Adorini, Luciano

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  5. Aguilar, Marie-Isabel

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

  6. Al-Sabah, Suleiman

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  7. Albiston, Anthony L.

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  8. Altman, Jessica K.

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

B

  1. Bai, Yushi

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  2. Bailey, Chris P.

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  3. Baptist, Myma

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  4. Barak, Larry S.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  5. Bee, Thomas

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  6. Beedanagari, Sudheer R.

    1. Role of Epigenetic Mechanisms in Differential Regulation of the Dioxin-Inducible Human CYP1A1 and CYP1B1 Genes
      Sudheer R. Beedanagari, Robert T. Taylor, Peter Bui, Feng Wang, Derek W. Nickerson and Oliver Hankinson
      Molecular Pharmacology October 2010, 78 (4) 608-616; DOI: https://doi.org/10.1124/mol.110.064899

  7. Bodendiek, Silke B.

    1. Potassium Channel Block by a Tripartite Complex of Two Cationophilic Ligands and a Potassium Ion
      Pavel I. Zimin, Bojan Garic, Silke B. Bodendiek, Cédrick Mahieux, Heike Wulff and Boris S. Zhorov
      Molecular Pharmacology October 2010, 78 (4) 588-599; DOI: https://doi.org/10.1124/mol.110.064014

  8. Brazier, Michel

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  9. Brown, Edward Meigs

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  10. Bui, Peter

    1. Role of Epigenetic Mechanisms in Differential Regulation of the Dioxin-Inducible Human CYP1A1 and CYP1B1 Genes
      Sudheer R. Beedanagari, Robert T. Taylor, Peter Bui, Feng Wang, Derek W. Nickerson and Oliver Hankinson
      Molecular Pharmacology October 2010, 78 (4) 608-616; DOI: https://doi.org/10.1124/mol.110.064899

C

  1. Caron, Marc G.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  2. Caudrillier, Axelle

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  3. Chai, Siew Yeen

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  4. Chan, Eric Chun Yong

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  5. Chang, Min-Hwang

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  6. Charlton, Steven J.

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  7. Chen, Wei

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  8. Cherian, Christina

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  9. Chung, Sung-Kee

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  10. Chung, Thomas D.Y.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  11. Ciaccioli, Gianmario

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  12. Cortés, Lorena

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  13. Cournarie, Fabienne

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  14. Cowan, Alan

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  15. Crouthamel, Marykate

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

D

  1. de Diego, Antonio M. G.

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  2. De Franco, Francesca

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  3. Desmoulin, Sita Kugel

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  4. Dewey, William L.

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  5. Díez-Dacal, Beatriz

    1. Cyclopentenone Prostaglandins with Dienone Structure Promote Cross-Linking of the Chemoresistance-Inducing Enzyme Glutathione Transferase P1-1
      Francisco J. Sánchez-Gómez, Beatriz Díez-Dacal, María A. Pajares, Oscar Llorca and Dolores Pérez-Sala
      Molecular Pharmacology October 2010, 78 (4) 723-733; DOI: https://doi.org/10.1124/mol.110.065391

  6. DiLizio, Cherisse

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

  7. Dinh, Diem T.

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

  8. Don, Anthony S.

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  9. Donadio, Loredana

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  10. Du, Ann T.

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

E

  1. Ehlert, Frederick J.

    1. Mutagenesis of Nucleophilic Residues near the Orthosteric Binding Pocket of M1 and M2 Muscarinic receptors: Effect on the Binding of Nitrogen Mustard Analogs of Acetylcholine and McN-A-343
      Hinako Suga, Gregory W. Sawyer and Frederick J. Ehlert
      Molecular Pharmacology October 2010, 78 (4) 745-755; DOI: https://doi.org/10.1124/mol.110.065367

  2. English, Dallas R.

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

F

  1. Faure, Helene

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  2. Ferguson, Stephen S.

    1. Synergistically Enhanced CYP2B6 Inducibility between a Polymorphic Mutation in CYP2B6 Promoter and Pregnane X Receptor Activation
      Haishan Li, Stephen S. Ferguson and Hongbing Wang
      Molecular Pharmacology October 2010, 78 (4) 704-713; DOI: https://doi.org/10.1124/mol.110.065185

  3. Fernández-Morales, José Carlos

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  4. Fozzard, Harry A.

    1. Molecular Model of Anticonvulsant Drug Binding to the Voltage-Gated Sodium Channel Inner Pore
      Gregory M. Lipkind and Harry A. Fozzard
      Molecular Pharmacology October 2010, 78 (4) 631-638; DOI: https://doi.org/10.1124/mol.110.064683

  5. Fukunaga, Rikiro

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

  6. Fulterer, Andreas

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  7. Furukawa, Hiro

    1. Control of Assembly and Function of Glutamate Receptors by the Amino-Terminal Domain
      Kasper B. Hansen, Hiro Furukawa and Stephen F. Traynelis
      Molecular Pharmacology October 2010, 78 (4) 535-549; DOI: https://doi.org/10.1124/mol.110.067157

G

  1. Gangjee, Aleem

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  2. García, Antonio G.

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  3. Gardner-Stephen, Dione

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  4. Garic, Bojan

    1. Potassium Channel Block by a Tripartite Complex of Two Cationophilic Ligands and a Potassium Ion
      Pavel I. Zimin, Bojan Garic, Silke B. Bodendiek, Cédrick Mahieux, Heike Wulff and Boris S. Zhorov
      Molecular Pharmacology October 2010, 78 (4) 588-599; DOI: https://doi.org/10.1124/mol.110.064014

  5. Geller, Ellen B.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  6. Giles, Graham G.

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  7. Gkountelias, Kostas

    1. Exploring the Binding Site Crevice of a Family B G Protein-Coupled Receptor, the Type 1 Corticotropin Releasing Factor Receptor
      Kostas Gkountelias, Maria Papadokostaki, Jonathan A. Javitch and George Liapakis
      Molecular Pharmacology October 2010, 78 (4) 785-793; DOI: https://doi.org/10.1124/mol.110.065474

  8. Glaser, Heather

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

  9. Godin, Corinne

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  10. González, José Carlos

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  11. Gorojankina, Tatiana

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  12. Gregory, Philip A.

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

H

  1. Hancock, John F.

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

  2. Hankinson, Oliver

    1. Role of Epigenetic Mechanisms in Differential Regulation of the Dioxin-Inducible Human CYP1A1 and CYP1B1 Genes
      Sudheer R. Beedanagari, Robert T. Taylor, Peter Bui, Feng Wang, Derek W. Nickerson and Oliver Hankinson
      Molecular Pharmacology October 2010, 78 (4) 608-616; DOI: https://doi.org/10.1124/mol.110.064899

  3. Hansen, Kasper B.

    1. Control of Assembly and Function of Glutamate Receptors by the Amino-Terminal Domain
      Kasper B. Hansen, Hiro Furukawa and Stephen F. Traynelis
      Molecular Pharmacology October 2010, 78 (4) 535-549; DOI: https://doi.org/10.1124/mol.110.067157

  4. Henderson, Graeme

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  5. Hernández-Guijo, Jesús Miguel

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  6. Heynen-Genel, Susanne

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  7. Ho, Han Kiat

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  8. Holien, Jessica K.

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  9. Hopper, John L.

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  10. Hou, Zhanjun

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  11. Hu, Dong Gui

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  12. Hurtel-Lemaire, Anne-Sophie

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

J

  1. Jacobson, Marlene A.

    1. The M1 Muscarinic Receptor Allosteric Agonists AC-42 and 1-[1′-(2-Methylbenzyl)-1,4′-bipiperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one Bind to a Unique Site Distinct from the Acetylcholine Orthosteric Site
      Marlene A. Jacobson, Constantine Kreatsoulas, Danette M. Pascarella, Julie A. O'Brien and Cyrille Sur
      Molecular Pharmacology October 2010, 78 (4) 648-657; DOI: https://doi.org/10.1124/mol.110.065771

  2. Jary, Eve

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  3. Javitch, Jonathan A.

    1. Exploring the Binding Site Crevice of a Family B G Protein-Coupled Receptor, the Type 1 Corticotropin Releasing Factor Receptor
      Kostas Gkountelias, Maria Papadokostaki, Jonathan A. Javitch and George Liapakis
      Molecular Pharmacology October 2010, 78 (4) 785-793; DOI: https://doi.org/10.1124/mol.110.065474

  4. Jiang, Tao

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  5. Joshi, Sonali

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

K

  1. Kalinowski, Danuta S.

    1. Membrane Transport and Intracellular Sequestration of Novel Thiosemicarbazone Chelators for the Treatment of Cancer
      Angelica M. Merlot, Namfon Pantarat, David B. Lovejoy, Danuta S. Kalinowski and Des R. Richardson
      Molecular Pharmacology October 2010, 78 (4) 675-684; DOI: https://doi.org/10.1124/mol.110.066126

  2. Kamel, Said

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  3. Kapur, Ankur

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  4. Kelly, Eamonn

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  5. Khadem, Shaheen

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

  6. Krasel, Cornelius

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  7. Kreatsoulas, Constantine

    1. The M1 Muscarinic Receptor Allosteric Agonists AC-42 and 1-[1′-(2-Methylbenzyl)-1,4′-bipiperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one Bind to a Unique Site Distinct from the Acetylcholine Orthosteric Site
      Marlene A. Jacobson, Constantine Kreatsoulas, Danette M. Pascarella, Julie A. O'Brien and Cyrille Sur
      Molecular Pharmacology October 2010, 78 (4) 648-657; DOI: https://doi.org/10.1124/mol.110.065771

  8. Kuruba, Ramalinga

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

L

  1. Levi, Moshe

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  2. Lew, Michael J.

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

  3. Lew, Rebecca A.

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  4. Li, Haishan

    1. Synergistically Enhanced CYP2B6 Inducibility between a Polymorphic Mutation in CYP2B6 Promoter and Pregnane X Receptor Activation
      Haishan Li, Stephen S. Ferguson and Hongbing Wang
      Molecular Pharmacology October 2010, 78 (4) 704-713; DOI: https://doi.org/10.1124/mol.110.065185

  5. Li, Song

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

  6. Liapakis, George

    1. Exploring the Binding Site Crevice of a Family B G Protein-Coupled Receptor, the Type 1 Corticotropin Releasing Factor Receptor
      Kostas Gkountelias, Maria Papadokostaki, Jonathan A. Javitch and George Liapakis
      Molecular Pharmacology October 2010, 78 (4) 785-793; DOI: https://doi.org/10.1124/mol.110.065474

  7. Lipkind, Gregory M.

    1. Molecular Model of Anticonvulsant Drug Binding to the Voltage-Gated Sodium Channel Inner Pore
      Gregory M. Lipkind and Harry A. Fozzard
      Molecular Pharmacology October 2010, 78 (4) 631-638; DOI: https://doi.org/10.1124/mol.110.064683

  8. Llorca, Oscar

    1. Cyclopentenone Prostaglandins with Dienone Structure Promote Cross-Linking of the Chemoresistance-Inducing Enzyme Glutathione Transferase P1-1
      Francisco J. Sánchez-Gómez, Beatriz Díez-Dacal, María A. Pajares, Oscar Llorca and Dolores Pérez-Sala
      Molecular Pharmacology October 2010, 78 (4) 723-733; DOI: https://doi.org/10.1124/mol.110.065391

  9. Llorente, Javier

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  10. Lovejoy, David B.

    1. Membrane Transport and Intracellular Sequestration of Novel Thiosemicarbazone Chelators for the Treatment of Cancer
      Angelica M. Merlot, Namfon Pantarat, David B. Lovejoy, Danuta S. Kalinowski and Des R. Richardson
      Molecular Pharmacology October 2010, 78 (4) 675-684; DOI: https://doi.org/10.1124/mol.110.066126

M

  1. Mackenzie, Peter I.

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  2. Mahieux, Cédrick

    1. Potassium Channel Block by a Tripartite Complex of Two Cationophilic Ligands and a Potassium Ion
      Pavel I. Zimin, Bojan Garic, Silke B. Bodendiek, Cédrick Mahieux, Heike Wulff and Boris S. Zhorov
      Molecular Pharmacology October 2010, 78 (4) 588-599; DOI: https://doi.org/10.1124/mol.110.064014

  3. Manetti, Fabrizio

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  4. Mann, Andre

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  5. Manning, David R.

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

  6. Matherly, Larry H.

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  7. McPherson, Jamie

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  8. Mentaverri, Romuald

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  9. Merlot, Angelica M.

    1. Membrane Transport and Intracellular Sequestration of Novel Thiosemicarbazone Chelators for the Treatment of Cancer
      Angelica M. Merlot, Namfon Pantarat, David B. Lovejoy, Danuta S. Kalinowski and Des R. Richardson
      Molecular Pharmacology October 2010, 78 (4) 675-684; DOI: https://doi.org/10.1124/mol.110.066126

  10. Morris, Jonathan C.

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  11. Morton, Craig J.

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

N

  1. Nelson, Sidney D.

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  2. Neubig, Richard R.

    1. Thinking Outside of the “RGS Box”: New Approaches to Therapeutic Targeting of Regulators of G Protein Signaling
      Benita Sjögren and Richard R. Neubig
      Molecular Pharmacology October 2010, 78 (4) 550-557; DOI: https://doi.org/10.1124/mol.110.065219
    2. Mind Your Salts: When the Inactive Constituent Isn't
      Richard R. Neubig
      Molecular Pharmacology October 2010, 78 (4) 558-559; DOI: https://doi.org/10.1124/mol.110.067645

  3. New, Lee Sun

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  4. Ng, Leelee

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  5. Nickerson, Derek W.

    1. Role of Epigenetic Mechanisms in Differential Regulation of the Dioxin-Inducible Human CYP1A1 and CYP1B1 Genes
      Sudheer R. Beedanagari, Robert T. Taylor, Peter Bui, Feng Wang, Derek W. Nickerson and Oliver Hankinson
      Molecular Pharmacology October 2010, 78 (4) 608-616; DOI: https://doi.org/10.1124/mol.110.064899

O

  1. O'Brien, Julie A.

    1. The M1 Muscarinic Receptor Allosteric Agonists AC-42 and 1-[1′-(2-Methylbenzyl)-1,4′-bipiperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one Bind to a Unique Site Distinct from the Acetylcholine Orthosteric Site
      Marlene A. Jacobson, Constantine Kreatsoulas, Danette M. Pascarella, Julie A. O'Brien and Cyrille Sur
      Molecular Pharmacology October 2010, 78 (4) 648-657; DOI: https://doi.org/10.1124/mol.110.065771

  2. Oh, Jing Wen

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  3. Onan, Döne

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

  4. Orallo, Francisco

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  5. Orlandi, Stefano

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

P

  1. Pajares, María A.

    1. Cyclopentenone Prostaglandins with Dienone Structure Promote Cross-Linking of the Chemoresistance-Inducing Enzyme Glutathione Transferase P1-1
      Francisco J. Sánchez-Gómez, Beatriz Díez-Dacal, María A. Pajares, Oscar Llorca and Dolores Pérez-Sala
      Molecular Pharmacology October 2010, 78 (4) 723-733; DOI: https://doi.org/10.1124/mol.110.065391

  2. Pantarat, Namfon

    1. Membrane Transport and Intracellular Sequestration of Novel Thiosemicarbazone Chelators for the Treatment of Cancer
      Angelica M. Merlot, Namfon Pantarat, David B. Lovejoy, Danuta S. Kalinowski and Des R. Richardson
      Molecular Pharmacology October 2010, 78 (4) 675-684; DOI: https://doi.org/10.1124/mol.110.066126

  3. Papadokostaki, Maria

    1. Exploring the Binding Site Crevice of a Family B G Protein-Coupled Receptor, the Type 1 Corticotropin Releasing Factor Receptor
      Kostas Gkountelias, Maria Papadokostaki, Jonathan A. Javitch and George Liapakis
      Molecular Pharmacology October 2010, 78 (4) 785-793; DOI: https://doi.org/10.1124/mol.110.065474

  4. Parker, Michael W.

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  5. Pascarella, Danette M.

    1. The M1 Muscarinic Receptor Allosteric Agonists AC-42 and 1-[1′-(2-Methylbenzyl)-1,4′-bipiperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one Bind to a Unique Site Distinct from the Acetylcholine Orthosteric Site
      Marlene A. Jacobson, Constantine Kreatsoulas, Danette M. Pascarella, Julie A. O'Brien and Cyrille Sur
      Molecular Pharmacology October 2010, 78 (4) 648-657; DOI: https://doi.org/10.1124/mol.110.065771

  6. Passeri, Daniela

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  7. Pattenden, Leonard K.

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

  8. Pérez-Sala, Dolores

    1. Cyclopentenone Prostaglandins with Dienone Structure Promote Cross-Linking of the Chemoresistance-Inducing Enzyme Glutathione Transferase P1-1
      Francisco J. Sánchez-Gómez, Beatriz Díez-Dacal, María A. Pajares, Oscar Llorca and Dolores Pérez-Sala
      Molecular Pharmacology October 2010, 78 (4) 723-733; DOI: https://doi.org/10.1124/mol.110.065391

  9. Petit, Jean-Pierre

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  10. Petit, Laurent

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  11. Pham, Vi

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  12. Platanias, Leonidas C.

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

  13. Pruzanski, Mark

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

R

  1. Reggio, Patricia H.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  2. Ren, Songrong

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

  3. Richardson, Des R.

    1. Membrane Transport and Intracellular Sequestration of Novel Thiosemicarbazone Chelators for the Treatment of Cancer
      Angelica M. Merlot, Namfon Pantarat, David B. Lovejoy, Danuta S. Kalinowski and Des R. Richardson
      Molecular Pharmacology October 2010, 78 (4) 675-684; DOI: https://doi.org/10.1124/mol.110.066126

  4. Rivero, Guadalupe

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  5. Rizzo, Giorgia

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  6. Rizzo, Giovanni

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  7. Romero, Michael F.

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  8. Rosethorne, Elizabeth M.

    1. μ-Opioid Receptors: Correlation of Agonist Efficacy for Signalling with Ability to Activate Internalization
      Jamie McPherson, Guadalupe Rivero, Myma Baptist, Javier Llorente, Suleiman Al-Sabah, Cornelius Krasel, William L. Dewey, Chris P. Bailey, Elizabeth M. Rosethorne, Steven J. Charlton, Graeme Henderson and Eamonn Kelly
      Molecular Pharmacology October 2010, 78 (4) 756-766; DOI: https://doi.org/10.1124/mol.110.066613

  9. Roudaut, Hermine

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  10. Ruat, Martial

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

S

  1. Sadeghpour, Bahman

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  2. Sánchez-Gómez, Francisco J.

    1. Cyclopentenone Prostaglandins with Dienone Structure Promote Cross-Linking of the Chemoresistance-Inducing Enzyme Glutathione Transferase P1-1
      Francisco J. Sánchez-Gómez, Beatriz Díez-Dacal, María A. Pajares, Oscar Llorca and Dolores Pérez-Sala
      Molecular Pharmacology October 2010, 78 (4) 723-733; DOI: https://doi.org/10.1124/mol.110.065391

  3. Sassano, Antonella

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

  4. Sauer, Michelle

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  5. Sawyer, Gregory W.

    1. Mutagenesis of Nucleophilic Residues near the Orthosteric Binding Pocket of M1 and M2 Muscarinic receptors: Effect on the Binding of Nitrogen Mustard Analogs of Acetylcholine and McN-A-343
      Hinako Suga, Gregory W. Sawyer and Frederick J. Ehlert
      Molecular Pharmacology October 2010, 78 (4) 745-755; DOI: https://doi.org/10.1124/mol.110.065367

  6. Schoenfelder, Angele

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  7. Seltzman, Herbert H.

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  8. Seo, Kyung-Chang

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  9. Severi, Gianluca

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  10. Sharir, Haleli

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  11. Sjögren, Benita

    1. Thinking Outside of the “RGS Box”: New Approaches to Therapeutic Targeting of Regulators of G Protein Signaling
      Benita Sjögren and Richard R. Neubig
      Molecular Pharmacology October 2010, 78 (4) 550-557; DOI: https://doi.org/10.1124/mol.110.065219

  12. Solinas, Antonio

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  13. Stout, Mark

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  14. Suga, Hinako

    1. Mutagenesis of Nucleophilic Residues near the Orthosteric Binding Pocket of M1 and M2 Muscarinic receptors: Effect on the Binding of Nitrogen Mustard Analogs of Acetylcholine and McN-A-343
      Hinako Suga, Gregory W. Sawyer and Frederick J. Ehlert
      Molecular Pharmacology October 2010, 78 (4) 745-755; DOI: https://doi.org/10.1124/mol.110.065367

  15. Sur, Cyrille

    1. The M1 Muscarinic Receptor Allosteric Agonists AC-42 and 1-[1′-(2-Methylbenzyl)-1,4′-bipiperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one Bind to a Unique Site Distinct from the Acetylcholine Orthosteric Site
      Marlene A. Jacobson, Constantine Kreatsoulas, Danette M. Pascarella, Julie A. O'Brien and Cyrille Sur
      Molecular Pharmacology October 2010, 78 (4) 648-657; DOI: https://doi.org/10.1124/mol.110.065771

T

  1. Taddei, Maurizio

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  2. Tallman, Martin S.

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

  3. Taylor, Robert T.

    1. Role of Epigenetic Mechanisms in Differential Regulation of the Dioxin-Inducible Human CYP1A1 and CYP1B1 Genes
      Sudheer R. Beedanagari, Robert T. Taylor, Peter Bui, Feng Wang, Derek W. Nickerson and Oliver Hankinson
      Molecular Pharmacology October 2010, 78 (4) 608-616; DOI: https://doi.org/10.1124/mol.110.064899

  4. Teng, Woon Chien

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  5. Terwilliger, Ernest

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  6. Thomas, Walter G.

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151

  7. Thompson, Philip E.

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

  8. Tilley, Wayne D.

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

  9. Traiffort, Elisabeth

    1. Virtual Screening-Based Discovery and Mechanistic Characterization of the Acylthiourea MRT-10 Family as Smoothened Antagonists
      Fabrizio Manetti, Helene Faure, Hermine Roudaut, Tatiana Gorojankina, Elisabeth Traiffort, Angele Schoenfelder, Andre Mann, Antonio Solinas, Maurizio Taddei and Martial Ruat
      Molecular Pharmacology October 2010, 78 (4) 658-665; DOI: https://doi.org/10.1124/mol.110.065102

  10. Traynelis, Stephen F.

    1. Control of Assembly and Function of Glutamate Receptors by the Amino-Terminal Domain
      Kasper B. Hansen, Hiro Furukawa and Stephen F. Traynelis
      Molecular Pharmacology October 2010, 78 (4) 535-549; DOI: https://doi.org/10.1124/mol.110.067157

  11. Treloar, Joanna

    1. A Novel Polymorphism in a Forkhead Box A1 (FOXA1) Binding Site of the Human UDP Glucuronosyltransferase 2B17 Gene Modulates Promoter Activity and Is Associated with Altered Levels of Circulating Androstane-3α,17β-diol Glucuronide
      Dong Gui Hu, Dione Gardner-Stephen, Gianluca Severi, Philip A. Gregory, Joanna Treloar, Graham G. Giles, Dallas R. English, John L. Hopper, Wayne D. Tilley and Peter I. Mackenzie
      Molecular Pharmacology October 2010, 78 (4) 714-722; DOI: https://doi.org/10.1124/mol.110.065953

U

  1. Ueda, Takeshi

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

W

  1. Wada, Tara

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

  2. Wahlin, Michelle D.

    1. Mechanism-Based Inactivation of Cytochrome P450 3A4 by Lapatinib
      Woon Chien Teng, Jing Wen Oh, Lee Sun New, Michelle D. Wahlin, Sidney D. Nelson, Han Kiat Ho and Eric Chun Yong Chan
      Molecular Pharmacology October 2010, 78 (4) 693-703; DOI: https://doi.org/10.1124/mol.110.065839

  3. Walker, Scott R.

    1. Elimination of a Hydroxyl Group in FTY720 Dramatically Improves the Phosphorylation Rate
      Eve Jary, Thomas Bee, Scott R. Walker, Sung-Kee Chung, Kyung-Chang Seo, Jonathan C. Morris and Anthony S. Don
      Molecular Pharmacology October 2010, 78 (4) 685-692; DOI: https://doi.org/10.1124/mol.110.064873

  4. Wang, Feng

    1. Role of Epigenetic Mechanisms in Differential Regulation of the Dioxin-Inducible Human CYP1A1 and CYP1B1 Genes
      Sudheer R. Beedanagari, Robert T. Taylor, Peter Bui, Feng Wang, Derek W. Nickerson and Oliver Hankinson
      Molecular Pharmacology October 2010, 78 (4) 608-616; DOI: https://doi.org/10.1124/mol.110.064899

  5. Wang, Hongbing

    1. Synergistically Enhanced CYP2B6 Inducibility between a Polymorphic Mutation in CYP2B6 Promoter and Pregnane X Receptor Activation
      Haishan Li, Stephen S. Ferguson and Hongbing Wang
      Molecular Pharmacology October 2010, 78 (4) 704-713; DOI: https://doi.org/10.1124/mol.110.065185

  6. Wang, Xiaoxin X.

    1. Functional Characterization of the Semisynthetic Bile Acid Derivative INT-767, a Dual Farnesoid X Receptor and TGR5 Agonist
      Giovanni Rizzo, Daniela Passeri, Francesca De Franco, Gianmario Ciaccioli, Loredana Donadio, Giorgia Rizzo, Stefano Orlandi, Bahman Sadeghpour, Xiaoxin X. Wang, Tao Jiang, Moshe Levi, Mark Pruzanski and Luciano Adorini
      Molecular Pharmacology October 2010, 78 (4) 617-630; DOI: https://doi.org/10.1124/mol.110.064501

  7. Wang, Yiqiang

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  8. Watanabe-Fukunaga, Rie

    1. Negative Regulatory Effects of Mnk Kinases in the Generation of Chemotherapy-Induced Antileukemic Responses
      Jessica K. Altman, Heather Glaser, Antonella Sassano, Sonali Joshi, Takeshi Ueda, Rie Watanabe-Fukunaga, Rikiro Fukunaga, Martin S. Tallman and Leonidas C. Platanias
      Molecular Pharmacology October 2010, 78 (4) 778-784; DOI: https://doi.org/10.1124/mol.110.064642

  9. Wattel, Alice

    1. Strontium Ranelate Decreases Receptor Activator of Nuclear Factor-κB Ligand-Induced Osteoclastic Differentiation In Vitro: Involvement of the Calcium-Sensing Receptor
      Axelle Caudrillier, Anne-Sophie Hurtel-Lemaire, Alice Wattel, Fabienne Cournarie, Corinne Godin, Laurent Petit, Jean-Pierre Petit, Ernest Terwilliger, Said Kamel, Edward Meigs Brown, Romuald Mentaverri and Michel Brazier
      Molecular Pharmacology October 2010, 78 (4) 569-576; DOI: https://doi.org/10.1124/mol.109.063347

  10. Wedegaertner, Philip B.

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

  11. Wu, Jianmei

    1. Targeting the Proton-Coupled Folate Transporter for Selective Delivery of 6-Substituted Pyrrolo[2,3-d]Pyrimidine Antifolate Inhibitors of De Novo Purine Biosynthesis in the Chemotherapy of Solid Tumors
      Sita Kugel Desmoulin, Yiqiang Wang, Jianmei Wu, Mark Stout, Zhanjun Hou, Andreas Fulterer, Min-Hwang Chang, Michael F. Romero, Christina Cherian, Aleem Gangjee and Larry H. Matherly
      Molecular Pharmacology October 2010, 78 (4) 577-587; DOI: https://doi.org/10.1124/mol.110.065896

  12. Wulff, Heike

    1. Potassium Channel Block by a Tripartite Complex of Two Cationophilic Ligands and a Potassium Ion
      Pavel I. Zimin, Bojan Garic, Silke B. Bodendiek, Cédrick Mahieux, Heike Wulff and Boris S. Zhorov
      Molecular Pharmacology October 2010, 78 (4) 588-599; DOI: https://doi.org/10.1124/mol.110.064014

X

  1. Xie, Wen

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

Y

  1. Yáñez, Matilde

    1. Blockade by Nanomolar Resveratrol of Quantal Catecholamine Release in Chromaffin Cells
      José Carlos Fernández-Morales, Matilde Yáñez, Francisco Orallo, Lorena Cortés, José Carlos González, Jesús Miguel Hernández-Guijo, Antonio G. García and Antonio M. G. de Diego
      Molecular Pharmacology October 2010, 78 (4) 734-744; DOI: https://doi.org/10.1124/mol.110.066423

  2. Ye, Siying

    1. Phenylalanine-544 Plays a Key Role in Substrate and Inhibitor Binding by Providing a Hydrophobic Packing Point at the Active Site of Insulin-Regulated Aminopeptidase
      Anthony L. Albiston, Vi Pham, Siying Ye, Leelee Ng, Rebecca A. Lew, Philip E. Thompson, Jessica K. Holien, Craig J. Morton, Michael W. Parker and Siew Yeen Chai
      Molecular Pharmacology October 2010, 78 (4) 600-607; DOI: https://doi.org/10.1124/mol.110.065458

Z

  1. Zhai, Yonggong

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

  2. Zhang, Bin

    1. A Functional Cross-Talk between Liver X Receptor-α and Constitutive Androstane Receptor Links Lipogenesis and Xenobiotic Responses
      Yonggong Zhai, Tara Wada, Bin Zhang, Shaheen Khadem, Songrong Ren, Ramalinga Kuruba, Song Li and Wen Xie
      Molecular Pharmacology October 2010, 78 (4) 666-674; DOI: https://doi.org/10.1124/mol.110.064618

  3. Zhang, Li

    1. An N-Terminal Polybasic Motif of Gαq Is Required for Signaling and Influences Membrane Nanodomain Distribution
      Marykate Crouthamel, Daniel Abankwa, Li Zhang, Cherisse DiLizio, David R. Manning, John F. Hancock and Philip B. Wedegaertner
      Molecular Pharmacology October 2010, 78 (4) 767-777; DOI: https://doi.org/10.1124/mol.110.066340

  4. Zhao, Pingwei

    1. Targeting of the Orphan Receptor GPR35 by Pamoic Acid: A Potent Activator of Extracellular Signal-Regulated Kinase and β-Arrestin2 with Antinociceptive Activity
      Pingwei Zhao, Haleli Sharir, Ankur Kapur, Alan Cowan, Ellen B. Geller, Martin W. Adler, Herbert H. Seltzman, Patricia H. Reggio, Susanne Heynen-Genel, Michelle Sauer, Thomas D.Y. Chung, Yushi Bai, Wei Chen, Marc G. Caron, Larry S. Barak and Mary E. Abood
      Molecular Pharmacology October 2010, 78 (4) 560-568; DOI: https://doi.org/10.1124/mol.110.066746

  5. Zhorov, Boris S.

    1. Potassium Channel Block by a Tripartite Complex of Two Cationophilic Ligands and a Potassium Ion
      Pavel I. Zimin, Bojan Garic, Silke B. Bodendiek, Cédrick Mahieux, Heike Wulff and Boris S. Zhorov
      Molecular Pharmacology October 2010, 78 (4) 588-599; DOI: https://doi.org/10.1124/mol.110.064014

  6. Zimin, Pavel I.

    1. Potassium Channel Block by a Tripartite Complex of Two Cationophilic Ligands and a Potassium Ion
      Pavel I. Zimin, Bojan Garic, Silke B. Bodendiek, Cédrick Mahieux, Heike Wulff and Boris S. Zhorov
      Molecular Pharmacology October 2010, 78 (4) 588-599; DOI: https://doi.org/10.1124/mol.110.064014

  7. Ziogas, James

    1. Ligand-Supported Purification of the Urotensin-II Receptor
      Ann T. Du, Döne Onan, Diem T. Dinh, Michael J. Lew, James Ziogas, Marie-Isabel Aguilar, Leonard K. Pattenden and Walter G. Thomas
      Molecular Pharmacology October 2010, 78 (4) 639-647; DOI: https://doi.org/10.1124/mol.110.065151
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