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ArticleS

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  N-Methyl-D-Aspartic Acid Receptor Activation Downregulates Expression of δ Subunit-Containing GABA_A Receptors in Cultured Hippocampal Neurons

  Suchitra Joshi and Jaideep Kapur

  Molecular Pharmacology July 2013, 84 (1) 1-11; DOI: https://doi.org/10.1124/mol.112.084715
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  Small Molecule Inhibitors of ERCC1-XPF Protein-Protein Interaction Synergize Alkylating Agents in Cancer Cells

  Lars Petter Jordheim, Khaled H. Barakat, Laurence Heinrich-Balard, Eva-Laure Matera, Emeline Cros-Perrial, Karima Bouledrak, Rana El Sabeh, Rolando Perez-Pineiro, David S. Wishart, Richard Cohen, Jack Tuszynski and Charles Dumontet

  Molecular Pharmacology July 2013, 84 (1) 12-24; DOI: https://doi.org/10.1124/mol.112.082347
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  Pharmacological Inhibition of Platelet-Tumor Cell Cross-Talk Prevents Platelet-Induced Overexpression of Cyclooxygenase-2 in HT29 Human Colon Carcinoma Cells

  Melania Dovizio, Thorsten J. Maier, Sara Alberti, Luigia Di Francesco, Emanuela Marcantoni, Götz Münch, Constance M. John, Beatrix Suess, Alessandro Sgambato, Dieter Steinhilber and Paola Patrignani

  Molecular Pharmacology July 2013, 84 (1) 25-40; DOI: https://doi.org/10.1124/mol.113.084988
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  A Selective High-Affinity Antagonist of the P2Y₁₄ Receptor Inhibits UDP-Glucose–Stimulated Chemotaxis of Human Neutrophils

  Matthew O. Barrett, Juliana I. Sesma, Christopher B. Ball, P. Suresh Jayasekara, Kenneth A. Jacobson, Eduardo R. Lazarowski and T. Kendall Harden

  Molecular Pharmacology July 2013, 84 (1) 41-49; DOI: https://doi.org/10.1124/mol.113.085654
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  Activation of UTP-Sensitive P2Y₂ Receptor Induces the Expression of Cholinergic Genes in Cultured Cortical Neurons: A Signaling Cascade Triggered by Ca²⁺ Mobilization and Extracellular Regulated Kinase Phosphorylation

  Roy C. Y. Choi, Glanice K. Y. Chu, Nina L. Siow, Amanda W. Y. Yung, Lisa Y. Yung, Pinky S. C. Lee, Christopher C. W. Lo, Joseph Simon, Tina T. X. Dong, Eric A. Barnard and Karl W. K. Tsim

  Molecular Pharmacology July 2013, 84 (1) 50-61; DOI: https://doi.org/10.1124/mol.112.084160
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  Nrf2 Activators Attenuate the Progression of Nonalcoholic Steatohepatitis–Related Fibrosis in a Dietary Rat Model

  Rieko Shimozono, Yoshiji Asaoka, Yoshitaka Yoshizawa, Takumi Aoki, Hidetoshi Noda, Masateru Yamada, Mie Kaino and Hidenori Mochizuki

  Molecular Pharmacology July 2013, 84 (1) 62-70; DOI: https://doi.org/10.1124/mol.112.084269
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  Exploration of the Orthosteric/Allosteric Interface in Human M1 Muscarinic Receptors by Bitopic Fluorescent Ligands

  Sandrine B. Daval, Esther Kellenberger, Dominique Bonnet, Valérie Utard, Jean-Luc Galzi and Brigitte Ilien

  Molecular Pharmacology July 2013, 84 (1) 71-85; DOI: https://doi.org/10.1124/mol.113.085670
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  Antifungal Azoles: Structural Insights into Undesired Tight Binding to Cholesterol-Metabolizing CYP46A1

  Natalia Mast, Wenchao Zheng, C. David Stout and Irina A. Pikuleva

  Molecular Pharmacology July 2013, 84 (1) 86-94; DOI: https://doi.org/10.1124/mol.113.085902
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  Inhibition of the Proton-Coupled Folate Transporter (PCFT-SLC46A1) by Bicarbonate and Other Anions

  Rongbao Zhao, Michele Visentin, Sylvia O. Suadicani and I. David Goldman

  Molecular Pharmacology July 2013, 84 (1) 95-103; DOI: https://doi.org/10.1124/mol.113.085605
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  Rapamycin Allosterically Inhibits the Proteasome

  Pawel A. Osmulski and Maria Gaczynska

  Molecular Pharmacology July 2013, 84 (1) 104-113; DOI: https://doi.org/10.1124/mol.112.083873
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  Structural Determinants of Agonist Efficacy at the Glutamate Binding Site of N-Methyl-d-Aspartate Receptors

  Kasper B. Hansen, Nami Tajima, Rune Risgaard, Riley E. Perszyk, Lars Jørgensen, Katie M. Vance, Kevin K. Ogden, Rasmus P. Clausen, Hiro Furukawa and Stephen F. Traynelis

  Molecular Pharmacology July 2013, 84 (1) 114-127; DOI: https://doi.org/10.1124/mol.113.085803
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  The Nuclear Factor κB Family Member RelB Facilitates Apoptosis of Renal Epithelial Cells Caused by Cisplatin/Tumor Necrosis Factor α Synergy by Suppressing an Epithelial to Mesenchymal Transition–Like Phenotypic Switch

  Giulia Benedetti, Michiel Fokkelman, Kuan Yan, Lisa Fredriksson, Bram Herpers, John Meerman, Bob van de Water and Marjo de Graauw

  Molecular Pharmacology July 2013, 84 (1) 128-138; DOI: https://doi.org/10.1124/mol.112.084053
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  Three Ubiquitination Sites of Organic Anion Transporter-1 Synergistically Mediate Protein Kinase C–Dependent Endocytosis of the Transporter

  Shanshan Li, Qiang Zhang and Guofeng You

  Molecular Pharmacology July 2013, 84 (1) 139-146; DOI: https://doi.org/10.1124/mol.113.086769
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  Low Molecular Weight Fucoidan Improves Endoplasmic Reticulum Stress-Reduced Insulin Sensitivity through AMP-Activated Protein Kinase Activation in L6 Myotubes and Restores Lipid Homeostasis in a Mouse Model of Type 2 Diabetes

  Yong-Tae Jeong, Yong Deuk Kim, Young-Mi Jung, Dong-Chan Park, Dong-Sub Lee, Sae-Kwang Ku, Xian Li, Yue Lu, Guang Hsuan Chao, Keuk-Jun Kim, Jai-Youl Lee, Moon-Chang Baek, Wonku Kang, Seung-Lark Hwang and Hyeun Wook Chang

  Molecular Pharmacology July 2013, 84 (1) 147-157; DOI: https://doi.org/10.1124/mol.113.085100