Table of Contents

Articles

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  Different N-Terminal Motifs Determine Plasma Membrane Targeting of the Human Concentrative Nucleoside Transporter 3 in Polarized and Nonpolarized Cells

  Ekaitz Errasti-Murugarren, F. Javier Casado and Marçal Pastor-Anglada

  Molecular Pharmacology November 2010, 78 (5) 795-803; DOI: https://doi.org/10.1124/mol.110.065920
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  Structure-Activity Relationships of GPR120 Agonists Based on a Docking Simulation

  Qi Sun, Akira Hirasawa, Takafumi Hara, Ikuo Kimura, Tetsuya Adachi, Takeo Awaji, Masaji Ishiguro, Takayoshi Suzuki, Naoki Miyata and Gozoh Tsujimoto

  Molecular Pharmacology November 2010, 78 (5) 804-810; DOI: https://doi.org/10.1124/mol.110.066324
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  Lyn Kinase-Dependent Regulation of miR181 and Myeloid Cell Leukemia-1 Expression: Implications for Drug Resistance in Myelogenous Leukemia

  Eric I. Zimmerman, Claudia M. Dollins, Melissa Crawford, Steven Grant, Serge P. Nana-Sinkam, Kristy L. Richards, Scott M. Hammond and Lee M. Graves

  Molecular Pharmacology November 2010, 78 (5) 811-817; DOI: https://doi.org/10.1124/mol.110.066258
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  Constitutive Activity of Serotonin_2C Receptors at G Protein-Independent Signaling: Modulation by RNA Editing and Antidepressants

  Marilyne Labasque, Julie Meffre, Gaelle Carrat, Carine Becamel, Joël Bockaert and Philippe Marin

  Molecular Pharmacology November 2010, 78 (5) 818-826; DOI: https://doi.org/10.1124/mol.110.066035
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  Auraptene Is an Inhibitor of Cholesterol Esterification and a Modulator of Estrogen Receptors

  Philippe de Medina, Salvatore Genovese, Michael R. Paillasse, Mahta Mazaheri, Stephanie Caze-Subra, Kerstin Bystricky, Massimo Curini, Sandrine Silvente-Poirot, Francesco Epifano and Marc Poirot

  Molecular Pharmacology November 2010, 78 (5) 827-836; DOI: https://doi.org/10.1124/mol.110.065250
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  The μ-Opioid Receptor Variant N190K Is Unresponsive to Peptide Agonists yet Can be Rescued by Small-Molecule Drugs

  Jean-Philippe Fortin, Lei Ci, Jonathan Schroeder, Carmit Goldstein, Maria Claudia Montefusco, Inga Peter, Steven E. Reis, Gordon S. Huggins, Martin Beinborn and Alan S. Kopin

  Molecular Pharmacology November 2010, 78 (5) 837-845; DOI: https://doi.org/10.1124/mol.110.064188
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  Pharmacological Targeting of Constitutively Active Truncated Androgen Receptor by Nigericin and Suppression of Hormone-Refractory Prostate Cancer Cell Growth

  Tetsuo Mashima, Sachiko Okabe and Hiroyuki Seimiya

  Molecular Pharmacology November 2010, 78 (5) 846-854; DOI: https://doi.org/10.1124/mol.110.064790
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  Amurensin G, a Potent Natural SIRT1 Inhibitor, Rescues Doxorubicin Responsiveness via Down-Regulation of Multidrug Resistance 1

  Won Keun Oh, Kyoung Bin Cho, Tran Thi Hien, Tae Hyung Kim, Hyung Sik Kim, Trong Tuan Dao, Hyo-Kyung Han, Seong-Min Kwon, Sang-Gun Ahn, Jung-Hoon Yoon, Tae Hyun Kim, Yoon Gyoon Kim and Keon Wook Kang

  Molecular Pharmacology November 2010, 78 (5) 855-864; DOI: https://doi.org/10.1124/mol.110.065961
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  Thapsigargin Induces Expression of Activating Transcription Factor 3 in Human Keratinocytes Involving Ca²⁺ Ions and c-Jun N-Terminal Protein Kinase

  Daniel Spohn, Oliver G. Rössler, Stephan E. Philipp, Michael Raubuch, Shigetaka Kitajima, Désirée Griesemer, Markus Hoth and Gerald Thiel

  Molecular Pharmacology November 2010, 78 (5) 865-876; DOI: https://doi.org/10.1124/mol.110.067637
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  A Nonthiazolidinedione Peroxisome Proliferator-Activated Receptor α/γ Dual Agonist CG301360 Alleviates Insulin Resistance and Lipid Dysregulation in db/db Mice

  Hyun Woo Jeong, Joo-Won Lee, Woo Sik Kim, Sung Sik Choe, Hyun Jung Shin, Gha Young Lee, Dongkyu Shin, Jun Hee Lee, Eun Bok Choi, Hyun Kyu Lee, Gyu Hwan Yon, Bongjun Cho, Hye Ryung Kim, Sung Hee Choi, Young Sun Chung, Seung Bum Park, Heekyoung Chung, Seonggu Ro and Jae Bum Kim

  Molecular Pharmacology November 2010, 78 (5) 877-885; DOI: https://doi.org/10.1124/mol.110.065748
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  Regulation of CYP2C19 Expression by Estrogen Receptor α: Implications for Estrogen-Dependent Inhibition of Drug Metabolism

  Jessica Mwinyi, Isa Cavaco, Rasmus Steen Pedersen, Anna Persson, Sabrina Burkhardt, Souren Mkrtchian and Magnus Ingelman-Sundberg

  Molecular Pharmacology November 2010, 78 (5) 886-894; DOI: https://doi.org/10.1124/mol.110.065540
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  Monepantel Allosterically Activates DEG-3/DES-2 Channels of the Gastrointestinal Nematode Haemonchus contortus

  Lucien Rufener, Roland Baur, Ronald Kaminsky, Pascal Mäser and Erwin Sigel

  Molecular Pharmacology November 2010, 78 (5) 895-902; DOI: https://doi.org/10.1124/mol.110.066498
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  Microtubule-Targeted Chemotherapeutic Agents Inhibit Signal Transducer and Activator of Transcription 3 (STAT3) Signaling

  Sarah R. Walker, Mousumi Chaudhury, Erik A. Nelson and David A. Frank

  Molecular Pharmacology November 2010, 78 (5) 903-908; DOI: https://doi.org/10.1124/mol.110.066316
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  Poly(ADP-Ribose) Polymerase 1 Modulates the Lethality of CHK1 Inhibitors in Carcinoma Cells

  Clint Mitchell, Margaret Park, Patrick Eulitt, Chen Yang, Adly Yacoub and Paul Dent

  Molecular Pharmacology November 2010, 78 (5) 909-917; DOI: https://doi.org/10.1124/mol.110.067199
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  Alcohol- and Alcohol Antagonist-Sensitive Human GABA_A Receptors: Tracking δ Subunit Incorporation into Functional Receptors

  Pratap Meera, Richard W. Olsen, Thomas S. Otis and Martin Wallner

  Molecular Pharmacology November 2010, 78 (5) 918-924; DOI: https://doi.org/10.1124/mol.109.062687
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  The Tetrahydroisoquinoline Derivative SB269,652 Is an Allosteric Antagonist at Dopamine D₃ and D₂ Receptors

  Elena Silvano, Mark J. Millan, Clotilde Mannoury la Cour, Yang Han, Lihua Duan, Suzy A. Griffin, Robert R. Luedtke, Gabriella Aloisi, Mario Rossi, Francesca Zazzeroni, Jonathan A. Javitch and Roberto Maggio

  Molecular Pharmacology November 2010, 78 (5) 925-934; DOI: https://doi.org/10.1124/mol.110.065755
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  Morphine Regulates Dopaminergic Neuron Differentiation via miR-133b

  Fatima Macho Sanchez-Simon, Xiao Xiao Zhang, Horace H. Loh, Ping-Yee Law and Raquel E. Rodriguez

  Molecular Pharmacology November 2010, 78 (5) 935-942; DOI: https://doi.org/10.1124/mol.110.066837
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  Nijmegen Breakage Syndrome Protein (NBN) Causes Resistance to Methylating Anticancer Drugs Such as Temozolomide

  Marcus Eich, Wynand P. Roos, Grigory L. Dianov, Martin Digweed and Bernd Kaina

  Molecular Pharmacology November 2010, 78 (5) 943-951; DOI: https://doi.org/10.1124/mol.110.066076
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  Inhibition of Large-Conductance Ca²⁺-Activated K⁺ Channels by Nanomolar Concentrations of Ag⁺

  Yu Zhou, Xiaoming Xia and Christopher J. Lingle

  Molecular Pharmacology November 2010, 78 (5) 952-960; DOI: https://doi.org/10.1124/mol.110.066407
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  Discovery of Novel Forkhead Box O1 Inhibitors for Treating Type 2 Diabetes: Improvement of Fasting Glycemia in Diabetic db/db Mice

  Takeyuki Nagashima, Nobuharu Shigematsu, Riyo Maruki, Yasuharu Urano, Hirotsugu Tanaka, Akiyoshi Shimaya, Teruhiko Shimokawa and Masayuki Shibasaki

  Molecular Pharmacology November 2010, 78 (5) 961-970; DOI: https://doi.org/10.1124/mol.110.065714
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  α6β2* and α4β2* Nicotinic Receptors Both Regulate Dopamine Signaling with Increased Nigrostriatal Damage: Relevance to Parkinson's Disease

  Xiomara A. Perez, Tanuja Bordia, J. Michael McIntosh and Maryka Quik

  Molecular Pharmacology November 2010, 78 (5) 971-980; DOI: https://doi.org/10.1124/mol.110.067561