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Molecular Pharmacology

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Table of Contents

October 01, 2012; Volume 82,Issue 4

Minireview

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    Ubiquitination of G Protein-Coupled Receptors: Functional Implications and Drug Discovery
    Michael R. Dores and JoAnn Trejo
    Molecular Pharmacology October 2012, 82 (4) 563-570; DOI: https://doi.org/10.1124/mol.112.079418

Perspective

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    Casting a Wider Net: Whole-Cell Assays to Capture Varied and Biased Signaling
    Terry Kenakin
    Molecular Pharmacology October 2012, 82 (4) 571-574; DOI: https://doi.org/10.1124/mol.112.081117

Accelerated Communication

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    Design and Functional Characterization of a Novel, Arrestin-Biased Designer G Protein-Coupled Receptor
    Ken-ichiro Nakajima and Jürgen Wess
    Molecular Pharmacology October 2012, 82 (4) 575-582; DOI: https://doi.org/10.1124/mol.112.080358

Articles

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    Increasing Human Th17 Differentiation through Activation of Orphan Nuclear Receptor Retinoid Acid-Related Orphan Receptor γ (RORγ) by a Class of Aryl Amide Compounds
    Wei Zhang, Jing Zhang, Leiping Fang, Ling Zhou, Shuai Wang, Zhijun Xiang, Yuan Li, Bruce Wisely, Guifeng Zhang, Gang An, Yonghui Wang, Stewart Leung and Zhong Zhong
    Molecular Pharmacology October 2012, 82 (4) 583-590; DOI: https://doi.org/10.1124/mol.112.078667
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    Functional Loss of the Reduced Folate Carrier Enhances the Antitumor Activities of Novel Antifolates with Selective Uptake by the Proton-Coupled Folate Transporter
    Sita Kugel Desmoulin, Lei Wang, Lisa Polin, Kathryn White, Juiwanna Kushner, Mark Stout, Zhanjun Hou, Christina Cherian, Aleem Gangjee and Larry H. Matherly
    Molecular Pharmacology October 2012, 82 (4) 591-600; DOI: https://doi.org/10.1124/mol.112.079004
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    Activator Protein-1 Regulation of Murine Aldehyde Dehydrogenase 1a1
    N. L. Makia, I. Amunom, K. C. Falkner, D. J. Conklin, S. Surapureddi, J. A. Goldstein and R. A. Prough
    Molecular Pharmacology October 2012, 82 (4) 601-613; DOI: https://doi.org/10.1124/mol.112.078147
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    Anacardic Acid Inhibits the Catalytic Activity of Matrix Metalloproteinase-2 and Matrix Metalloproteinase-9
    Athira Omanakuttan, Jyotsna Nambiar, Rodney M. Harris, Chinchu Bose, Nanjan Pandurangan, Rebu K. Varghese, Geetha B. Kumar, John A. Tainer, Asoke Banerji, J. Jefferson P. Perry and Bipin G. Nair
    Molecular Pharmacology October 2012, 82 (4) 614-622; DOI: https://doi.org/10.1124/mol.112.079020
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    RNA Aptamer-Based Functional Ligands of the Neurotrophin Receptor, TrkB
    Yang Zhong Huang, Frank J. Hernandez, Bin Gu, Katie R. Stockdale, Kishore Nanapaneni, Todd E. Scheetz, Mark A. Behlke, Andrew S. Peek, Thomas Bair, Paloma H. Giangrande and James O. McNamara
    Molecular Pharmacology October 2012, 82 (4) 623-635; DOI: https://doi.org/10.1124/mol.112.078220
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    P-Glycoprotein, Multidrug-Resistance Associated Protein 2, Cyp3a, and Carboxylesterase Affect the Oral Availability and Metabolism of Vinorelbine
    Jurjen S. Lagas, Carola W. N. Damen, Robert A. B. van Waterschoot, Dilek Iusuf, Jos H. Beijnen and Alfred H. Schinkel
    Molecular Pharmacology October 2012, 82 (4) 636-644; DOI: https://doi.org/10.1124/mol.111.077099
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    Discovery of Regulators of Receptor Internalization with High-Throughput Flow Cytometry
    Yang Wu, Phillip H. Tapia, Gregory W. Fisher, Peter C. Simons, J. Jacob Strouse, Terry Foutz, Alan S. Waggoner, Jonathan Jarvik and Larry A. Sklar
    Molecular Pharmacology October 2012, 82 (4) 645-657; DOI: https://doi.org/10.1124/mol.112.079897
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    Block of Human CaV3 Channels by the Diuretic Amiloride
    Osbaldo Lopez-Charcas, Manuel Rivera and Juan C. Gomora
    Molecular Pharmacology October 2012, 82 (4) 658-667; DOI: https://doi.org/10.1124/mol.112.078923
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    D2-Dopaminergic Receptor-Linked Pathways: Critical Regulators of CYP3A, CYP2C, and CYP2D
    Evangelos P. Daskalopoulos, Matti A. Lang, Marios Marselos, Foteini Malliou and Maria Konstandi
    Molecular Pharmacology October 2012, 82 (4) 668-678; DOI: https://doi.org/10.1124/mol.112.078709
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    CYP4V2 in Bietti's Crystalline Dystrophy: Ocular Localization, Metabolism of ω-3-Polyunsaturated Fatty Acids, and Functional Deficit of the p.H331P Variant
    Mariko Nakano, Edward J. Kelly, Constanze Wiek, Helmut Hanenberg and Allan E. Rettie
    Molecular Pharmacology October 2012, 82 (4) 679-686; DOI: https://doi.org/10.1124/mol.112.080085
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    Synthesis of Selective Agonists for the α7 Nicotinic Acetylcholine Receptor with In Situ Click-Chemistry on Acetylcholine-Binding Protein Templates
    John G. Yamauchi, Kimberly Gomez, Neil Grimster, Mikael Dufouil, Ákos Nemecz, Joseph R. Fotsing, Kwok-Yiu Ho, Todd T. Talley, K. Barry Sharpless, Valery V. Fokin and Palmer Taylor
    Molecular Pharmacology October 2012, 82 (4) 687-699; DOI: https://doi.org/10.1124/mol.112.080291
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    Therapeutic Potential of Nitric Oxide-Modified Drugs in Colon Cancer Cells
    Marija Mojic, Sanja Mijatovic, Danijela Maksimovic-Ivanic, Djordje Miljkovic, Stanislava Stosic-Grujicic, Marija Stankovic, Katia Mangano, Salvatore Travali, Marco Donia, Paolo Fagone, Mai-Britt Zocca, Yousef Al-Abed, James A. McCubrey and Ferdinando Nicoletti
    Molecular Pharmacology October 2012, 82 (4) 700-710; DOI: https://doi.org/10.1124/mol.112.077842
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    Efficient Binding of 4/7 α-Conotoxins to Nicotinic α4β2 Receptors Is Prevented by Arg185 and Pro195 in the α4 Subunit
    Mirko Beissner, Sébastien Dutertre, Rudolf Schemm, Timm Danker, Annett Sporning, Helmut Grubmüller and Annette Nicke
    Molecular Pharmacology October 2012, 82 (4) 711-718; DOI: https://doi.org/10.1124/mol.112.078683
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    Regulation of Sphingomyelin Phosphodiesterase Acid-Like 3A Gene (SMPDL3A) by Liver X Receptors
    Paul B. Noto, Yuri Bukhtiyarov, Meng Shi, Brian M. McKeever, Gerard M. McGeehan and Deepak S. Lala
    Molecular Pharmacology October 2012, 82 (4) 719-727; DOI: https://doi.org/10.1124/mol.112.078865
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    Sustained Activation of N-Methyl-d-Aspartate Receptors in Podoctyes Leads to Oxidative Stress, Mobilization of Transient Receptor Potential Canonical 6 Channels, Nuclear Factor of Activated T Cells Activation, and Apoptotic Cell Death
    Eun Young Kim, Marc Anderson and Stuart E. Dryer
    Molecular Pharmacology October 2012, 82 (4) 728-737; DOI: https://doi.org/10.1124/mol.112.079376
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    A Role for Kalirin in the Response of Rat Medium Spiny Neurons to Cocaine
    Xin-Ming Ma, Jian-ping Huang, Xiaonan Xin, Yan Yan, Richard E. Mains and Betty A. Eipper
    Molecular Pharmacology October 2012, 82 (4) 738-745; DOI: https://doi.org/10.1124/mol.112.080044
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    Intrinsically Low Open Probability of α7 Nicotinic Acetylcholine Receptors Can Be Overcome by Positive Allosteric Modulation and Serum Factors Leading to the Generation of Excitotoxic Currents at Physiological Temperatures
    Dustin K. Williams, Can Peng, Matthew R. Kimbrell and Roger L. Papke
    Molecular Pharmacology October 2012, 82 (4) 746-759; DOI: https://doi.org/10.1124/mol.112.080317
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    Activation of Trimeric P2X2 Receptors by Fewer than Three ATP Molecules
    Olga Stelmashenko, Ulyana Lalo, Yue Yang, Laricia Bragg, R. Alan North and Vincent Compan
    Molecular Pharmacology October 2012, 82 (4) 760-766; DOI: https://doi.org/10.1124/mol.112.080903
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    Identification of DNA Repair Pathways That Affect the Survival of Ovarian Cancer Cells Treated with a Poly(ADP-Ribose) Polymerase Inhibitor in a Novel Drug Combination
    Amelia M. Huehls, Jill M. Wagner, Catherine J. Huntoon and Larry M. Karnitz
    Molecular Pharmacology October 2012, 82 (4) 767-776; DOI: https://doi.org/10.1124/mol.112.080614
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In this issue

Molecular Pharmacology: 82 (4)
Molecular Pharmacology
Vol. 82, Issue 4
1 Oct 2012
  • Table of Contents
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  • The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints
  • Pharmacological Properties of Y-27632, a Specific Inhibitor of Rho-Associated Kinases
  • Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
  • The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation of CYP3A4 by Rifampicin through a Distal Enhancer Module
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