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Molecular Pharmacology

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Table of Contents

September 01, 2013; Volume 84,Issue 3

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    Oral Benzo[a]pyrene: Understanding Pharmacokinetics, Detoxication, and Consequences—Cyp1 Knockout Mouse Lines as a Paradigm
    Daniel W. Nebert, Zhanquan Shi, Marina Gálvez-Peralta, Shigeyuki Uno and Nadine Dragin
    Molecular Pharmacology September 2013, 84 (3) 304-313; DOI: https://doi.org/10.1124/mol.113.086637

Articles

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    Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries
    Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten
    Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595
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    Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate
    Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera
    Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548
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    Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5
    Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde
    Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702
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    Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane
    Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert
    Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868
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    Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish
    Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman
    Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413
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    Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity
    Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz
    Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967
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    Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes
    Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal
    Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312
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    Novel Amino-Carbonitrile-Pyrazole Identified in a Small Molecule Screen Activates Wild-Type and ∆F508 Cystic Fibrosis Transmembrane Conductance Regulator in the Absence of a cAMP Agonist
    Wan Namkung, Jinhong Park, Yohan Seo and A. S. Verkman
    Molecular Pharmacology September 2013, 84 (3) 384-392; DOI: https://doi.org/10.1124/mol.113.086348
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    α4α6β2* Nicotinic Acetylcholine Receptor Activation on Ventral Tegmental Area Dopamine Neurons Is Sufficient to Stimulate a Depolarizing Conductance and Enhance Surface AMPA Receptor Function
    Staci E. Engle, Pei-Yu Shih, J. Michael McIntosh and Ryan M. Drenan
    Molecular Pharmacology September 2013, 84 (3) 393-406; DOI: https://doi.org/10.1124/mol.113.087346
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    Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation
    Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer
    Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835
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    Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface
    James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi
    Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080
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    Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M1 Muscarinic Acetylcholine Receptor
    Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos
    Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320
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    The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells
    Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius
    Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801
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    Specificity Determinants of CYP1B1 Estradiol Hydroxylation
    Clinton R. Nishida, Steven Everett and Paul R. Ortiz de Montellano
    Molecular Pharmacology September 2013, 84 (3) 451-458; DOI: https://doi.org/10.1124/mol.113.087700
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    Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents
    Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke
    Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462
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    Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing Gβγ Subunits in Human Embryonic Kidney 293T Cells
    Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya
    Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288

Erratum

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    Correction to “Protease-Activated Receptor (PAR) 1 and PAR4 Differentially Regulate Factor V Expression from Human Platelets”
    Molecular Pharmacology September 2013, 84 (3) 487; DOI: https://doi.org/10.1124/mol.113.09er13
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Molecular Pharmacology: 84 (3)
Molecular Pharmacology
Vol. 84, Issue 3
1 Sep 2013
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