Table of Contents

Articles

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  Interactions of Key Charged Residues Contributing to Selective Block of Neuronal Sodium Channels by μ-Conotoxin KIIIA

  J. R. McArthur, G. Singh, D. McMaster, R. Winkfein, D. P. Tieleman and R. J. French

  Molecular Pharmacology October 2011, 80 (4) 573-584; DOI: https://doi.org/10.1124/mol.111.073460
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  Elucidation of the Contribution of Active Site and Exosite Interactions to Affinity and Specificity of Peptidylic Serine Protease Inhibitors Using Non-Natural Arginine Analogs

  Masood Hosseini, Longguang Jiang, Hans Peter Sørensen, Jan K. Jensen, Anni Christensen, Sarah Fogh, Cai Yuan, Lisbeth M. Andersen, Mingdong Huang, Peter A. Andreasen and Knud J. Jensen

  Molecular Pharmacology October 2011, 80 (4) 585-597; DOI: https://doi.org/10.1124/mol.111.072280
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  Novel Thiosemicarbazone Iron Chelators Induce Up-Regulation and Phosphorylation of the Metastasis Suppressor N-myc Down-Stream Regulated Gene 1: A New Strategy for the Treatment of Pancreatic Cancer

  Zaklina Kovacevic, Sherin Chikhani, David B. Lovejoy and Des R. Richardson

  Molecular Pharmacology October 2011, 80 (4) 598-609; DOI: https://doi.org/10.1124/mol.111.073627
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  The Selective Estrogen Receptor Modulator Bazedoxifene Inhibits Hormone-Independent Breast Cancer Cell Growth and Down-Regulates Estrogen Receptor α and Cyclin D1

  Joan S. Lewis-Wambi, Helen Kim, Ramona Curpan, Ronald Grigg, Mohammed A. Sarker and V. Craig Jordan

  Molecular Pharmacology October 2011, 80 (4) 610-620; DOI: https://doi.org/10.1124/mol.111.072249
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  The Antiepileptic Drugs Phenobarbital and Carbamazepine Reduce Transport of Methotrexate in Rat Choroid Plexus by Down-Regulation of the Reduced Folate Carrier

  Sandra Halwachs, Cathleen Lakoma, Ingo Schäfer, Peter Seibel and Walther Honscha

  Molecular Pharmacology October 2011, 80 (4) 621-629; DOI: https://doi.org/10.1124/mol.111.072421
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  Molecular Determinants for Activation of Human Ether-à-go-go-related Gene 1 Potassium Channels by 3-Nitro-N-(4-phenoxyphenyl) Benzamide

  Vivek Garg, Anna Stary-Weinzinger, Frank Sachse and Michael C. Sanguinetti

  Molecular Pharmacology October 2011, 80 (4) 630-637; DOI: https://doi.org/10.1124/mol.111.073809
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  Curcumin-Induced Mitotic Spindle Defect and Cell Cycle Arrest in Human Bladder Cancer Cells Occurs Partly through Inhibition of Aurora A

  Hsiao-Sheng Liu, Ching-Shiun Ke, Hung-Chi Cheng, Chi-Ying F. Huang and Chun-Li Su

  Molecular Pharmacology October 2011, 80 (4) 638-646; DOI: https://doi.org/10.1124/mol.111.072512
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  Three Arginines in the GABA_A Receptor Binding Pocket Have Distinct Roles in the Formation and Stability of Agonist- versus Antagonist-Bound Complexes

  Marcel P. Goldschen-Ohm, David A. Wagner and Mathew V. Jones

  Molecular Pharmacology October 2011, 80 (4) 647-656; DOI: https://doi.org/10.1124/mol.111.072033
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  Isoform-Selective Inhibition of Phosphoinositide 3-Kinase: Identification of a New Region of Nonconserved Amino Acids Critical for p110α Inhibition

  Zhaohua Zheng, Syazwani I. Amran, Philip E. Thompson and Ian G. Jennings

  Molecular Pharmacology October 2011, 80 (4) 657-664; DOI: https://doi.org/10.1124/mol.111.072546
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  Cooperative Role of Caveolin-1 and C-Terminal Src Kinase Binding Protein in C-Terminal Src Kinase-Mediated Negative Regulation of c-Src

  Aaron T. Place, Zhenlong Chen, Farnaz R. Bakhshi, Guoquan Liu, John P. O'Bryan and Richard D. Minshall

  Molecular Pharmacology October 2011, 80 (4) 665-672; DOI: https://doi.org/10.1124/mol.111.073957
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  Aryl Hydrocarbon Receptor Activation in Hematopoietic Stem/Progenitor Cells Alters Cell Function and Pathway-Specific Gene Modulation Reflecting Changes in Cellular Trafficking and Migration

  Fanny L. Casado, Kameshwar P. Singh and Thomas A. Gasiewicz

  Molecular Pharmacology October 2011, 80 (4) 673-682; DOI: https://doi.org/10.1124/mol.111.071381
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  Cyanoquinolines with Independent Corrector and Potentiator Activities Restore ΔPhe508-Cystic Fibrosis Transmembrane Conductance Regulator Chloride Channel Function in Cystic Fibrosis

  Puay-Wah Phuan, Baoxue Yang, John M. Knapp, Alex B. Wood, Gergely L. Lukacs, Mark J. Kurth and A. S. Verkman

  Molecular Pharmacology October 2011, 80 (4) 683-693; DOI: https://doi.org/10.1124/mol.111.073056
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  Novel Betulin Derivatives as Antileishmanial Agents with Mode of Action Targeting Type IB DNA Topoisomerase

  Sayan Chowdhury, Tulika Mukherjee, Souvik Sengupta, Somenath Roy Chowdhury, Sibabrata Mukhopadhyay and Hemanta K. Majumder

  Molecular Pharmacology October 2011, 80 (4) 694-703; DOI: https://doi.org/10.1124/mol.111.072785
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  Rat Embryo Exposure to All-Trans Retinoic Acid Results in Postnatal Oxidative Damage of Respiratory Complex I in the Cerebellum

  Anna Signorile, Nicola Sardaro, Domenico De Rasmo, Salvatore Scacco, Francesco Papa, Pietro Borracci, Maria Rosaria Carratù and Sergio Papa

  Molecular Pharmacology October 2011, 80 (4) 704-713; DOI: https://doi.org/10.1124/mol.111.073353
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  Valproic Acid Induces Monoamine Oxidase A via Akt/Forkhead Box O1 Activation

  Jason Boyang Wu and Jean C. Shih

  Molecular Pharmacology October 2011, 80 (4) 714-723; DOI: https://doi.org/10.1124/mol.111.072744
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  Inhibition of Navβ4 Peptide-Mediated Resurgent Sodium Currents in Nav1.7 Channels by Carbamazepine, Riluzole, and Anandamide

  Jonathan W. Theile and Theodore R. Cummins

  Molecular Pharmacology October 2011, 80 (4) 724-734; DOI: https://doi.org/10.1124/mol.111.072751
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  Identification of Cysteines Involved in the Effects of Methanethiosulfonate Reagents on Human Equilibrative Nucleoside Transporter 1

  Jamie S. Park, Scott J. Hughes, Frances K. M. Cunningham and James R. Hammond

  Molecular Pharmacology October 2011, 80 (4) 735-746; DOI: https://doi.org/10.1124/mol.111.072587
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  Long-Term α_1A-Adrenergic Receptor Stimulation Improves Synaptic Plasticity, Cognitive Function, Mood, and Longevity

  Van A. Doze, Robert S. Papay, Brianna L. Goldenstein, Manveen K. Gupta, Katie M. Collette, Brian W. Nelson, Mariaha J. Lyons, Bethany A. Davis, Elizabeth J. Luger, Sarah G. Wood, James R. Haselton, Paul C. Simpson and Dianne M. Perez

  Molecular Pharmacology October 2011, 80 (4) 747-758; DOI: https://doi.org/10.1124/mol.111.073734