Table of Contents

Articles

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  AC927, a σ Receptor Ligand, Blocks Methamphetamine-Induced Release of Dopamine and Generation of Reactive Oxygen Species in NG108-15 Cells

  Nidhi Kaushal, Meenal Elliott, Matthew J. Robson, Anand Krishnan V. Iyer, Yon Rojanasakul, Andrew Coop and Rae R. Matsumoto

  Molecular Pharmacology March 2012, 81 (3) 299-308; DOI: https://doi.org/10.1124/mol.111.074120
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  Lateral Allosterism in the Glucagon Receptor Family: Glucagon-Like Peptide 1 Induces G-Protein-Coupled Receptor Heteromer Formation

  Dominik Schelshorn, Fanny Joly, Sophie Mutel, Cornelia Hampe, Billy Breton, Vincent Mutel and Robert Lütjens

  Molecular Pharmacology March 2012, 81 (3) 309-318; DOI: https://doi.org/10.1124/mol.111.074757
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  Rosiglitazone and Metformin Have Opposite Effects on Intestinal Absorption of Oligopeptides via the Proton-Dependent PepT1 Transporter

  Patrick Hindlet, Claire Barraud, Laura Boschat, Robert Farinotti, André Bado and Marion Buyse

  Molecular Pharmacology March 2012, 81 (3) 319-327; DOI: https://doi.org/10.1124/mol.111.073874
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  Xanthines Down-Regulate the Drug Transporter ABCG2 and Reverse Multidrug Resistance

  Rui Ding, Jia Shi, Kirk Pabon and Kathleen W. Scotto

  Molecular Pharmacology March 2012, 81 (3) 328-337; DOI: https://doi.org/10.1124/mol.111.075556
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  A Novel Nonconsensus Xenobiotic Response Element Capable of Mediating Aryl Hydrocarbon Receptor-Dependent Gene Expression

  Gengming Huang and Cornelis J. Elferink

  Molecular Pharmacology March 2012, 81 (3) 338-347; DOI: https://doi.org/10.1124/mol.111.075952
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  Desensitization and Trafficking of μ-Opioid Receptors in Locus Ceruleus Neurons: Modulation by Kinases

  Seksiri Arttamangkul, Elaine K. Lau, Hsin-Wei Lu and John T. Williams

  Molecular Pharmacology March 2012, 81 (3) 348-355; DOI: https://doi.org/10.1124/mol.111.076208
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  Defining Substrate and Blocker Activity of Alanine-Serine-Cysteine Transporter 2 (ASCT2) Ligands with Novel Serine Analogs

  Thomas Albers, William Marsiglia, Taniya Thomas, Armanda Gameiro and Christof Grewer

  Molecular Pharmacology March 2012, 81 (3) 356-365; DOI: https://doi.org/10.1124/mol.111.075648
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  Role of the Local Anesthetic Receptor in the State-Dependent Inhibition of Voltage-Gated Sodium Channels by the Insecticide Metaflumizone

  Richard T. von Stein and David M. Soderlund

  Molecular Pharmacology March 2012, 81 (3) 366-374; DOI: https://doi.org/10.1124/mol.111.075283
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  Signaling Cascades for δ-Opioid Receptor-Mediated Inhibition of GABA Synaptic Transmission and Behavioral Antinociception

  Zhi Zhang and Zhizhong Z. Pan

  Molecular Pharmacology March 2012, 81 (3) 375-383; DOI: https://doi.org/10.1124/mol.111.076307
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  Heteromeric Canonical Transient Receptor Potential 1 and 4 Channels Play a Critical Role in Epileptiform Burst Firing and Seizure-Induced Neurodegeneration

  Kevin D. Phelan, Matthew M. Mock, Oliver Kretz, U. Thaung Shwe, Maxim Kozhemyakin, L. John Greenfield, Alexander Dietrich, Lutz Birnbaumer, Marc Freichel, Veit Flockerzi and Fang Zheng

  Molecular Pharmacology March 2012, 81 (3) 384-392; DOI: https://doi.org/10.1124/mol.111.075341
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  Covalent Modification of a Volatile Anesthetic Regulatory Site Activates TASK-3 (KCNK9) Tandem-Pore Potassium Channels

  Kevin E. Conway and Joseph F. Cotten

  Molecular Pharmacology March 2012, 81 (3) 393-400; DOI: https://doi.org/10.1124/mol.111.076281
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  Antitumor Indolequinones Induced Apoptosis in Human Pancreatic Cancer Cells via Inhibition of Thioredoxin Reductase and Activation of Redox Signaling

  Chao Yan, David Siegel, Jeffery Newsome, Aurelie Chilloux, Christopher J. Moody and David Ross

  Molecular Pharmacology March 2012, 81 (3) 401-410; DOI: https://doi.org/10.1124/mol.111.076091
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  Transient Receptor Potential Vanilloid-1 (TRPV1) Is a Mediator of Lung Toxicity for Coal Fly Ash Particulate Material

  Cassandra E. Deering-Rice, Mark E. Johansen, Jessica K. Roberts, Karen C. Thomas, Erin G. Romero, Jeewoo Lee, Garold S. Yost, John M. Veranth and Christopher A. Reilly

  Molecular Pharmacology March 2012, 81 (3) 411-419; DOI: https://doi.org/10.1124/mol.111.076067
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  Protein Kinase C Regulation of 12-Lipoxygenase-Mediated Human Platelet Activation

  Jennifer Yeung, Patrick L. Apopa, Joanne Vesci, Victor Kenyon, Ganesha Rai, Ajit Jadhav, Anton Simeonov, Theodore R. Holman, David J. Maloney, Olivier Boutaud and Michael Holinstat

  Molecular Pharmacology March 2012, 81 (3) 420-430; DOI: https://doi.org/10.1124/mol.111.075630
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  Polygamain, a New Microtubule Depolymerizing Agent That Occupies a Unique Pharmacophore in the Colchicine Site

  R. M. Hartley, J. Peng, G. A. Fest, S. Dakshanamurthy, D. E. Frantz, M. L. Brown and S. L. Mooberry

  Molecular Pharmacology March 2012, 81 (3) 431-439; DOI: https://doi.org/10.1124/mol.111.075838
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  Inhibition of Prohormone Convertases PC1/3 and PC2 by 2,5-Dideoxystreptamine Derivatives

  Mirella Vivoli, Thomas R. Caulfield, Karina Martínez-Mayorga, Alan T. Johnson, Guan-Sheng Jiao and Iris Lindberg

  Molecular Pharmacology March 2012, 81 (3) 440-454; DOI: https://doi.org/10.1124/mol.111.077040
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  Specificity Protein 1 (Sp1) Oscillation Is Involved in Copper Homeostasis Maintenance by Regulating Human High-Affinity Copper Transporter 1 Expression

  Zheng D. Liang, Wen-Bin Tsai, Mei-Yi Lee, Niramol Savaraj and Macus Tien Kuo

  Molecular Pharmacology March 2012, 81 (3) 455-464; DOI: https://doi.org/10.1124/mol.111.076422
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  Alteration in Accumulated Aldosterone Synthesis As a Result of N-Terminal Cleavage of Aldosterone Synthase

  Brian P. Adams and Himangshu S. Bose

  Molecular Pharmacology March 2012, 81 (3) 465-474; DOI: https://doi.org/10.1124/mol.111.076471
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  A Novel Nonribose Agonist, LUF5834, Engages Residues That Are Distinct from Those of Adenosine-Like Ligands to Activate the Adenosine A_2a Receptor

  J. Robert Lane, Carmen Klein Herenbrink, Gerard J. P. van Westen, Jelle A. Spoorendonk, Carsten Hoffmann and Adriaan P. IJzerman

  Molecular Pharmacology March 2012, 81 (3) 475-487; DOI: https://doi.org/10.1124/mol.111.075937
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  Characterization of the Substituted N-Triazole Oxindole TROX-1, a Small-Molecule, State-Dependent Inhibitor of Ca_v2 Calcium Channels

  Andrew M. Swensen, James Herrington, Randal M. Bugianesi, Ge Dai, Rodolfo J. Haedo, Kevin S. Ratliff, McHardy M. Smith, Vivien A. Warren, Stephen P. Arneric, Cyrus Eduljee, David Parker, Terrance P. Snutch, Scott B. Hoyt, Clare London, Joseph L. Duffy, Gregory J. Kaczorowski and Owen B. McManus

  Molecular Pharmacology March 2012, 81 (3) 488-497; DOI: https://doi.org/10.1124/mol.111.075226