Table of Contents

Articles

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  Selective Agonists and Antagonists of Formylpeptide Receptors: Duplex Flow Cytometry and Mixture-Based Positional Scanning Libraries

  Clemencia Pinilla, Bruce S. Edwards, Jon R. Appel, Tina Yates-Gibbins, Marc A. Giulianotti, Jose L. Medina-Franco, Susan M. Young, Radleigh G. Santos, Larry A. Sklar and Richard A. Houghten

  Molecular Pharmacology September 2013, 84 (3) 314-324; DOI: https://doi.org/10.1124/mol.113.086595
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  Mechanisms of Transient Receptor Potential Vanilloid 1 Activation and Sensitization by Allyl Isothiocyanate

  Maarten Gees, Yeranddy A. Alpizar, Brett Boonen, Alicia Sanchez, Wouter Everaerts, Andrei Segal, Fenqin Xue, Annelies Janssens, Grzegorz Owsianik, Bernd Nilius, Thomas Voets and Karel Talavera

  Molecular Pharmacology September 2013, 84 (3) 325-334; DOI: https://doi.org/10.1124/mol.113.085548
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  Extracellular Disulfide Bridges Serve Different Purposes in Two Homologous Chemokine Receptors, CCR1 and CCR5

  Pia C. Rummel, Stefanie Thiele, Lærke S. Hansen, Trine P. Petersen, Alexander H. Sparre-Ulrich, Trond Ulven and Mette M. Rosenkilde

  Molecular Pharmacology September 2013, 84 (3) 335-345; DOI: https://doi.org/10.1124/mol.113.086702
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  Segregation of Family A G Protein–Coupled Receptor Protomers in the Plasma Membrane

  Anthony Gavalas, Tien-Hung Lan, Qiuju Liu, Ivan R. Corrêa, Jonathan A. Javitch and Nevin A. Lambert

  Molecular Pharmacology September 2013, 84 (3) 346-352; DOI: https://doi.org/10.1124/mol.113.086868
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  Sox9b Is Required for Epicardium Formation and Plays a Role in TCDD-Induced Heart Malformation in Zebrafish

  Peter Hofsteen, Jessica Plavicki, Shaina D. Johnson, Richard E. Peterson and Warren Heideman

  Molecular Pharmacology September 2013, 84 (3) 353-360; DOI: https://doi.org/10.1124/mol.113.086413
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  Human Immunodeficiency Virus Protease Inhibitors Interact with ATP Binding Cassette Transporter 4/Multidrug Resistance Protein 4: A Basis for Unanticipated Enhanced Cytotoxicity

  Yu Fukuda, Kazumasa Takenaka, Alex Sparreboom, Satish B. Cheepala, Chung-Pu Wu, Sean Ekins, Suresh V. Ambudkar and John D. Schuetz

  Molecular Pharmacology September 2013, 84 (3) 361-371; DOI: https://doi.org/10.1124/mol.113.086967
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  Connective Tissue Growth Factor/CCN2 Attenuates β-Adrenergic Receptor Responsiveness and Cardiotoxicity by Induction of G Protein–Coupled Receptor Kinase-5 in Cardiomyocytes

  Jørgen Gravning, M. Shakil Ahmed, Eirik Qvigstad, Kurt Krobert, Thor Edvardsen, Ingvild Tronstad Moe, Else Marie V. Hagelin, Julia Sagave, Guro Valen, Finn Olav Levy, Jan-Bjørn Osnes, Tor Skomedal and Håvard Attramadal

  Molecular Pharmacology September 2013, 84 (3) 372-383; DOI: https://doi.org/10.1124/mol.113.087312
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  Novel Amino-Carbonitrile-Pyrazole Identified in a Small Molecule Screen Activates Wild-Type and ∆F508 Cystic Fibrosis Transmembrane Conductance Regulator in the Absence of a cAMP Agonist

  Wan Namkung, Jinhong Park, Yohan Seo and A. S. Verkman

  Molecular Pharmacology September 2013, 84 (3) 384-392; DOI: https://doi.org/10.1124/mol.113.086348
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  α4α6β2* Nicotinic Acetylcholine Receptor Activation on Ventral Tegmental Area Dopamine Neurons Is Sufficient to Stimulate a Depolarizing Conductance and Enhance Surface AMPA Receptor Function

  Staci E. Engle, Pei-Yu Shih, J. Michael McIntosh and Ryan M. Drenan

  Molecular Pharmacology September 2013, 84 (3) 393-406; DOI: https://doi.org/10.1124/mol.113.087346
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  Potent Inhibition of Aldehyde Dehydrogenase-2 by Diphenyleneiodonium: Focus on Nitroglycerin Bioactivation

  Regina Neubauer, Andrea Neubauer, Gerald Wölkart, Christine Schwarzenegger, Barbara Lang, Kurt Schmidt, Michael Russwurm, Doris Koesling, Antonius C. F. Gorren, Astrid Schrammel and Bernd Mayer

  Molecular Pharmacology September 2013, 84 (3) 407-414; DOI: https://doi.org/10.1124/mol.113.086835
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  Hits of a High-Throughput Screen Identify the Hydrophobic Pocket of Autotaxin/Lysophospholipase D As an Inhibitory Surface

  James I. Fells, Sue Chin Lee, Yuko Fujiwara, Derek D. Norman, Keng Gat Lim, Ryoko Tsukahara, Jianxiong Liu, Renukadevi Patil, Duane D. Miller, R. Jason Kirby, Sandra Nelson, William Seibel, Ruben Papoian, Abby L. Parrill, Daniel L. Baker, Robert Bittman and Gabor Tigyi

  Molecular Pharmacology September 2013, 84 (3) 415-424; DOI: https://doi.org/10.1124/mol.113.087080
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  Reverse Engineering of the Selective Agonist TBPB Unveils Both Orthosteric and Allosteric Modes of Action at the M₁ Muscarinic Acetylcholine Receptor

  Peter Keov, Celine Valant, Shane M. Devine, J. Robert Lane, Peter J. Scammells, Patrick M. Sexton and Arthur Christopoulos

  Molecular Pharmacology September 2013, 84 (3) 425-437; DOI: https://doi.org/10.1124/mol.113.087320
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  The Role of Human Equilibrative Nucleoside Transporter 1 on the Cellular Transport of the DNA Methyltransferase Inhibitors 5-Azacytidine and CP-4200 in Human Leukemia Cells

  Johanna Hummel-Eisenbeiss, Antje Hascher, Petter-Arnt Hals, Marit Liland Sandvold, Carsten Müller-Tidow, Frank Lyko and Maria Rius

  Molecular Pharmacology September 2013, 84 (3) 438-450; DOI: https://doi.org/10.1124/mol.113.086801
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  Specificity Determinants of CYP1B1 Estradiol Hydroxylation

  Clinton R. Nishida, Steven Everett and Paul R. Ortiz de Montellano

  Molecular Pharmacology September 2013, 84 (3) 451-458; DOI: https://doi.org/10.1124/mol.113.087700
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  Multiple Modes of α7 nAChR Noncompetitive Antagonism of Control Agonist-Evoked and Allosterically Enhanced Currents

  Can Peng, Matthew R. Kimbrell, Chengju Tian, Thomas F. Pack, Peter A. Crooks, E. Kim Fifer and Roger L. Papke

  Molecular Pharmacology September 2013, 84 (3) 459-475; DOI: https://doi.org/10.1124/mol.113.086462
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  Prostaglandin E Receptor EP1 Forms a Complex with Dopamine D1 Receptor and Directs D1-Induced cAMP Production to Adenylyl Cyclase 7 through Mobilizing G_βγ Subunits in Human Embryonic Kidney 293T Cells

  Aliza T. Ehrlich, Tomoyuki Furuyashiki, Shiho Kitaoka, Akira Kakizuka and Shuh Narumiya

  Molecular Pharmacology September 2013, 84 (3) 476-486; DOI: https://doi.org/10.1124/mol.113.087288