Table of Contents

Articles

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  Effect of Ifenprodil on GluN1/GluN2B N-Methyl-D-aspartate Receptor Gating

  Jay M. Bhatt, Anand Prakash, Pratyush S. Suryavanshi and Shashank M. Dravid

  Molecular Pharmacology January 2013, 83 (1) 9-21; DOI: https://doi.org/10.1124/mol.112.080952
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  DCPIB, the Proposed Selective Blocker of Volume-Regulated Anion Channels, Inhibits Several Glutamate Transport Pathways in Glial Cells

  Nicole H. Bowens, Preeti Dohare, Yu-Hung Kuo and Alexander A. Mongin

  Molecular Pharmacology January 2013, 83 (1) 22-32; DOI: https://doi.org/10.1124/mol.112.080457
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  Mithramycin A Inhibits Myeloid Cell Leukemia-1 to Induce Apoptosis in Oral Squamous Cell Carcinomas and Tumor Xenograft through Activation of Bax and Oligomerization

  Ji-Ae Shin, Ji-Youn Jung, Mi Heon Ryu, Stephen Safe and Sung-Dae Cho

  Molecular Pharmacology January 2013, 83 (1) 33-41; DOI: https://doi.org/10.1124/mol.112.081364
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  Functional Selectivity in Serotonin Receptor 2A (5-HT_2A) Endocytosis, Recycling, and Phosphorylation

  Ishier Raote, Samarjit Bhattacharyya and Mitradas M. Panicker

  Molecular Pharmacology January 2013, 83 (1) 42-50; DOI: https://doi.org/10.1124/mol.112.078626
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  Glitazones Exert Multiple Effects on β-Cell Stimulus-Secretion Coupling

  Martina Düfer, Katja Noack, Armin Edalat, Peter Krippeit-Drews and Gisela Drews

  Molecular Pharmacology January 2013, 83 (1) 51-60; DOI: https://doi.org/10.1124/mol.112.081638
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  Identification and Characterization of Poly(I:C)-induced Molecular Responses Attenuated by Nicotine in Mouse Macrophages

  Wen-Yan Cui, Shufang Zhao, Renata Polanowska-Grabowska, Ju Wang, Jinxue Wei, Bhagirathi Dash, Sulie L. Chang, Jeffrey J. Saucerman, Jun Gu and Ming D. Li

  Molecular Pharmacology January 2013, 83 (1) 61-72; DOI: https://doi.org/10.1124/mol.112.081497
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  Salt Bridge Switching from Arg290/Glu167 to Arg290/ATP Promotes the Closed-to-Open Transition of the P2X2 Receptor

  Ralf Hausmann, Janka Günther, Achim Kless, Daniel Kuhlmann, Matthias U. Kassack, Gregor Bahrenberg, Fritz Markwardt and Günther Schmalzing

  Molecular Pharmacology January 2013, 83 (1) 73-84; DOI: https://doi.org/10.1124/mol.112.081489
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  Claudin-3 and Claudin-4 Regulate Sensitivity to Cisplatin by Controlling Expression of the Copper and Cisplatin Influx Transporter CTR1

  Xiying Shang, Xinjian Lin, Gerald Manorek and Stephen B. Howell

  Molecular Pharmacology January 2013, 83 (1) 85-94; DOI: https://doi.org/10.1124/mol.112.079798
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  A New Site and Mechanism of Action for the Widely Used Adenylate Cyclase Inhibitor SQ22,536

  Andrew C. Emery, Maribeth V. Eiden and Lee E. Eiden

  Molecular Pharmacology January 2013, 83 (1) 95-105; DOI: https://doi.org/10.1124/mol.112.081760
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  Activation of Group I Metabotropic Glutamate Receptors Potentiates Heteromeric Kainate Receptors

  Asheebo Rojas, Jonathon Wetherington, Renee Shaw, Geidy Serrano, Sharon Swanger and Raymond Dingledine

  Molecular Pharmacology January 2013, 83 (1) 106-121; DOI: https://doi.org/10.1124/mol.112.081802
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  A Novel EPAC-Specific Inhibitor Suppresses Pancreatic Cancer Cell Migration and Invasion

  Muayad Almahariq, Tamara Tsalkova, Fang C. Mei, Haijun Chen, Jia Zhou, Sarita K. Sastry, Frank Schwede and Xiaodong Cheng

  Molecular Pharmacology January 2013, 83 (1) 122-128; DOI: https://doi.org/10.1124/mol.112.080689
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  β-Adrenergic Agonists Mediate Enhancement of β₁-Adrenergic Receptor N-terminal Cleavage and Stabilization In Vivo and In Vitro

  Anna E. Hakalahti, Hamayun Khan, Miia M. Vierimaa, Emilia H. Pekkala, Jarkko J. Lackman, Johanna Ulvila, Risto Kerkelä and Ulla E. Petäjä-Repo

  Molecular Pharmacology January 2013, 83 (1) 129-141; DOI: https://doi.org/10.1124/mol.112.080440
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  Neurounina-1, a Novel Compound That Increases Na⁺/Ca²⁺ Exchanger Activity, Effectively Protects against Stroke Damage

  Pasquale Molinaro, Maria Cantile, Ornella Cuomo, Agnese Secondo, Anna Pannaccione, Paolo Ambrosino, Giuseppe Pignataro, Ferdinando Fiorino, Beatrice Severino, Elena Gatta, Maria José Sisalli, Marco Milanese, Antonella Scorziello, Giambattista Bonanno, Mauro Robello, Vincenzo Santagada, Giuseppe Caliendo, Gianfranco Di Renzo and Lucio Annunziato

  Molecular Pharmacology January 2013, 83 (1) 142-156; DOI: https://doi.org/10.1124/mol.112.080986
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  The Biarylpyrazole Compound AM251 Alters Mitochondrial Physiology via Proteolytic Degradation of ERRα

  Susan M. Krzysik-Walker, Isabel González-Mariscal, Morten Scheibye-Knudsen, Fred E. Indig and Michel Bernier

  Molecular Pharmacology January 2013, 83 (1) 157-166; DOI: https://doi.org/10.1124/mol.112.082651
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  Pivotal Role of Reactive Oxygen Species in Differential Regulation of Lipopolysaccharide-Induced Prostaglandins Production in Macrophages

  Guiqing Zhao, Rui Yu, Jing Deng, Qiong Zhao, Yongchao Li, Myungsoo Joo, Richard B. van Breemen, John W. Christman and Lei Xiao

  Molecular Pharmacology January 2013, 83 (1) 167-178; DOI: https://doi.org/10.1124/mol.112.080762
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  The Iron Chelator, Deferasirox, as a Novel Strategy for Cancer Treatment: Oral Activity Against Human Lung Tumor Xenografts and Molecular Mechanism of Action

  Goldie Y. L. Lui, Peyman Obeidy, Samuel J. Ford, Chris Tselepis, Danae M. Sharp, Patric J. Jansson, Danuta S. Kalinowski, Zaklina Kovacevic, David B. Lovejoy and Des R. Richardson

  Molecular Pharmacology January 2013, 83 (1) 179-190; DOI: https://doi.org/10.1124/mol.112.081893
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  Potentiation of Sulfonylurea Action by an EPAC-selective cAMP Analog in INS-1 Cells: Comparison of Tolbutamide and Gliclazide and a Potential Role for EPAC Activation of a 2-APB-sensitive Ca²⁺ Influx

  Rachel E. Jarrard, Yuchen Wang, Amy E. Salyer, Evan P.S. Pratt, Ian M. Soderling, Marcy L. Guerra, Allison M. Lange, Hilary J. Broderick and Gregory H. Hockerman

  Molecular Pharmacology January 2013, 83 (1) 191-205; DOI: https://doi.org/10.1124/mol.112.081943
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  Extracellular Loop II Modulates GTP Sensitivity of the Prostaglandin EP3 Receptor

  Chandramohan Natarajan, Aaron N. Hata, Heidi E. Hamm, Roy Zent and Richard M. Breyer

  Molecular Pharmacology January 2013, 83 (1) 206-216; DOI: https://doi.org/10.1124/mol.112.080473
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  Lysine 48-Linked Polyubiquitination of Organic Anion Transporter-1 Is Essential for Its Protein Kinase C–Regulated Endocytosis

  Qiang Zhang, Shanshan Li, Cam Patterson and Guofeng You

  Molecular Pharmacology January 2013, 83 (1) 217-224; DOI: https://doi.org/10.1124/mol.112.082065
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  The Anticancer Ruthenium Complex KP1019 Induces DNA Damage, Leading to Cell Cycle Delay and Cell Death in Saccharomyces cerevisiae

  Shannon K. Stevens, Amy P. Strehle, Rebecca L. Miller, Sarah H. Gammons, Kyle J. Hoffman, John T. McCarty, Mary E. Miller, Laura K. Stultz and Pamela K. Hanson

  Molecular Pharmacology January 2013, 83 (1) 225-234; DOI: https://doi.org/10.1124/mol.112.079657
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  Distinct Sensitivity of Slo1 Channel Proteins to Ethanol

  Jianxi Liu, Anna N. Bukiya, Guruprasad Kuntamallappanavar, Aditya K. Singh and Alex M. Dopico

  Molecular Pharmacology January 2013, 83 (1) 235-244; DOI: https://doi.org/10.1124/mol.112.081240
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  Requirement of Apoptotic Protease-Activating Factor-1 for Bortezomib-Induced Apoptosis but Not for Fas-Mediated Apoptosis in Human Leukemic Cells

  Astrid Ottosson-Wadlund, Rebecca Ceder, Giulio Preta, Katja Pokrovskaja, Roland C. Grafström, Mats Heyman, Stefan Söderhäll, Dan Grandér, Ingrid Hedenfalk, John D. Robertson and Bengt Fadeel

  Molecular Pharmacology January 2013, 83 (1) 245-255; DOI: https://doi.org/10.1124/mol.112.080788
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  Identification of Determinants Required for Agonistic and Inverse Agonistic Ligand Properties at the ADP Receptor P2Y₁₂

  Philipp Schmidt, Lars Ritscher, Elizabeth N. Dong, Thomas Hermsdorf, Maxi Cöster, Doreen Wittkopf, Jens Meiler and Torsten Schöneberg

  Molecular Pharmacology January 2013, 83 (1) 256-266; DOI: https://doi.org/10.1124/mol.112.082198
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  N-Arachidonyl Glycine Does Not Activate G Protein–Coupled Receptor 18 Signaling via Canonical Pathways

  Van B. Lu, Henry L. Puhl and Stephen R. Ikeda

  Molecular Pharmacology January 2013, 83 (1) 267-282; DOI: https://doi.org/10.1124/mol.112.081182
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  BET Bromodomain Proteins Mediate Downstream Signaling Events following Growth Factor Stimulation in Human Lung Fibroblasts and Are Involved in Bleomycin-Induced Pulmonary Fibrosis

  Xiaoyan Tang, Ruoqi Peng, Yonglin Ren, Subramanium Apparsundaram, Jeremy Deguzman, Carla M. Bauer, Ann F. Hoffman, Shannon Hamilton, Zhenmin Liang, Hang Zeng, Maria E. Fuentes, Julie A. DeMartino, Christopher Kitson, Christopher S. Stevenson and David C. Budd

  Molecular Pharmacology January 2013, 83 (1) 283-293; DOI: https://doi.org/10.1124/mol.112.081661
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  Hydrogen Sulfide as an Allosteric Modulator of ATP-Sensitive Potassium Channels in Colonic Inflammation

  Aravind R. Gade, Minho Kang and Hamid I. Akbarali

  Molecular Pharmacology January 2013, 83 (1) 294-306; DOI: https://doi.org/10.1124/mol.112.081596