Table of Contents

Articles

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  New Insights for Drug Design from the X-Ray Crystallographic Structures of G-Protein-Coupled Receptors

  Kenneth A. Jacobson and Stefano Costanzi

  Molecular Pharmacology September 2012, 82 (3) 361-371; DOI: https://doi.org/10.1124/mol.112.079335
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  Vm24, a Natural Immunosuppressive Peptide, Potently and Selectively Blocks Kv1.3 Potassium Channels of Human T Cells

  Zoltan Varga, Georgina Gurrola-Briones, Ferenc Papp, Ricardo C. Rodríguez de la Vega, Gustavo Pedraza-Alva, Rajeev B. Tajhya, Rezso Gaspar, Luis Cardenas, Yvonne Rosenstein, Christine Beeton, Lourival D. Possani and Gyorgy Panyi

  Molecular Pharmacology September 2012, 82 (3) 372-382; DOI: https://doi.org/10.1124/mol.112.078006
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  Carbonylation Induces Heterogeneity in Cardiac Ryanodine Receptor Function in Diabetes Mellitus

  Chun Hong Shao, Chengju Tian, Shouqiang Ouyang, Caronda J. Moore, Fadhel Alomar, Ina Nemet, Alicia D'Souza, Ryoji Nagai, Shelby Kutty, George J. Rozanski, Sasanka Ramanadham, Jaipaul Singh and Keshore R. Bidasee

  Molecular Pharmacology September 2012, 82 (3) 383-399; DOI: https://doi.org/10.1124/mol.112.078352
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  A New 2-Pyrone Derivative, 5-Bromo-3-(3-hydroxyprop-1-ynyl)-2H-pyran-2-one, Suppresses Stemness in Glioma Stem-Like Cells

  Rae-Kwon Kim, Min-Jung Kim, Chang-Hwan Yoon, Eun-Jung Lim, Ki-Chun Yoo, Ga-Haeng Lee, Young-Heon Kim, Hyeonmi Kim, Yeung Bae Jin, Yoon-Jin Lee, Cheon-Gyu Cho, Yeong Seok Oh, Myung Chan Gye, Yongjoon Suh and Su-Jae Lee

  Molecular Pharmacology September 2012, 82 (3) 400-407; DOI: https://doi.org/10.1124/mol.112.078402
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  Neurosteroid Analog Photolabeling of a Site in the Third Transmembrane Domain of the β3 Subunit of the GABA_A Receptor

  Zi-Wei Chen, Brad Manion, R. Reid Townsend, David E. Reichert, Douglas F. Covey, Joe Henry Steinbach, Werner Sieghart, Karoline Fuchs and Alex S. Evers

  Molecular Pharmacology September 2012, 82 (3) 408-419; DOI: https://doi.org/10.1124/mol.112.078410
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  Tetrahydrobiopterin Protects Soluble Guanylate Cyclase against Oxidative Inactivation

  Kurt Schmidt, Andrea Neubauer, Bernd Kolesnik, Johannes-Peter Stasch, Ernst R. Werner, Antonius C. F. Gorren and Bernd Mayer

  Molecular Pharmacology September 2012, 82 (3) 420-427; DOI: https://doi.org/10.1124/mol.112.079855
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  Long QT2 Mutation on the Kv11.1 Ion Channel Inhibits Current Activity by Ablating a Protein Kinase Cα Consensus Site

  Alexander J. Donovan, Katherine Lansu, Jason G. Williams, Mitchell F. Denning and Saverio Gentile

  Molecular Pharmacology September 2012, 82 (3) 428-437; DOI: https://doi.org/10.1124/mol.112.077966
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  Functional and Pharmacological Characteristics of Metabotropic Glutamate Receptors 2/4 Heterodimers

  Paul J. Kammermeier

  Molecular Pharmacology September 2012, 82 (3) 438-447; DOI: https://doi.org/10.1124/mol.112.078501
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  Computational and Experimental Analysis of the Transmembrane Domain 4/5 Dimerization Interface of the Serotonin 5-HT_1A Receptor

  Nataliya Gorinski, Noga Kowalsman, Ute Renner, Alexander Wirth, Michael T. Reinartz, Roland Seifert, Andre Zeug, Evgeni Ponimaskin and Masha Y. Niv

  Molecular Pharmacology September 2012, 82 (3) 448-463; DOI: https://doi.org/10.1124/mol.112.079137
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  Optical Recording Reveals Novel Properties of GSK1016790A-Induced Vanilloid Transient Receptor Potential Channel TRPV4 Activity in Primary Human Endothelial Cells

  Michelle N. Sullivan, Michael Francis, Natalie L. Pitts, Mark S. Taylor and Scott Earley

  Molecular Pharmacology September 2012, 82 (3) 464-472; DOI: https://doi.org/10.1124/mol.112.078584
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  Prolonged Stimulation of μ-Opioid Receptors Produces β-Arrestin-2-Mediated Heterologous Desensitization of α₂-Adrenoceptor Function in Locus Ceruleus Neurons

  Vu C. Dang, Billy C. Chieng and MacDonald J. Christie

  Molecular Pharmacology September 2012, 82 (3) 473-480; DOI: https://doi.org/10.1124/mol.112.079350
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  Common Mechanisms of Drug Interactions with Sodium and T-Type Calcium Channels

  Chris Bladen and Gerald W. Zamponi

  Molecular Pharmacology September 2012, 82 (3) 481-487; DOI: https://doi.org/10.1124/mol.112.079715
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  Casein Kinase 2α Regulates Multidrug Resistance-Associated Protein 1 Function via Phosphorylation of Thr249

  Elzbieta I. Stolarczyk, Cassandra J. Reiling, Kerry A. Pickin, Ryan Coppage, Marc R. Knecht and Christian M. Paumi

  Molecular Pharmacology September 2012, 82 (3) 488-499; DOI: https://doi.org/10.1124/mol.112.078295
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  Cardiotonic Steroids Stabilize Regulator of G Protein Signaling 2 Protein Levels

  Benita Sjögren, Sergio Parra, Lauren J. Heath, Kevin B. Atkins, Zie-Jian Xie and Richard R. Neubig

  Molecular Pharmacology September 2012, 82 (3) 500-509; DOI: https://doi.org/10.1124/mol.112.079293
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  Sec61β Controls Sensitivity to Platinum-Containing Chemotherapeutic Agents through Modulation of the Copper-Transporting ATPase ATP7A

  Paolo B. Abada, Christopher A. Larson, Gerald Manorek, Preston Adams and Stephen B. Howell

  Molecular Pharmacology September 2012, 82 (3) 510-520; DOI: https://doi.org/10.1124/mol.112.079822
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  Transcriptome Analysis and In Vivo Activity of Fluvastatin versus Zoledronic Acid in a Murine Breast Cancer Metastasis Model

  Nadejda Vintonenko, Jean-Philippe Jais, Nadim Kassis, Mohamed Abdelkarim, Gerard-Yves Perret, Marc Lecouvey, Michel Crepin and Melanie Di Benedetto

  Molecular Pharmacology September 2012, 82 (3) 521-528; DOI: https://doi.org/10.1124/mol.111.077248
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  Human CYP2C8 Is Post-Transcriptionally Regulated by MicroRNAs 103 and 107 in Human Liver

  Shu-Yun Zhang, Sailesh Surapureddi, Sherry Coulter, Stephen S. Ferguson and Joyce A. Goldstein

  Molecular Pharmacology September 2012, 82 (3) 529-540; DOI: https://doi.org/10.1124/mol.112.078386
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  Calcium Channel Blockers Act through Nuclear Factor Y to Control Transcription of Key Cardiac Genes

  Hyunjoo Cha-Molstad, Guanlan Xu, Junqin Chen, Gu Jing, Martin E. Young, John C. Chatham and Anath Shalev

  Molecular Pharmacology September 2012, 82 (3) 541-549; DOI: https://doi.org/10.1124/mol.112.078253
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  Contribution of Subunits to Caenorhabditis elegans Levamisole-Sensitive Nicotinic Receptor Function

  Guillermina Hernando, Ignacio Bergé, Diego Rayes and Cecilia Bouzat

  Molecular Pharmacology September 2012, 82 (3) 550-560; DOI: https://doi.org/10.1124/mol.112.079962